Studies towards the conception of new selective PPARβ/δ ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 17, 2006, Pages 4528-4532

  Ekambomé Basséne, Carine ^a   Suzenet, Franck ^a   Hennuyer, Nathalie ^b   Staels, Bart ^b   Caignard, Daniel Henri ^c   Dacquet, Catherine ^d   Renard, Pierre ^d   Guillaumet, Gérald ^a  

^a Université d'Orléans   (France)

^b INSTITUT PASTEUR DE LILLE   (France)

^c INSTITUT DE RECHERCHES SERVIER   (France)

^d INSTITUT DE RECHERCHES SERVIER   (France)

Author keywords

Nuclear receptor; PPAR ; Pyridine

Indexed keywords

4 [4 [3 (4 ACETYL 3 HYDROXY 2 PROPYLPHENOXY)PROPOXY]PHENOXY]ACETIC ACID; [2 METHYL 4 [4 METHYL 2 (4 TRIFLUOROMETHYLPHENYL) 5 THIAZOLYLMETHYLTHIO]PHENOXY]ACETIC ACID; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR AGONIST; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR DELTA; PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG ACTIVITY; DRUG SELECTIVITY; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANIMALS; CERCOPITHECUS AETHIOPS; COS CELLS; HUMANS; LIGANDS; MOLECULAR STRUCTURE; PPAR DELTA; PPAR-BETA; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33746196476     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.06.028     Document Type: Article

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