Highly efficient microwave assisted α-trichlorination reaction of α-methylated nitrogen containing heterocycles

Tetrahedron

Volumn 62, Issue 34, 2006, Pages 8173-8176

  Verhaeghe, Pierre ^a   Rathelot, Pascal ^a   Gellis, Armand ^a   Rault, Sylvain ^b   Vanelle, Patrice ^a  

^a CNRS   (France)

^b CENTRE D ETUDES ET DE RECHERCHE SUR LE MÉDICAMENT DE NORMANDIE   (France)

Author keywords

Ionic polychlorination; Microwave assisted reactions; Nitrogen containing heterocycles

Indexed keywords

CHLORINE; METHYL GROUP; NITROGEN; OXYGEN; PHOSPHORUS 31;

ARTICLE; CHLORINATION; FLUORINATION; METHODOLOGY; METHYLATION; NITRATION; PRIORITY JOURNAL; REACTION ANALYSIS; STRUCTURE ANALYSIS; TECHNOLOGY;

EID: 33745727399     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tet.2006.05.081     Document Type: Article

References (15)

1. Singh B., and Lesher G. J. Heterocycl. Chem. 20 (1983) 491
2. Beer R.H., Jimenez J., and Drago R.S. J. Org. Chem. 58 (1993) 1746
3. In: Vanelle P. (Ed). Electron Transfer Reactions in Organic Synthesis (2002), Research Signpost, Trivandrum
4. Vanelle P., Benakli K., Giraud L., and Crozet M.P. Synlett (1999) 801
5. Newkome G.R., Kiefer G.E., Xia Y.J., and Gupta V.K. Synthesis (1984) 676
6. Mizuno Y., Adachi K., and Kanda S. J. Pharm. Soc. Japan 72 (1952) 1263
7. Chupp J.P., Grabiak R.C., Leschinsky K.L., and Neumann T.L. Synthesis (1986) 224
8. Kato T., Hayashi H., and Anzai T. Yakugaku Zasshi 87 (1967) 387
9. Kato T., Katagiri N., and Wagai A. Tetrahedron 34 (1978) 3445
10. Kato T., Katagiri N., and Wagai A. Chem. Pharm. Bull. 29 (1981) 1069
11. Boufatah N., Gellis A., Maldonado J., and Vanelle P. Tetrahedron 60 (2004) 9131
12. Dehoff L.H. J. Prakt. Chem. 42 (1890) 352
13. Smith R.F., and Kent R.A. J. Org. Chem. 30 (1964) 1312
14. Cartwright D., Ferguson J.R., Giannopoulos T., Varvounis G., and Wakefield B.J. J. Chem. Soc., Perkin Trans. 1 (1995) 2595
15. Holan G., Samuel E.L., Ennis B.C., and Hinde R.W. J. Chem. Soc. C (1967) 20