Schild (apparent pA2) analysis of a κ-opioid antagonist in Planaria

European Journal of Pharmacology

Volumn 540, Issue 1-3, 2006, Pages 200-201

  Raffa, Robert B ^a,b   Baron, David A ^a   Tallarida, Ronald J ^b  

^a TEMPLE UNIVERSITY SCHOOL OF PHARMACY   (United States)

^b TEMPLE UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

opioid receptor; Planaria; Schild (pA2) analysis

Indexed keywords

3,4 DICHLORO N METHYL N [2 (1 PYRROLIDINYL)CYCLOHEXYL]BENZENEACETAMIDE METHANESULFONATE; KAPPA OPIATE RECEPTOR; KAPPA OPIATE RECEPTOR ANTAGONIST; NORBINALTORPHIMINE; 3,4 DICHLORO N METHYL N [2 (1 PYRROLIDINYL)CYCLOHEXYL]BENZENEACETAMIDE; ANALGESIC AGENT; DRUG DERIVATIVE; NALTREXONE; NARCOTIC ANTAGONIST;

ANALYTIC METHOD; ARTICLE; DRUG ANTAGONISM; DRUG SELECTIVITY; IN VIVO STUDY; MATHEMATICAL ANALYSIS; NONHUMAN; PRIORITY JOURNAL; QUANTITATIVE ANALYSIS; SCHILD ANALYSIS; TURBELLARIA; ALGORITHM; ANIMAL; DOSE RESPONSE; DRUG EFFECT; LOCOMOTION; PHYSIOLOGY; REGRESSION ANALYSIS;

3,4-DICHLORO-N-METHYL-N-(2-(1-PYRROLIDINYL)-CYCLOHEXYL)-BENZENEACETAMIDE, (TRANS)-ISOMER; ALGORITHMS; ANALGESICS, NON-NARCOTIC; ANIMALS; DOSE-RESPONSE RELATIONSHIP, DRUG; LOCOMOTION; NALTREXONE; NARCOTIC ANTAGONISTS; PLANARIANS; RECEPTORS, OPIOID, KAPPA; REGRESSION ANALYSIS;

EID: 33745007055     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2006.04.027     Document Type: Article

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