-
2
-
-
0024404979
-
-
Ife R.J., Dyke C.A., Keeling D.J., Meenan E., Meeson M.L., Parsons M.E., Price C.A., Theobald C.J., and Underwood A.H. J. Med. Chem. 32 (1989) 1970
-
(1989)
J. Med. Chem.
, vol.32
, pp. 1970
-
-
Ife, R.J.1
Dyke, C.A.2
Keeling, D.J.3
Meenan, E.4
Meeson, M.L.5
Parsons, M.E.6
Price, C.A.7
Theobald, C.J.8
Underwood, A.H.9
-
5
-
-
37049073467
-
-
Guerrera F., Salerno L., Lamartina L., and Spinelli D. J. Chem. Soc., Perkin Trans. 1 (1995) 1243
-
(1995)
J. Chem. Soc., Perkin Trans. 1
, pp. 1243
-
-
Guerrera, F.1
Salerno, L.2
Lamartina, L.3
Spinelli, D.4
-
8
-
-
37049066671
-
-
Barrow P., Bullen J.V., Murphy A., Ridd D., T.J.H., and Sabek O. J. Chem. Soc., Chem. Commun. (1986) 1649
-
(1986)
J. Chem. Soc., Chem. Commun.
, pp. 1649
-
-
Barrow, P.1
Bullen, J.V.2
Murphy, A.3
Ridd D.,, T.J.H.4
Sabek, O.5
-
13
-
-
33744502543
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-
note
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We have tried different conditions for the deoxygenation of 1, but the results are complicated due to the replacement of nitro-group by different nucleophiles (Cl, Br, et al.) and reduction of the nitro-group. The reaction a (Scheme 1) affords the desired product (2) in 11% yield along with 80% 3,4-dibromopyridine, which are difficult to purify by column.
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-
-
-
18
-
-
0031772124
-
-
Nakagawa H., Higuchi T., Kikuchi K., Urano Y., and Nagano T. Chem. Pharm. Bull. 46 (1998) 1656
-
(1998)
Chem. Pharm. Bull.
, vol.46
, pp. 1656
-
-
Nakagawa, H.1
Higuchi, T.2
Kikuchi, K.3
Urano, Y.4
Nagano, T.5
-
22
-
-
33744487071
-
-
Unpublished results.
-
-
-
-
30
-
-
0028783851
-
-
Kelley J.L., Koble C.S., Davis R.G., McLean E.W., Soroko F.E., and Coopert B.R. J. Med. Chem. 38 (1995) 4131
-
(1995)
J. Med. Chem.
, vol.38
, pp. 4131
-
-
Kelley, J.L.1
Koble, C.S.2
Davis, R.G.3
McLean, E.W.4
Soroko, F.E.5
Coopert, B.R.6
-
31
-
-
0028273009
-
-
Romero D.L., Merge R.D., Biles C., Berrios-PBna N., May P.D., Palmer J.R., Johnson P.D., Smith H.W., Busso M., Tan C., Voorman R.L., Reusse F., Althaus I.W., Downey W.M., So A.G., Resnick L., Tarpley W.G., and Aristoff P.A. J. Med. Chem. 37 (1994) 999
-
(1994)
J. Med. Chem.
, vol.37
, pp. 999
-
-
Romero, D.L.1
Merge, R.D.2
Biles, C.3
Berrios-PBna, N.4
May, P.D.5
Palmer, J.R.6
Johnson, P.D.7
Smith, H.W.8
Busso, M.9
Tan, C.10
Voorman, R.L.11
Reusse, F.12
Althaus, I.W.13
Downey, W.M.14
So, A.G.15
Resnick, L.16
Tarpley, W.G.17
Aristoff, P.A.18
-
33
-
-
0030739747
-
-
Spinelli D., Zanirato P., Miceli E.D., Lamartina L., and Guerrera F. J. Org. Chem. 62 (1997) 4921
-
(1997)
J. Org. Chem.
, vol.62
, pp. 4921
-
-
Spinelli, D.1
Zanirato, P.2
Miceli, E.D.3
Lamartina, L.4
Guerrera, F.5
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