The first and reliable synthesis of thieno[2,3-e][1,2,4]-triazolo[1,5-c]pyrimidin-5(6H)-ones via their [4,3-c] compounds by dimroth rearrangement

Heterocycles

Volumn 65, Issue 11, 2005, Pages 2683-2692

  Nagamatsu, Tomohisa ^a   Ahmed, Shoeb ^a  

^a OKAYAMA UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 33646856213     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/COM-05-10518     Document Type: Article

References (24)

1. Nagamatsu T., Yamasaki H., Akiyama T., Hara S., Mori K., and Kusakabe H. Synthesis (1999) 655
2. Nagamatsu T., Yamasaki H., Fujita T., Endo K., and Machida H. J. Chem. Soc., Perkin Trans. 1 (1999) 3117
3. Nagamatsu T., and Fujita T. Chem. Commun. (1999) 1461
4. Nagamatsu T., Fujita T., and Endo K. J. Chem. Soc., Perkin Trans. 1 (2000) 33
5. R.W. R., Wyngaarden J.B., Hitching G.H., Elion G.B., and Silberman H.R. Trans. Assoc. Am. Physicians 76 (1963) 126
6. Yü T.F., and Gutman A.B. Am. J. Med. 37 (1964) 885
7. Klinenberg J.R., Goldfinger S.E., and Seegmiller J.E. Ann, Intern. Med. 62 (1965) 639
8. Young J.L., Boswell R.B., and Nies A.S. Arch. Intern. Med. 134 (1974) 553
9. Hande K.R., Noone R.M., and Stone W.J. Am. J. Med. 76 (1984) 47
10. Elion G.B. Ann. Rheumat. Dis. 25 (1966) 608
11. Duggan D.E., Noll R.M., Baer J.E., Novello F.C., and Baldwin J.J. J. Med. Chem. 18 (1975) 900
12. Wortmann R.L., Ridolfo A.S., Lightfoot Jr. R.W., and Fox I.H. J. Rheumatol. 12 (1985) 540
13. Bindoli A., Valente M., and Cavallini L. Pharmacol. Res. Commun. 17 (1985) 831
14. Spector T., Hall W.W., Porter D.J., Lambe C.U., Nelson D.J., and Krenitsky T.A. Biochem. Pharmacol. 38 (1989) 4315
15. Sato S., Tatsumi K., and Nishino T. Purine and Pyrimidine Metabolism in Man VII, Part A: Chemotherapy, ATP Depletion and Gout. In: Harkness R.A., Elion G.B., and Zöllner N. (Eds) (1991), Plenum Press, New York 135-138
16. Osada Y., Tsuchimoto M., Fukushima H., Takahashi K., Kondo S., Hasegawa M., and Komoriya K. Eur. J. Pharmacol. 241 (1993) 183
17. Biagi G., Giorgi I., Livi O., Scartoni V., Tonetti I., and Costantino L. Farmacol. 50 (1995) 257
18. Elion G.B., Callahan S., Nathan H., Bieber S., Rundles R.W., and Hitchings G.H. Biochem. Pharmacol. 12 (1963) 85
19. Nagamatsu T., and Fujita T. Heterocycles 57 (2002) 631
20. Brown D.J., and Nagamatsu T. Aust. J. Chem. 31 (1978) 2505
21. Brown D.J., and Nagamatsu T. Aust. J. Chem. 32 (1979) 1585
22. Brown D.J., and Shinozuka K. Aust. J. Chem. 33 (1980) 1147
23. J. L. Primeau, and L. M. Garrick, US Patent 5, 187, 168/1993
24. Chem. Abstr. 119 (1993) 139256