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Volumn 1, Issue 3, 2006, Pages 303-305

Tuning wasp toxin structure for nicotinic receptor antagonism: Cyclohexylalanine-containing analogues as potent and voltage-dependent blockers

(7) Olsen, Christian A a Mellor, Ian R b Wellendorph, Petrine a Usherwood, Peter N R b Witt, Matthias c Franzyk, Henrik a Jaroszewski, Jerzy W a

a UNIVERSITY OF COPENHAGEN (Denmark)

b UNIVERSITY OF NOTTINGHAM (United Kingdom)

c BRUKER DALTONIK GMBH (Germany)

Author keywords

Acetylcholine receptors; Ion channels; Natural products; Polyamine toxins; Solid phase synthesis

Indexed keywords

CYCLOHEXYLALANINE; DELTA-PHILANTHOTOXIN; DRUG DERIVATIVE; NICOTINIC RECEPTOR; NICOTINIC RECEPTOR BLOCKING AGENT; PHENYLALANINE; PHILANTHOTOXIN; POLYAMINE; WASP VENOM;

ARTICLE; CHANNEL GATING; CHEMISTRY; DRUG EFFECT; HUMAN;

HUMANS; ION CHANNEL GATING; NICOTINIC ANTAGONISTS; PHENYLALANINE; POLYAMINES; RECEPTORS, NICOTINIC; WASP VENOMS;

EID: 33646473365 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200500067 Document Type: Article

Times cited : (13)

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