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Volumn 95, Issue 4, 2006, Pages 917-928

Identification, preparation, and characterization of several polymorphs and solvates of terazosin hydrochloride

Author keywords

Dehydrate; Methanolate; Molecular modeling; Polymorphs; Terazosin; X ray diffraction

Indexed keywords

TERAZOSIN;

EID: 33645999665     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.20425     Document Type: Article
Times cited : (17)

References (35)
  • 1
    • 0024512048 scopus 로고
    • Alpha-blocking potencies of antihypertensive agents (prazosin, teraazosin, bunazosin, SGB-1534 and ketanserin) with quinazoline or quinazolinedione as assassed by radioligand binding assay methods in rat brain
    • Tsuchihashi H, Nagatomo T. 1989. Alpha-blocking potencies of antihypertensive agents (prazosin, teraazosin, bunazosin, SGB-1534 and ketanserin) with quinazoline or quinazolinedione as assassed by radioligand binding assay methods in rat brain. J Pharmacobio Dyn 12:170-174.
    • (1989) J Pharmacobio Dyn , vol.12 , pp. 170-174
    • Tsuchihashi, H.1    Nagatomo, T.2
  • 3
    • 0022007032 scopus 로고
    • Anti-hypertensive effectiveness of terazosin: A new long acting alpha adrenergic inhibitor
    • Chrysant S, Bal I, Johnson B, McPherson M. 1985. Anti-hypertensive effectiveness of terazosin: A new long acting alpha adrenergic inhibitor. Clin Cardiol 8:486-489.
    • (1985) Clin Cardiol , vol.8 , pp. 486-489
    • Chrysant, S.1    Bal, I.2    Johnson, B.3    McPherson, M.4
  • 8
    • 0029939081 scopus 로고    scopus 로고
    • The Hytrin Community Assessment Trial Study: A one year study of terazosin versus placebo in the treatment of men with symptomatic benign prostatic hyperplasia
    • Roehrborn CG, Oesterling JE, Auerbach S, Kaplan SA, Lloyd LK, Milam DF, Padley RJ. 1996. The Hytrin Community Assessment Trial Study: A one year study of terazosin versus placebo in the treatment of men with symptomatic benign prostatic hyperplasia. Urology 47:159-168.
    • (1996) Urology , vol.47 , pp. 159-168
    • Roehrborn, C.G.1    Oesterling, J.E.2    Auerbach, S.3    Kaplan, S.A.4    Lloyd, L.K.5    Milam, D.F.6    Padley, R.J.7
  • 12
    • 1042298894 scopus 로고    scopus 로고
    • A timely re-examination of drug polymorphism in pharmaceutical development and regulation
    • Grant DW, Byrn SR. 2004. A timely re-examination of drug polymorphism in pharmaceutical development and regulation, Adv Drug Deliv Rev 56:237-239.
    • (2004) Adv Drug Deliv Rev , vol.56 , pp. 237-239
    • Grant, D.W.1    Byrn, S.R.2
  • 13
    • 0014559313 scopus 로고
    • Pharmaceutical applications of polymorphism
    • Haleblian J, McCrone W. 1969. Pharmaceutical applications of polymorphism. J Pharm Sci 58:911-929.
    • (1969) J Pharm Sci , vol.58 , pp. 911-929
    • Haleblian, J.1    McCrone, W.2
  • 15
    • 0343471485 scopus 로고    scopus 로고
    • Characterization of famotidine polymorphs, inter
    • Hassan M, et al. 1997. Characterization of famotidine polymorphs, inter. J Pharmaceutics 149:227-232.
    • (1997) J Pharmaceutics , vol.149 , pp. 227-232
    • Hassan, M.1
  • 16
    • 85030606047 scopus 로고    scopus 로고
    • 1977. Antihypertensive agents. U.S. Patent 4112097
    • Winn M, Kyncl J, et al. 1977. Antihypertensive agents. U.S. Patent 4112097
    • Winn, M.1    Kyncl, J.2
  • 17
    • 85030609695 scopus 로고    scopus 로고
    • 1994. Terazosin polymorph and pharmaceutical composition. U.S.Patent 5294615
    • Meyer G, Bauer J. 1994. Terazosin polymorph and pharmaceutical composition. U.S.Patent 5294615.
    • Meyer, G.1    Bauer, J.2
  • 18
    • 85030604416 scopus 로고    scopus 로고
    • 1994. Terazosin polymorph and pharmaceutical composition. U.S. Patent 5362730
    • Bauer J, Morley J. 1994. Terazosin polymorph and pharmaceutical composition. U.S. Patent 5362730.
    • Bauer, J.1    Morley, J.2
  • 19
    • 85030609132 scopus 로고    scopus 로고
    • 1995. Terazosin monohydrochloride and processes and intermediates for its production. U.S. Patent 5412095
    • Morley J, Bauer J. 1995. Terazosin monohydrochloride and processes and intermediates for its production. U.S. Patent 5412095.
    • Morley, J.1    Bauer, J.2
  • 20
    • 85030606016 scopus 로고    scopus 로고
    • 1996. process and intermediate for the preparation of terazosin hydrochloride dihydrate. U.S. Patent 5,504,207
    • Mannino A, Henry R, et al. 1996. process and intermediate for the preparation of terazosin hydrochloride dihydrate. U.S. Patent 5,504,207.
    • Mannino, A.1    Henry, R.2
  • 21
    • 33645969750 scopus 로고
    • Terazosin crystalline polymorph and pharmaceutical compositions thereof. U.S. Patent 5,587,377
    • Patel M, et al. 1995. Terazosin crystalline polymorph and pharmaceutical compositions thereof. U.S. Patent 5,587,377.
    • (1995)
    • Patel, M.1
  • 22
    • 0018618861 scopus 로고
    • On the polymorphism of pharmaceuticals and other molecular crystals II
    • Burger A, Ramberger R. 1979. On the polymorphism of pharmaceuticals and other molecular crystals II. Mikrochim Acta (Wien) 11:273-316.
    • (1979) Mikrochim Acta (Wien) , vol.11 , pp. 273-316
    • Burger, A.1    Ramberger, R.2
  • 23
  • 24
    • 0036253941 scopus 로고    scopus 로고
    • X-ray powder diffraction of pharmaceutical materials
    • Brittain HG. 2002. X-ray powder diffraction of pharmaceutical materials. Am Pharm Rev 5:74-76, 78, 80.
    • (2002) Am Pharm Rev , vol.5 , pp. 74-76
    • Brittain, H.G.1
  • 25
    • 0242322069 scopus 로고    scopus 로고
    • Comparison of the four anhydrous polymorphs of carbamazepine and the crystal structure of form I
    • Grzesiak AL, Lang M, Kim K, Matzger AJ. 2003. Comparison of the four anhydrous polymorphs of carbamazepine and the crystal structure of form I. J Pharm Sci 92:2260-2271.
    • (2003) J Pharm Sci , vol.92 , pp. 2260-2271
    • Grzesiak, A.L.1    Lang, M.2    Kim, K.3    Matzger, A.J.4
  • 26
    • 0034820059 scopus 로고    scopus 로고
    • Estimating the relative stability of polymorphs and hydrates from heats of solution and solubility data
    • Gu CH, Grant DJW. 2001. Estimating the relative stability of polymorphs and hydrates from heats of solution and solubility data. J Pharm Sci 90:1277-1287.
    • (2001) J Pharm Sci , vol.90 , pp. 1277-1287
    • Gu, C.H.1    Grant, D.J.W.2
  • 27
    • 20344362958 scopus 로고    scopus 로고
    • Single crystal and powder diffraction characterization of three polymorphic forms of acitretin
    • Malpezzi L, Magnone GA, Masciocchi N, Sironi A. 2005. Single crystal and powder diffraction characterization of three polymorphic forms of acitretin. J Pharm Sci 94:1067-1078.
    • (2005) J Pharm Sci , vol.94 , pp. 1067-1078
    • Malpezzi, L.1    Magnone, G.A.2    Masciocchi, N.3    Sironi, A.4
  • 28
    • 0037369922 scopus 로고    scopus 로고
    • Solid-state nuclear magnetic resonance spectroscopy-Pharmaceutical applications
    • Tishmack PA, Bugay DE, Byrn SR. 2003. Solid-state nuclear magnetic resonance spectroscopy-Pharmaceutical applications. J Pharm Sci 92:441-474.
    • (2003) J Pharm Sci , vol.92 , pp. 441-474
    • Tishmack, P.A.1    Bugay, D.E.2    Byrn, S.R.3
  • 29
    • 0030724408 scopus 로고    scopus 로고
    • Polymorphism in anhydrous theophylline - Implications on the dissolution rate of theophylline tablets
    • Phadnis NV, et al. 1997. Polymorphism in anhydrous theophylline- Implications on the dissolution rate of theophylline tablets. J Pharm Sci 86:1256-1263.
    • (1997) J Pharm Sci , vol.86 , pp. 1256-1263
    • Phadnis, N.V.1
  • 31
    • 0032949617 scopus 로고    scopus 로고
    • Demonstration of the terms enantiotropy and monotropy in polymorphism research exemplified by flurbiprofen
    • Kuhnert-Brandstatter M. 1999. Demonstration of the terms enantiotropy and monotropy in polymorphism research exemplified by flurbiprofen. J Pharm Sci 88:103-108.
    • (1999) J Pharm Sci , vol.88 , pp. 103-108
    • Kuhnert-Brandstatter, M.1
  • 32
    • 0030230960 scopus 로고    scopus 로고
    • Ab initio prediction of polymorphs
    • Leusen FJJ. 1996. Ab initio prediction of polymorphs. J Crystal Growth 166:900-903.
    • (1996) J Crystal Growth , vol.166 , pp. 900-903
    • Leusen, F.J.J.1
  • 33
    • 0032343232 scopus 로고    scopus 로고
    • Computer simulation to predict possible crystal polymorphs
    • Verwer P, Leusen FJJ. 1998. Computer simulation to predict possible crystal polymorphs. Rev Comp Chem 12:327-365.
    • (1998) Rev Comp Chem , vol.12 , pp. 327-365
    • Verwer, P.1    Leusen, F.J.J.2
  • 34
    • 9144240095 scopus 로고
    • DREIDING: A generic force field for molecular simulations
    • Mayo SL, Olafson BD, Goddard WA, III. 1990. DREIDING: A generic force field for molecular simulations. J Phys Chem 94:8897-8909.
    • (1990) J Phys Chem , vol.94 , pp. 8897-8909
    • Mayo, S.L.1    Olafson, B.D.2    Goddard III, W.A.3
  • 35
    • 0002211129 scopus 로고
    • A profile refinement method for nuclear and magnetic structures
    • Rietveld HM. 1969. A profile refinement method for nuclear and magnetic structures. J Appl Crystallogr 2:65-71.
    • (1969) J Appl Crystallogr , vol.2 , pp. 65-71
    • Rietveld, H.M.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.