Synthesis and liposome encapsulation of a novel 18F-conjugate of ω-conotoxin GVIA for the potential imaging of N-type Ca2+ channels in the brain by positron emission tomography

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 49, Issue 3, 2006, Pages 269-283

  Azarian, Vahe ^a   Gangloff, Anne ^a   Seimbille, Yann ^a   Delaloye, Sibylle ^a   Czernin, Johannes ^a   Phelps, Michael E ^a   Silverman, Daniel H S ^a,b  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b MC694215   (United States)

Author keywords

Fluorine 18; Liposome; Peptide labeling; PET brain imaging; conotoxin GVIA

Indexed keywords

AMINO ACIDS; BRAIN MAPPING; FLUORINE; LIPOSOMES; MASS SPECTROMETRY; POSITRON EMISSION TOMOGRAPHY; POSITRONS;

BRAIN IMAGING; CA 2+; CONOTOXINS; FLUORINE-18; IN-VIVO; LABELINGS; PEPTIDE LABELING; PET BRAIN IMAGING; POTENTIAL IMAGING; Ω-CONOTOXIN GVIA;

BINDING ENERGY;

CALCIUM CHANNEL N TYPE; FLUORINE 18; N HYDROXYSUCCINIMIDYL 4 FLUOROBENZOATE F 18; OMEGA CONOTOXIN GVIA; UNCLASSIFIED DRUG;

ARTICLE; BLOOD BRAIN BARRIER; COLORIMETRY; DRUG STRUCTURE; DRUG SYNTHESIS; MATRIX ASSISTED LASER DESORPTION IONIZATION TIME OF FLIGHT MASS SPECTROMETRY; NEUROIMAGING; POSITRON EMISSION TOMOGRAPHY; RADIOCHEMISTRY;

EID: 33645791268     PISSN: 03624803     EISSN: 10991344     Source Type: Journal    
DOI: 10.1002/jlcr.1029     Document Type: Article

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