Isomerization-free sulfonylation and its application in the synthesis of PHA-565272A

Organic Process Research and Development

Volumn 10, Issue 2, 2006, Pages 334-338

  Fleck, Thomas J ^a   Chen, Jiong Jack ^a,b   Lu, Cuong V ^a   Hanson, Kari J ^a  

^a PFIZER INC   (United States)

^b GLAXOSMITHKLINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 33645547306     PISSN: 10836160     EISSN: None     Source Type: Journal    
DOI: 10.1021/op050208a     Document Type: Article

References (11)

1. Fu, J.-M. In PCT Intl WO 03011284, 2003.
2. Hugel, H. M.; Kennaway, D. J. Org. Prep. Proced. Int. 1995, 27, 1-31.
3. Wagaw, S.; Yang, B. H.; Buchwald, S. L. J. Am. Chem. Soc. 1999, 121, 10251-10263.
4. Hartwig, J. F. Angew. Chem., Int. Ed. 1998, 37, 2090-2093.
5. Dowdy, D.; Gore, P. H.; Waters, D. N. J. Chem. Soc., Perkin Trans. 2 1991, 1149-1159.
6. Pivsa-Art, S.; Okuro, K.; Miura, M.; Murata, S.; Nomura, M. J. Chem. Soc., Perkin Trans, 1 1994, 1703-1707.
7. Yoshii, Y.; Ito, A.; Manabe, O. Nippon Kagaku Kaishi 1973, 2395-2397.
8. Chen, J. J.; Fleck, T. J.; Lu, C. V.; Hanson, K. J. 224th ACS National Meeting, August 18-22, Boston, MA; American Chemical Society: Washington, DC, 2002.
9. Medina, F.; Manjarrez, A. Tetrahedron 1964, 20, 1807-10.
10. Hughes, D. L. Org. Prep. Proced. Int. 1993, 25, 607-32.
11. Hyatt, J. A.; White, A. W. Synthesis 1984, 214-7.