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33645417985
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US Patent Appl. 2003/114517, 2003
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A Scifinder search based on substructure A revealed more than 90 patents claiming bioactivities of cyclosulfonamide derivatives. See: (a) Greenlee, W. J.; Huang, Y.; Kelly, J. M.; McCombie, S. W.; Stamford, A. W.; Wu, Y. US Patent Appl. 2003/114517, 2003.
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Greenlee, W.J.1
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(b) Miller, M. W.; Scott, J. D. PCT Int. Appl. WO 2004/056770, 2004.
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(c) Paliwal, S.; Reichard, G. A.; Wang, C.; Xiao, D.; Tsui, H.-C.; Shih, N.-Y.; Arredondo, J. D.; Wrobleski, M. L.; Palani, A. PCT Int. Appl. WO 2003/051840, 2003.
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(f) Glunz, P. W.; Bisacchi, G. S.; Morton, G. C.; Holubec, A. A.; Priestley, E. S.; Zhang, X.; Treuner, U. D. PCT Int. Appl. WO 2004/072101, 2004.
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(g) Walter, R.; Heckel, A.; Roth, G. J.; Kley, J.; Schnapp, G.; Lenter, M.; Van Meel, J. C. A.; Spevak, W.; Weyer-Czernilofsky, U. PCT Int. Appl. WO 2002/36564, 2002.
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(h) Zhu, H. Y.; Njoroge, F. G.; Cooper, A. B.; Guzi, T.; Dinanath, F. R.; Minor, K. P.; Doll, R. J.; Girijavallabhan, V. M.; Santhanam, B.; Pinto, P. A.; Vibulbhan, B.; Keertikar, K. M.; Alvarez, C. S.; Baldwin, J. J.; Li, G.; Huang, C.-Y.; James, R. A.; Bishop, W. R.; Wang, J. J.-S.; Desai, J. A. US Patent Appl. 2004/122018, 2004.
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28
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33645389071
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note
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2S: C, 29.74; H, 5.82; N, 11.56. Found: C, 30.02; H, 5.61; N, 11.37.
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29
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33645387928
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note
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2S: C, 35.54; H, 6.71; N, 10.36. Found: C, 35.67; H, 6.80; N, 10.40.
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30
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33645381021
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US Patent Appl. 2004/0077551, 2004
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For procedures on synthesis of 3a,c, 4b, 5b and removal of t-Boc group, see: Campbell, J. A.; D'Andrea, S.; Good, A.; Li, J.; McPhee, F.; Ripka, A.; Scola, P. M.; Tu, Y. US Patent Appl. 2004/0077551, 2004.
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Campbell, J.A.1
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Good, A.3
Li, J.4
McPhee, F.5
Ripka, A.6
Scola, P.M.7
Tu, Y.8
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