Synthesis and peptidyl-prolyl isomerase inhibitory activity of quinoxalines as ligands of cyclophilin A

Chemical and Pharmaceutical Bulletin

Volumn 54, Issue 3, 2006, Pages 372-376

  Wang, Feng ^a   Chen, Jing ^a   Liu, Xuejun ^a   Shen, Xu ^a   He, Xuchang ^a   Jiang, Hualiang ^a   Bai, Donglu ^a  

^a SHANGHAI INSTITUTE OF MATERIA MEDICA   (China)

Author keywords

Cyclophilin A; Ligand; Peptidyl prolyl isomerase inhibitory activity; Quinoxaline

Indexed keywords

CYCLOPHILIN A; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; QUINOXALINE DERIVATIVE;

ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CRYSTAL STRUCTURE; DRUG SCREENING; DRUG SYNTHESIS; INFRARED SPECTROMETRY; KINETICS; LIGAND BINDING; PROTON NUCLEAR MAGNETIC RESONANCE;

CYCLOPHILIN A; ENZYME INHIBITORS; INDICATORS AND REAGENTS; KINETICS; MAGNETIC RESONANCE SPECTROSCOPY; PEPTIDYLPROLYL ISOMERASE; QUINOXALINES; SPECTROPHOTOMETRY, INFRARED; STRUCTURE-ACTIVITY RELATIONSHIP; SURFACE PLASMON RESONANCE;

EID: 33645244301     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.54.372     Document Type: Article

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