Synthesis of new potentially bioactive bicyclic 2-pyridones

Molecules

Volumn 10, Issue 10, 2005, Pages 1318-1324

  Crozet, Maxime D ^a   George, Pascal ^b   Crozet, Michel P ^a   Vanelle, Patrice ^a  

^a AIX MARSEILLE UNIVERSITY   (France)

^b SANOFI   (France)

Author keywords

Bicyclic 2 pyridones; Cyclization; Imidazopyridines; Nitro reduction; Thiazolopyridines

Indexed keywords

2 HYDROXYPYRIDINE; 2-HYDROXYPYRIDINE; PYRIDONE DERIVATIVE;

BIOLOGICAL MODEL; CHEMISTRY; CONFERENCE PAPER; CYCLIZATION; NITROSATION; SYNTHESIS;

CYCLIZATION; MODELS, BIOLOGICAL; NITROSATION; PYRIDONES;

EID: 33644793990     PISSN: 14203049     EISSN: 14203049     Source Type: Journal    
DOI: 10.3390/10101318     Document Type: Conference Paper

References (7)

1. Crozet, M. D.; Perfetti, P.; Kaafarani, M.; Crozet, M. P.; Vanelle, P. Rapid syntheses of nitroheterocycles that bear a diethyl methylenemalonate group β to a nitro group. Lett. Org. Chem. 2004, 7, 326-330.
2. 2-THF system. Tetrahedron Lett. 1990, 31, 4065-4066.
3. George, J.; Chandrasekaran, S. Selective reduction of nitro compounds with titanium(II) reagents. Synth. Commun. 1983, 73, 495-499.
4. Ho, T.-L.; Wong, C. M. Reduction of aromatic nitro compounds by titanium(III) chloride. Synthesis 1974, 45.
5. Boothroyd, S. R.; Kerr, M. A. A mild and efficient method for the preparation of anilines from nitroarenes. Tetrahedron Lett. 1995, 36, 2411-2414.
6. Entwistle, I. D.; Jackson, A. E.; Johnstone, R. A. W.; Telford, R. P. Reduction of nitro compounds. J. Chem. Soc., Perkin Trans. 1 1977, 443-444.
7. Crozet, M. D.; Suspène, C.; Kaafarani, M.; Crozet, M. P.; Vanelle, P. Synthesis of a new imidazo[4,5-b]pyridin-5-one via a vicarious nucleophilic substitution of hydrogen. Heterocycles 2004, 63, 1629-1635.