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Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 7, 2006, Pages 1920-1923

β-Diketo acids with purine nucleobase scaffolds: Novel, selective inhibitors of the strand transfer step of HIV integrase

(3) Nair, Vasu a Uchil, Vinod a Neamati, Nouri b

a UNIVERSITY OF GEORGIA (United States)

b UNIVERSITY OF SOUTHERN CALIFORNIA (United States)

Author keywords

HIV integrase inhibitors; Mechanism of inhibition; Purine diketo acids

Indexed keywords

INTEGRASE; INTEGRASE INHIBITOR; NUCLEIC ACID BASE; OXOACID;

ARTICLE; DNA STRAND; DNA TRANSFER; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS 1; WILD TYPE;

ACIDS; HIV INTEGRASE INHIBITORS; MODELS, MOLECULAR; PURINES;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 33144458429 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.12.093 Document Type: Article

Times cited : (26)

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