The mode of promoting activity of O-ethylmenthol as a transdermal absorption enhancer

Pharmaceutical Research

Volumn 23, Issue 2, 2006, Pages 392-400

  Obata, Yasuko ^a   Maruyama, Yoshimichi ^a   Takayama, Kozo ^a  

^a HOSHI UNIVERSITY   (Japan)

Author keywords

Confocal laser scanning microscopy; O ethylmenthol; Skin permeation; Transdermal drug delivery

Indexed keywords

ALCOHOL DERIVATIVE; CERAMIDE; CHOLESTEROL; CHOLESTEROL 3 SULFATE; CHOLESTEROL DERIVATIVE; FLUORESCENT DYE; LIPOSOME; O ETHYLMENTHOL; PALMITIC ACID; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CELL SWELLING; CONFOCAL LASER MICROSCOPY; CONTROLLED STUDY; DRUG DELIVERY SYSTEM; INTRACELLULAR FLUID; INTRACELLULAR SPACE; KERATINOCYTE; LASER MICROSCOPY; MALE; MORPHOLOGY; MOUSE; NONHUMAN; PRIORITY JOURNAL; SKIN SURFACE; STRATUM CORNEUM;

ADMINISTRATION, CUTANEOUS; ALGORITHMS; ANIMALS; ANISOTROPY; DRUG CARRIERS; EXCIPIENTS; KERATINOCYTES; LIPIDS; LIPOSOMES; MALE; MEMBRANE FLUIDITY; MENTHOL; MICE; MICE, INBRED HRS; MICROSCOPY, CONFOCAL; PHARMACEUTICAL SOLUTIONS; SKIN ABSORPTION;

EID: 32544432528     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1007/s11095-005-9257-6     Document Type: Article

References (24)

1. V. P. Shah C. C. Peck R. L. William 1993 Skin penetration enhancement K. A. Walter J. Hadgraft Pharmaceutical Skin Penetration Enhancement Marcel Dekker New York 417 427
2. R. H. Guy J. Hadgraft 1989 Structure-activity correlation R. L. Bronough H. I. Maibach Percutaneous Absorption 2 Marcel Dekker New York 95 109
3. J. Negishi K. Takayama K. Higashiyama Y. Chiba K. Isowa T. Nagai 1995 Promoting effect of O-alkylmenthol and O-acylmenthol derivatives on the percutaneous absorption of ketoprofen in rats STP Pharma Sci. 5 156 164
4. Y. Nakamura K. Takayama K. Higashiyama T. Suzuki T. Nagai 1996 Promoting effect of O-ethylmenthol on the percutaneous absorption of ketoprofen Int. J. Pharm. 145 29 36
5. Y. Obata K. Takayama Y. Maitani Y. Machida T. Nagai 1993 Effect of pretreatment of skin with cyclic monoterpenes on permeation of diclofenac in hairless rat Biol. Pharm. Bull. 16 312 314
6. Y. Obata C. J. Li M. Fujikawa K. Takayama H. Sato K. Higashiyama K. Isowa T. Nagai 2001 Evaluation and structure-activity relationship of synthesized cyclohexanol derivatives on percutaneous absorption of ketoprofen using artificial neural network Int. J. Pharm. 212 223 231
7. C. J. Li K. Higashiyama Y. Yoshimura T. Nagai K. Takayama Y. Obata 2001 Promoting mechanism of menthol derivative, 1-O-ethyl-3-buthylcyclohexanol, on the percutaneous absorption of ketoprofen Biol. Pharm. Bull. 24 1044 1048
8. H. Meerwein U. Eisenmenger H. Matthiae 1950 Tertiary oxonium salts. III. The addition of ethers to epichlorohydrin Annals 566 150 161
9. C. J. Lauter E. G. Trams 1962 A spectrophotometric determination of sphingosine J. Lipid Res. 3 136 138
10. T. Kai M. Nakayama Y. Kurosaki T. Nakayam T. Kimura 1993 Leratinized epithelial transport of β-blocking agents. III. Evaluation of enhancing effect on percutaneous absorption using model lipid liposomes Biol. Pharm. Bull. 16 801 805
11. M. R. Prausnitz J. A. Gimm R. H. Guy R. J. Janger C. Weaver C. Cullander 1996 Imaging regions of transport across human stratum corneum during high-voltage and low-voltage exposures J. Pharm. Sci. 85 1363 1370
12. N. G. Turner R. H. Guy 1997 Iontophoretic transport pathways: dependence on penetrant physicochemical properties J. Pharm. Sci. 86 1385 1389
13. M. E. van Kuijk-Meuwissen L. Mougin H. E. Junginger J. A. Bouwstra 1998 Application of vesicles to rat skin in vivo: a confocal laser scanning microscopy study J. Control. Release 56 189 196
14. C. Lombry N. Dujardin V. Preat 2000 Transdermal delivery of macromolecules using skin electroporation Pharm. Res. 17 32 37
15. O. D. Uitto H. S. White 2003 Electroosmotic pore transport in human skin Pharm. Res. 20 352 646
16. R. Alvarez-Roman A. Naik Y. N. Kalia H. Fessi R. H. Guy 2004 Visualization of skin penetration using confocal laser scanning microscopy Eur. J. Pharm. Biopharm. 58 301 316
17. A. H. Ghanem H. Mahmoud W. I. Higuchi U. D. Rohr S. Borsadia P. Liu J. L. Fox W. R. Good 1987 The effect of ethanol on the transport of β-estradiol and other permeants in hairless mouse skin. II. A new quantitative approach J. Control. Release 6 75 83
18. T. Kurihara-Bergstrom K. Knutson L. J. DeNoble C. Goates 1990 Percutaneous absorption enhancement of an ionic molecule by ethanol-water system in human skin Pharm. Res. 7 762 766
19. Y. Obata K. Takayama Y. Maitani Y. Machida T. Nagai 1993 Effect of ethanol of skin permeation of nonionized and ionized diclofenac Int. J. Pharm. 89 191 198
20. A. C. Williams B. W. Barry 2004 Penetration enhancers Adv. Drug Deliv. Rev. 56 603 618
21. Y. Obata T. Sesumi K. Takayama K. Isowa S. Grosh S. Wick R. Sitz T. Nagai 2000 Evaluation of skin damage caused by percutaneous absorption enhancers using fractal analysis J.Pharm. Sci. 89 556 561
22. T. Okusa Y. Obata K. Takayama K. Higashiyama T. Nagai 1997 Effect of menthol derivatives on skin permeation of oxybutynin Drug Deliv. Syst. 12 327 333
23. P. W. Wertz W. Abraham L. Landmann D. T. Downing 1986 Preparation of liposomes from stratum corneum lipids J. Invest. Dermatol. 87 582 584
24. W. Abraham D. T. Downing 1989 Preparation of model membranes for skin permeability studies using stratum corneum lipids J. Invest. Dermatol. 93 809 813