Syntheses and GABA uptake properties of 6-ether- and 6-enol ether-substituted nipecotic acids

European Journal of Medicinal Chemistry

Volumn 39, Issue 7, 2004, Pages 633-638

  N'Goka, Victor ^a   Bissantz, Caterina ^a   Bisel, Philippe ^a   Stenbøl, Tine B ^b   Krogsgaard Larsen, Povl ^b   Schlewer, Gilbert ^a  

^a Laboratoire de Pharmacochimie   (France)

^b UNIVERSITY OF COPENHAGEN   (Denmark)

Author keywords

Enol ether; Ether; GABA; GABA uptake inhibitors; Nipecotic acid

Indexed keywords

4 AMINOBUTYRIC ACID DERIVATIVE; NIPECOTIC ACID DERIVATIVE;

4 AMINOBUTYRIC ACID UPTAKE; ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG UPTAKE;

ETHERS; GAMMA-AMINOBUTYRIC ACID; NIPECOTIC ACIDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 3242741181     PISSN: 02235234     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejmech.2004.03.006     Document Type: Article

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