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Volumn 280, Issue 1-2, 2004, Pages 137-150

The effects of additives on the growth and morphology of paracetamol (acetaminophen) crystals

Author keywords

Acetaminophen; Additive; Atomic force microscopy; Crystal growth; Crystal morphology; Paracetamol

Indexed keywords

4 ACETOXYBENZOIC ACID; ACETANILIDE; METACETAMOL; METHYL PARABEN; ORTHOCETAMOL; PARACETAMOL; UNCLASSIFIED DRUG;

EID: 3242719432     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2004.05.010     Document Type: Article
Times cited : (74)

References (40)
  • 1
    • 0000067621 scopus 로고
    • The growth of crystals and the equilibrium structure of their surfaces
    • Burton W.K., Cabrera N., Frank F.C. The growth of crystals and the equilibrium structure of their surfaces. Phil. Trans. R. Soc., Lond. A243:1951;299-358
    • (1951) Phil. Trans. R. Soc., Lond. , vol.243 , pp. 299-358
    • Burton, W.K.1    Cabrera, N.2    Frank, F.C.3
  • 2
    • 0002893781 scopus 로고
    • The growth of crystals from solution
    • Doremus, R.H., Turnbull, D. (Eds.), Wiley, New York
    • Cabrera, N., Vermilyea, D.A., 1958. The growth of crystals from solution. In: Doremus, R.H., Turnbull, D. (Eds.), Growth and Perfection of Crystals. Wiley, New York, pp. 393-410.
    • (1958) Growth and Perfection of Crystals , pp. 393-410
    • Cabrera, N.1    Vermilyea, D.A.2
  • 3
    • 0021821356 scopus 로고
    • Modification of acetaminophen crystals: Influence of growth in aqueous solutions containing p-acetoxyacetanilide on crystal properties
    • Chow A.H.-L., Chow P.K.K., Zhongshan W., Grant D.J.W. Modification of acetaminophen crystals: influence of growth in aqueous solutions containing p-acetoxyacetanilide on crystal properties. Int. J. Pharm. 24:1985;239-258
    • (1985) Int. J. Pharm. , vol.24 , pp. 239-258
    • Chow, A.H.-L.1    Chow, P.K.K.2    Zhongshan, W.3    Grant, D.J.W.4
  • 4
    • 0023870479 scopus 로고
    • Modification of acetaminophen crystals. II. Influence of stirring rate during solution-phase growth on crystal properties in the presence and absence of p-acetoxyacetanilide
    • Chow A.H.-L., Grant D.J.W. Modification of acetaminophen crystals. II. Influence of stirring rate during solution-phase growth on crystal properties in the presence and absence of p-acetoxyacetanilide. Int. J. Pharm. 41:1988a;29-39
    • (1988) Int. J. Pharm. , vol.41 , pp. 29-39
    • Chow, A.H.-L.1    Grant, D.J.W.2
  • 5
    • 0023875577 scopus 로고
    • Modification of acetaminophen crystals. III. Influence of initial supersaturation during solution-phase growth on crystal properties in the presence and absence of p-acetoxyacetanilide
    • Chow A.H.-L., Grant D.J.W. Modification of acetaminophen crystals. III. Influence of initial supersaturation during solution-phase growth on crystal properties in the presence and absence of p-acetoxyacetanilide. Int. J. Pharm. 42:1988b;123-133
    • (1988) Int. J. Pharm. , vol.42 , pp. 123-133
    • Chow, A.H.-L.1    Grant, D.J.W.2
  • 6
    • 0021239020 scopus 로고
    • Modification of adipic acid crystals: Influence of growth in the presence of fatty acid additives on crystal properties
    • Chow K.Y., Go J., Mehdizadeh M., Grant D.J.W. Modification of adipic acid crystals: influence of growth in the presence of fatty acid additives on crystal properties. Int. J. Pharm. 20:1984;3-34
    • (1984) Int. J. Pharm. , vol.20 , pp. 3-34
    • Chow, K.Y.1    Go, J.2    Mehdizadeh, M.3    Grant, D.J.W.4
  • 7
    • 0001144994 scopus 로고
    • Structural and kinetic features of the crystal growth inhibition - Adipic acid growing in the presence of n-alkanoic acids
    • Davey R.J., Black S.N., Logan D., Maginn S.J., Fairbrother J.E., Grant D.J.W. Structural and kinetic features of the crystal growth inhibition - adipic acid growing in the presence of n-alkanoic acids. J. Chem. Soc. Faraday Trans. 88:1992;3461-3466
    • (1992) J. Chem. Soc. Faraday Trans. , vol.88 , pp. 3461-3466
    • Davey, R.J.1    Black, S.N.2    Logan, D.3    Maginn, S.J.4    Fairbrother, J.E.5    Grant, D.J.W.6
  • 10
    • 0027272306 scopus 로고
    • Effect of the opposite enantiomer on the physicochemical properties of (-)-ephedrinium 2-naphthalenesulphonate crystals
    • Duddu S.P., Fung F.K.Y., Grant D.J.W. Effect of the opposite enantiomer on the physicochemical properties of (-)-ephedrinium 2-naphthalenesulphonate crystals. Int. J. Pharm. 94:1993;171-179
    • (1993) Int. J. Pharm. , vol.94 , pp. 171-179
    • Duddu, S.P.1    Fung, F.K.Y.2    Grant, D.J.W.3
  • 11
    • 0030030510 scopus 로고    scopus 로고
    • Effects of crystallization in the presence of the opposite enantiomer on the crystal properties of (SS)-(+)-pseudoephedrinium
    • Duddu S.P., Fung F.K.Y., Grant D.J.W. Effects of crystallization in the presence of the opposite enantiomer on the crystal properties of (SS)-(+)-pseudoephedrinium. Int. J. Pharm. 127:1996;53-63
    • (1996) Int. J. Pharm. , vol.127 , pp. 53-63
    • Duddu, S.P.1    Fung, F.K.Y.2    Grant, D.J.W.3
  • 12
    • 0027485934 scopus 로고
    • Compression ability improvement by solvation/desolvation process: Application to paracetamol for direct compression
    • Fachaux J.M., Guyot-Hermann A.M., Guyot J.C. Compression ability improvement by solvation/desolvation process: application to paracetamol for direct compression. Int. J. Pharm. 99:1993;99-107
    • (1993) Int. J. Pharm. , vol.99 , pp. 99-107
    • Fachaux, J.M.1    Guyot-Hermann, A.M.2    Guyot, J.C.3
  • 14
    • 0001277493 scopus 로고
    • Pure paracetamol for direct compression. Part II. Study of the physicochemical and mechanical properties of sintered-like crystals of paracetamol
    • Fachaux J.M., Guyot-Hermann A.M., Guyot J.C., Conflant P., Drache M., Veesler S., Boistelle R. Pure paracetamol for direct compression. Part II. Study of the physicochemical and mechanical properties of sintered-like crystals of paracetamol. Powder Technol. 82:1995b;129-133
    • (1995) Powder Technol. , vol.82 , pp. 129-133
    • Fachaux, J.M.1    Guyot-Hermann, A.M.2    Guyot, J.C.3    Conflant, P.4    Drache, M.5    Veesler, S.6    Boistelle, R.7
  • 15
    • 0018117899 scopus 로고
    • The crystal habit modification of a tablet lubricant, adipic acid
    • Fairbrother J.E., Grant D.J.W. The crystal habit modification of a tablet lubricant, adipic acid. J. Pharm. Pharmacol. 30:1978;S19
    • (1978) J. Pharm. Pharmacol. , vol.30 , pp. 19
    • Fairbrother, J.E.1    Grant, D.J.W.2
  • 16
    • 0027963532 scopus 로고
    • Studies on paracetamol crystals produced by growth in aqueous solutions
    • Femi-Oyewo M.N., Spring M.S. Studies on paracetamol crystals produced by growth in aqueous solutions. Int. J. Pharm. 112:1994;17-28
    • (1994) Int. J. Pharm. , vol.112 , pp. 17-28
    • Femi-Oyewo, M.N.1    Spring, M.S.2
  • 17
    • 0034955290 scopus 로고    scopus 로고
    • Microhardness and dislocation identification studies on paracetamol single crystals
    • Finnie S.D., Prasad K.V.R., Sheen D.B., Sherwood J.N. Microhardness and dislocation identification studies on paracetamol single crystals. Pharm. Res. 18:2001;674-681
    • (2001) Pharm. Res. , vol.18 , pp. 674-681
    • Finnie, S.D.1    Prasad, K.V.R.2    Sheen, D.B.3    Sherwood, J.N.4
  • 18
    • 0033364606 scopus 로고    scopus 로고
    • Morphological and growth rate distributions of small self-nucleated paracetamol crystals grown from pure aqueous solutions
    • Finnie S.D., Ristic R.I., Sherwood J.N., Zikic A.M. Morphological and growth rate distributions of small self-nucleated paracetamol crystals grown from pure aqueous solutions. J. Cryst. Growth. 207:1999;308-318
    • (1999) J. Cryst. Growth , vol.207 , pp. 308-318
    • Finnie, S.D.1    Ristic, R.I.2    Sherwood, J.N.3    Zikic, A.M.4
  • 21
    • 0036131451 scopus 로고    scopus 로고
    • Influence of supersaturation and structurally related additives on the crystal growth of alpha-lactose monohydrate
    • Garnier S., Petit S., Coquerel G. Influence of supersaturation and structurally related additives on the crystal growth of alpha-lactose monohydrate. J. Cryst. Growth. 234:2002;201-219
    • (2002) J. Cryst. Growth , vol.234 , pp. 201-219
    • Garnier, S.1    Petit, S.2    Coquerel, G.3
  • 22
    • 0035997343 scopus 로고    scopus 로고
    • Relationship between particle size and impurity incorporation during crystallization of (+)-pseudoephedrine hydrochloride, acetaminophen, and adipic acid from aqueous solution
    • Gu C.-H., Grant D.J.W. Relationship between particle size and impurity incorporation during crystallization of (+)-pseudoephedrine hydrochloride, acetaminophen, and adipic acid from aqueous solution. Pharm. Res. 19:2002;1068-1070
    • (2002) Pharm. Res. , vol.19 , pp. 1068-1070
    • Gu, C.-H.1    Grant, D.J.W.2
  • 23
    • 0001125628 scopus 로고
    • The orthorhombic form of p-hydroxyacetanilide
    • Haisa M., Kashino S., Haeda H. The orthorhombic form of p-hydroxyacetanilide. Acta Cryst. B30:1974;2510-2512
    • (1974) Acta Cryst. , vol.30 , pp. 2510-2512
    • Haisa, M.1    Kashino, S.2    Haeda, H.3
  • 24
    • 0001335827 scopus 로고
    • The monoclinic form of p-hydroxyacetanilide
    • Haisa M., Kashino S., Kawai R., Maeda H. The monoclinic form of p-hydroxyacetanilide. Acta Cryst. B32:1976;1283-1285
    • (1976) Acta Cryst. , vol.32 , pp. 1283-1285
    • Haisa, M.1    Kashino, S.2    Kawai, R.3    Maeda, H.4
  • 25
    • 0029633485 scopus 로고
    • The effect of structurally related substances on the nucleation kinetics of paracetamol (acetaminophen)
    • Hendriksen B.A., Grant D.J.W. The effect of structurally related substances on the nucleation kinetics of paracetamol (acetaminophen). J. Cryst. Growth. 156:1995;252-260
    • (1995) J. Cryst. Growth , vol.156 , pp. 252-260
    • Hendriksen, B.A.1    Grant, D.J.W.2
  • 26
    • 0032002437 scopus 로고    scopus 로고
    • Crystallisation of paracetamol (acetaminophen) in the presence of structurally related substances
    • Hendriksen B.A., Grant D.J.W., Meenan P., Green D.A. Crystallisation of paracetamol (acetaminophen) in the presence of structurally related substances. J. Cryst. Growth. 183:1998;629-640
    • (1998) J. Cryst. Growth , vol.183 , pp. 629-640
    • Hendriksen, B.A.1    Grant, D.J.W.2    Meenan, P.3    Green, D.A.4
  • 27
    • 0002499611 scopus 로고
    • The influence of impurities and solvents on crystallisation
    • Myerson, A. (Ed.), Butterworth-Heinemann, Boston
    • Klug, D.L., 1993. The influence of impurities and solvents on crystallisation. In: Myerson, A. (Ed.), Handbook of Industrial Crystallization. Butterworth-Heinemann, Boston, pp. 65-87.
    • (1993) Handbook of Industrial Crystallization , pp. 65-87
    • Klug, D.L.1
  • 28
    • 0033900784 scopus 로고    scopus 로고
    • The evolution of growth modes and activity of growth sources on canavalin investigated by in situ atomic force microscopy
    • Land T.A., De Yoreo J.J. The evolution of growth modes and activity of growth sources on canavalin investigated by in situ atomic force microscopy. J. Cryst. Growth. 208:2000;623-637
    • (2000) J. Cryst. Growth , vol.208 , pp. 623-637
    • Land, T.A.1    De Yoreo, J.J.2
  • 30
    • 0033906037 scopus 로고    scopus 로고
    • Growth of potassium sulphate crystals in the presence of organic dyes: In situ characterization by atomic force microscopy
    • Mauri A., Moret M. Growth of potassium sulphate crystals in the presence of organic dyes: in situ characterization by atomic force microscopy. J. Cryst. Growth. 208:2000;599-614
    • (2000) J. Cryst. Growth , vol.208 , pp. 599-614
    • Mauri, A.1    Moret, M.2
  • 32
    • 0029509885 scopus 로고
    • A comparison of binding-energy and metastable zone width for adipic acid with various additives
    • Myerson A.S., Jang S.M. A comparison of binding-energy and metastable zone width for adipic acid with various additives. J. Cryst. Growth. 156:1995;459-466
    • (1995) J. Cryst. Growth , vol.156 , pp. 459-466
    • Myerson, A.S.1    Jang, S.M.2
  • 34
    • 0342345810 scopus 로고    scopus 로고
    • Optical properties of polymorphic forms I and II of paracetamol
    • Nichols G. Optical properties of polymorphic forms I and II of paracetamol. Microscope. 46:1998;117-122
    • (1998) Microscope , vol.46 , pp. 117-122
    • Nichols, G.1
  • 35
    • 0031808764 scopus 로고    scopus 로고
    • Physicochemical characterization of the orthorhombic polymorph of paracetamol crystallized from solution
    • Nichols G., Frampton C.S. Physicochemical characterization of the orthorhombic polymorph of paracetamol crystallized from solution. J. Pharm. Sci. 87:1998;684-693
    • (1998) J. Pharm. Sci. , vol.87 , pp. 684-693
    • Nichols, G.1    Frampton, C.S.2
  • 36
    • 0035857724 scopus 로고    scopus 로고
    • Crystallization of paracetamol from solution in the presence and absence of impurity
    • Prasad K.V.R., Ristic R.I., Sheen D.B., Sherwood J.N. Crystallization of paracetamol from solution in the presence and absence of impurity. Int. J. Pharm. 215:2001;29-44
    • (2001) Int. J. Pharm. , vol.215 , pp. 29-44
    • Prasad, K.V.R.1    Ristic, R.I.2    Sheen, D.B.3    Sherwood, J.N.4
  • 37
    • 0035960211 scopus 로고    scopus 로고
    • Macro- and micromorphology of monoclinic paracetamol grown from pure aqueous solution
    • Ristic R.I., Finnie S., Sheen D.B., Sherwood J.N. Macro- and micromorphology of monoclinic paracetamol grown from pure aqueous solution. J. Phys. Chem. B. 105:2001;9057-9066
    • (2001) J. Phys. Chem. B. , vol.105 , pp. 9057-9066
    • Ristic, R.I.1    Finnie, S.2    Sheen, D.B.3    Sherwood, J.N.4
  • 38
    • 0000299224 scopus 로고    scopus 로고
    • In situ optical interferometric studies of the growth and dissolution behaviour of paracetamol (acetaminophen). 1. Growth kinetics
    • Shekunov B.Y., Grant D.J.W. In situ optical interferometric studies of the growth and dissolution behaviour of paracetamol (acetaminophen). 1. Growth kinetics. J. Phys. Chem. B. 101:1997;3973-3979
    • (1997) J. Phys. Chem. B. , vol.101 , pp. 3973-3979
    • Shekunov, B.Y.1    Grant, D.J.W.2
  • 39
    • 0031247438 scopus 로고    scopus 로고
    • In situ optical interferometric studies of the growth and dissolution behaviour of paracetamol (acetaminophen) crystals. 3. Influence of growth in the presence of p-acetoxyacetanilide
    • Shekunov B.Y., Grant D.J.W., Latham R.J., Sherwood J.N. In situ optical interferometric studies of the growth and dissolution behaviour of paracetamol (acetaminophen) crystals. 3. Influence of growth in the presence of p-acetoxyacetanilide. J. Phys. Chem. B. 101:1997;9107-9112
    • (1997) J. Phys. Chem. B. , vol.101 , pp. 9107-9112
    • Shekunov, B.Y.1    Grant, D.J.W.2    Latham, R.J.3    Sherwood, J.N.4
  • 40
    • 0001495753 scopus 로고
    • Tailor-made additives and impurities
    • Mersmann, A. (Ed.), Marcel Dekker, New York
    • Weissbuch, I., Leiserowitz, L., Lahav, M., 1995. Tailor-made additives and impurities. In: Mersmann, A. (Ed.), Crystallization Technology Handbook. Marcel Dekker, New York, pp. 401-457.
    • (1995) Crystallization Technology Handbook , pp. 401-457
    • Weissbuch, I.1    Leiserowitz, L.2    Lahav, M.3


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