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Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 6, 2006, Pages 1731-1734

Seco-prolinenitrile inhibitors of dipeptidyl peptidase IV define minimal pharmacophore requirements at P1

(7) Magnin, David R a Taunk, Prakash C a Robertson, James G a Wang, Aiying a Marcinkeviciene, Jovita a Kirby, Mark S a Hamann, Lawrence G a

a BRISTOL MYERS SQUIBB (United States)

Author keywords

Antidiabetic; Dipeptidyl peptidase IV; Enzyme inhibitors; Serine protease

Indexed keywords

DIPEPTIDYL PEPTIDASE IV; DIPEPTIDYL PEPTIDASE IV INHIBITOR;

ARTICLE; ENZYME INHIBITION; ENZYME STRUCTURE; NON INSULIN DEPENDENT DIABETES MELLITUS; PHARMACOPHORE; STRUCTURE ACTIVITY RELATION;

ADENOSINE DEAMINASE; ANILINE COMPOUNDS; ANTIGENS, CD26; DIPEPTIDES; ENZYME INHIBITORS; GLYCOPROTEINS; HUMANS; NITRILES; PROLINE;

EID: 32044457012 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.11.098 Document Type: Article

Times cited : (5)

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