Synthesis of 2-aminoaryl-5-substituted-1,3,4-thiadiazoles in a thermal 1,3-dipolar cycloaddition reaction

Phosphorus, Sulfur and Silicon and the Related Elements

Volumn 180, Issue 12, 2005, Pages 2653-2666

  Gobis, Katarzyna ^a   Foks, Henryk ^a   Zwolska, Zofia ^b   Augustynowicz Kopeć, Ewa ^b  

^a MEDICAL UNIVERSITY OF GDANSK   (Poland)

^b NATIONAL TUBERCULOSIS AND LUNG DISEASES RESEARCH INSTITUTE   (Poland)

Author keywords

1,3,4 thiadiazoles; 1,3 Dipolar cycloaddition; 4 substituted thiosemicarbazides; Antituberculosis activity; Hydroxamoyl chlorides; Methyl dithiocarbazinate

Indexed keywords

EID: 31544473773     PISSN: 10426507     EISSN: 15635325     Source Type: Journal    
DOI: 10.1080/104265090930399     Document Type: Article

References (11)

1. F. A. Ashour, N. S. Habbib, M. el Taibbi, S. el Dine, and A.S. el Dine, Farmaco, 45, 1341 (1990).
2. A. Foroumadi, M. Daneshtalb, M. Mahmoudian, M. Falahati, N. Nateghian, N. Shahsavarani, and A. Shafiee, Pharm. Pharmacol. Commun., 4, 95 (1998).
3. A. Foroumadi, M. Mirzaei, and A. Shafiee, Pharmazie, 56, 610 (2001).
4. V. R. Rao and V. R. Srinivasan, Indian J. Chem., 8, 509 (1970).
5. I. Lalezari and A. Shafiee, J. Heterocyclic Chem., 8, 835 (1971).
6. A. Dornow and K. Fischer, Chem. Ber., 99, 72 (1966).
7. T. Sasaki and T. Yoshioka, Bull. Chem. Soc. Jpn., 41, 2211 (1968).
8. M. Kočevar, S. Polanc, M. Sollner, M. Tišler, and B. Verček, Synth. Commun., 18, 1427 (1988).
9. D. L. Kleyman, J. F. Bartosevich, T. S. Griffin, C. J. Mason, and J. P. Scovill, J. Med. Chem., 22, 855 (1979).
10. K. C. Agrawal, M. H. Lee, B. A. Booth, E. C. Moore, and A. C. Sartorelli, J. Med. Chem., 17, 934 (1974).
11. H. Foks, M. Buraczewska, W. Manowska, and J. Sawlewicz, Dissert. Pharm. Pharmacol., 23, 49 (1971).