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Volumn 29, Issue 1, 2004, Pages 53-66

Drug-carrier interaction in solid dispersions prepared by co-grinding and melt-quenching

Author keywords

[No Author keywords available]

Indexed keywords

CRYSTALLIZATION; DRUG PRODUCTS; GRINDING (MACHINING); QUENCHING; STRESS ANALYSIS;

EID: 3042794601     PISSN: 01519107     EISSN: None     Source Type: Journal    
DOI: 10.3166/acsm.29.53-66     Document Type: Review
Times cited : (11)

References (35)
  • 1
    • 0015124656 scopus 로고
    • Pharmaceutical applications of solid dispersion system
    • W. L. Chiou, S. Riegelman, Pharmaceutical applications of solid dispersion system, J. Pharm. Sci. 60 (1971) 1281-1302.
    • (1971) J. Pharm. Sci. , vol.60 , pp. 1281-1302
    • Chiou, W.L.1    Riegelman, S.2
  • 2
    • 0000550329 scopus 로고    scopus 로고
    • 2 under moderate mechanical stressing. I: A solid state acid-base reaction and charge transfer due to complex formation
    • 2 under moderate mechanical stressing. I: A solid state acid-base reaction and charge transfer due to complex formation, J. Solid State Chem. 122 (1) (1996) 74-80.
    • (1996) J. Solid State Chem. , vol.122 , Issue.1 , pp. 74-80
    • Watanabe, T.1    Isobe, T.2    Senna, M.3
  • 3
    • 0000550326 scopus 로고    scopus 로고
    • 2 under moderate mechanical stressing. II: Examination of a radical mechanism by an EPR study
    • 2 under moderate mechanical stressing. II: examination of a radical mechanism by an EPR study, J. Solid State Chem. 122 (2) (1996) 291-296.
    • (1996) J. Solid State Chem. , vol.122 , Issue.2 , pp. 291-296
    • Watanabe, T.1    Isobe, T.2    Senna, M.3
  • 4
    • 0001156142 scopus 로고    scopus 로고
    • 2 under moderate mechanical stressing. III. Changes in the short range ordering throughout the mechanical and thermal processes
    • 2 under moderate mechanical stressing. III. Changes in the short range ordering throughout the mechanical and thermal processes, J. Solid State Chem. 130 (2) (1997) 284-289.
    • (1997) J. Solid State Chem. , vol.130 , Issue.2 , pp. 284-289
    • Watanabe, T.1    Isobe, T.2    Senna, M.3
  • 5
    • 0000727947 scopus 로고    scopus 로고
    • Electronegativity equalization during mechanochemical addition reaction
    • T. Watanabe, T. Isobe, M. Senna, Electronegativity equalization during mechanochemical addition reaction, Chem. Sustainable Dev. 6 (1998) 165-168.
    • (1998) Chem. Sustainable Dev. , vol.6 , pp. 165-168
    • Watanabe, T.1    Isobe, T.2    Senna, M.3
  • 6
    • 0027109587 scopus 로고
    • Application of the DV-Xα cluster method to calculations of the electronic structure of silicate and phosphate glasses
    • Y. Kowada, H. Adachi, M. Tatsumisago, T. Minami, Application of the DV-Xα cluster method to calculations of the electronic structure of silicate and phosphate glasses, J. Non-Cryst. Solids 150 (1992) 318-321.
    • (1992) J. Non-Cryst. Solids , vol.150 , pp. 318-321
    • Kowada, Y.1    Adachi, H.2    Tatsumisago, M.3    Minami, T.4
  • 7
    • 4243153481 scopus 로고
    • Discrete variational Xα cluster calculation. II. Application to surface electronic structure of MgO
    • C. Satoko, M. Tsukada, H. Adachi, Discrete variational Xα cluster calculation. II. Application to surface electronic structure of MgO, J. Phys. Soc. Jpn. 45 (1978) 1333-1340.
    • (1978) J. Phys. Soc. Jpn. , vol.45 , pp. 1333-1340
    • Satoko, C.1    Tsukada, M.2    Adachi, H.3
  • 8
    • 1642330656 scopus 로고    scopus 로고
    • Study of the interaction of ethanol with the Brønsted and Lewis acid sites on metal oxide surfaces using the DV-Xα method
    • Y. Shinohara, H. Satozono, T. Nakajima, S. Suzuki, S. Mishima, Study of the interaction of ethanol with the Brønsted and Lewis acid sites on metal oxide surfaces using the DV-Xα method, J. Chem. Software 4 (1998) 41-50.
    • (1998) J. Chem. Software , vol.4 , pp. 41-50
    • Shinohara, Y.1    Satozono, H.2    Nakajima, T.3    Suzuki, S.4    Mishima, S.5
  • 10
    • 0004053069 scopus 로고    scopus 로고
    • A molecular orbital approach toward soft-mechanochemical synthesis from the view point of hetero-metalloxane bonding under mechanical stressing
    • Y. Fujiwara, T. Isobe, M. Senna, J. Tanaka, A molecular orbital approach toward soft-mechanochemical synthesis from the view point of hetero-metalloxane bonding under mechanical stressing, Trans. Mater. Res. Soc. Jpn. 25 (2000) 139-142.
    • (2000) Trans. Mater. Res. Soc. Jpn. , vol.25 , pp. 139-142
    • Fujiwara, Y.1    Isobe, T.2    Senna, M.3    Tanaka, J.4
  • 11
    • 0035330347 scopus 로고    scopus 로고
    • Molecular dynamic-molecular orbital combined study on the solid state interfacial reaction under mechanical stressing
    • M. Senna, Y. Fujiwara, T. Isobe, J. Tanaka, Molecular dynamic-molecular orbital combined study on the solid state interfacial reaction under mechanical stressing, Solid State Ionics 141-142 (2001) 31-38.
    • (2001) Solid State Ionics , vol.141-142 , pp. 31-38
    • Senna, M.1    Fujiwara, Y.2    Isobe, T.3    Tanaka, J.4
  • 12
    • 0031056536 scopus 로고    scopus 로고
    • Effects of sorbed water on the crystallization of indomethacin from the amorphous state
    • V. Andronis, M. Yoshioka, G. Zografi, Effects of sorbed water on the crystallization of indomethacin from the amorphous state, J. Pharm. Sci. 86 (1997) 346-351.
    • (1997) J. Pharm. Sci. , vol.86 , pp. 346-351
    • Andronis, V.1    Yoshioka, M.2    Zografi, G.3
  • 14
    • 0036330185 scopus 로고    scopus 로고
    • Solid state radical recombination and charge transfer across the boundary between indomethacin and silica under mechanical stress
    • T. Watanabe, S. Hasegawa, N. Wakiyama, F. Usui, A. Kusai, T. Isobe, M. Senna, Solid state radical recombination and charge transfer across the boundary between indomethacin and silica under mechanical stress, J. Solid State Chem. 164 (2002) 27-33.
    • (2002) J. Solid State Chem. , vol.164 , pp. 27-33
    • Watanabe, T.1    Hasegawa, S.2    Wakiyama, N.3    Usui, F.4    Kusai, A.5    Isobe, T.6    Senna, M.7
  • 15
    • 0037043078 scopus 로고    scopus 로고
    • Stabilization of amorphous indomethacin by co-grinding in a ternary mixture
    • T. Watanabe, I. Ohno, N. Wakiyama, A. Kusai, M. Senna, Stabilization of amorphous indomethacin by co-grinding in a ternary mixture, Int. J. Pharm. 241 (2002) 103-111.
    • (2002) Int. J. Pharm. , vol.241 , pp. 103-111
    • Watanabe, T.1    Ohno, I.2    Wakiyama, N.3    Kusai, A.4    Senna, M.5
  • 16
    • 0036856710 scopus 로고    scopus 로고
    • Controlled dissolution properties of indomethacin by compounding with silica
    • T. Watanabe, I. Ohno, N. Wakiyama, A. Kusai, M. Senna, Controlled dissolution properties of indomethacin by compounding with silica, S.T.P. Pharma Sciences 12 (2002) 363-367.
    • (2002) S.T.P. Pharma Sciences , vol.12 , pp. 363-367
    • Watanabe, T.1    Ohno, I.2    Wakiyama, N.3    Kusai, A.4    Senna, M.5
  • 17
    • 0032528994 scopus 로고    scopus 로고
    • Dissolution improvement of RS-8359 by the solid dispersion prepared by the solvent method
    • F. Usui, K. Maeda, A. Kusai, M. Ikeda, K. Nishimura, K. Yamamoto, Dissolution improvement of RS-8359 by the solid dispersion prepared by the solvent method, Int. J. Pharm. 170 (1998) 247-256.
    • (1998) Int. J. Pharm. , vol.170 , pp. 247-256
    • Usui, F.1    Maeda, K.2    Kusai, A.3    Ikeda, M.4    Nishimura, K.5    Yamamoto, K.6
  • 18
    • 0022869176 scopus 로고
    • La diffrattometria a raggi X nell'analisl di prodotti farmaceutici: Fenomeni di polimorfismo nell'indometacina
    • R. Zannetti, A. Marigo, A. Guerrato, B. Bortoletti, La diffrattometria a raggi X nell'analisl di prodotti farmaceutici: fenomeni di polimorfismo nell'indometacina, Boll.Chem.Farm. 125 (1986) 180-189.
    • (1986) Boll.Chem.Farm. , vol.125 , pp. 180-189
    • Zannetti, R.1    Marigo, A.2    Guerrato, A.3    Bortoletti, B.4
  • 19
    • 0345337277 scopus 로고    scopus 로고
    • Spectroscopic identification of an amorphous-to crystalline drug transition in a solid dispersion SCH 48461 capsule formation
    • R. J. Markovich, C. A. Evans, C. B. Coscolluela, S. A. Zibas, J. Rosen, Spectroscopic identification of an amorphous-to crystalline drug transition in a solid dispersion SCH 48461 capsule formation, J. Pharm. Biomed. Anal. 16 (1997) 661-673.
    • (1997) J. Pharm. Biomed. Anal. , vol.16 , pp. 661-673
    • Markovich, R.J.1    Evans, C.A.2    Coscolluela, C.B.3    Zibas, S.A.4    Rosen, J.5
  • 20
    • 0031792334 scopus 로고    scopus 로고
    • Comparison of solid-state NMR and isothermal microcalorimetry in the assessment of the amorphous component of lactose
    • C. Gustafsson, H. Lennholm, T. Iversen, C. Nystrom, Comparison of solid-state NMR and isothermal microcalorimetry in the assessment of the amorphous component of lactose, Int. J. Pharm. 174 (1998) 243-252.
    • (1998) Int. J. Pharm. , vol.174 , pp. 243-252
    • Gustafsson, C.1    Lennholm, H.2    Iversen, T.3    Nystrom, C.4
  • 21
    • 0033004759 scopus 로고    scopus 로고
    • Nucleation and crystallization kinetics of hydrated amorphous lactose above glass transition temperature
    • E. A. Schmitt, D. Law, G. G. Z. Zhang, Nucleation and crystallization kinetics of hydrated amorphous lactose above glass transition temperature, J. Pharm. Sci. 88 (1999) 291-296.
    • (1999) J. Pharm. Sci. , vol.88 , pp. 291-296
    • Schmitt, E.A.1    Law, D.2    Zhang, G.G.Z.3
  • 22
  • 23
    • 0026705833 scopus 로고
    • Isolation and solid-state characteristics of a new crystal form of indomethacin
    • S. Y. Lin, Isolation and solid-state characteristics of a new crystal form of indomethacin, J. Pharm. Sci. 81 (1992) 572-576.
    • (1992) J. Pharm. Sci. , vol.81 , pp. 572-576
    • Lin, S.Y.1
  • 24
    • 0027535951 scopus 로고
    • Vacancy-associated type ESR centres observed in natural silica and their application to geology
    • T. Fukuchi, Vacancy-associated type ESR centres observed in natural silica and their application to geology, Appl. Radiat. Isot. 44 (1993) 179-184.
    • (1993) Appl. Radiat. Isot. , vol.44 , pp. 179-184
    • Fukuchi, T.1
  • 26
    • 0026240981 scopus 로고
    • Optical properties and structure of defects in silica glass
    • D. L. Griscom, Optical properties and structure of defects in silica glass, J. Ceram. Soc. Jpn. 99 (1991) 923-942.
    • (1991) J. Ceram. Soc. Jpn. , vol.99 , pp. 923-942
    • Griscom, D.L.1
  • 27
    • 0001459245 scopus 로고
    • Correlation of preexisting diamagnetic defect centres with induced paramagnetic defect centres by ultraviolet or vacuum-ultraviolet photons in high-purity silica glasses
    • H. Nishikawa, R. Nakamura, Y. Ohki, Y. Hama, Correlation of preexisting diamagnetic defect centres with induced paramagnetic defect centres by ultraviolet or vacuum-ultraviolet photons in high-purity silica glasses, Phys. Rev. B 48 (1993) 15584-15594.
    • (1993) Phys. Rev. B , vol.48 , pp. 15584-15594
    • Nishikawa, H.1    Nakamura, R.2    Ohki, Y.3    Hama, Y.4
  • 28
    • 0000003126 scopus 로고
    • Radiation damage of germanium-doped silica glasses: Spectral simplification by photo-and thermal bleaching, spectral identification and microwave saturation characteristics
    • W. Chamulitrat, L. Kevan, R. N. Schwartz, G. Richard, G. L. Tangonan, Radiation damage of germanium-doped silica glasses: Spectral simplification by photo-and thermal bleaching, spectral identification and microwave saturation characteristics, J. Appl. Phys. 59 (1986) 2933-2939.
    • (1986) J. Appl. Phys. , vol.59 , pp. 2933-2939
    • Chamulitrat, W.1    Kevan, L.2    Schwartz, R.N.3    Richard, G.4    Tangonan, G.L.5
  • 29
    • 0000181579 scopus 로고    scopus 로고
    • In situ radiolysis steady-state ESR study of carboxyalkyl radical trapping by 5,5-dimethyl-1-pyrroline-N-oxide
    • H. Taniguchi, K. P. Madden, In situ radiolysis steady-state ESR study of carboxyalkyl radical trapping by 5,5-dimethyl-1-pyrroline-N-oxide, J. Phys. Chem. A 102 (1998) 6753-6759.
    • (1998) J. Phys. Chem. A , vol.102 , pp. 6753-6759
    • Taniguchi, H.1    Madden, K.P.2
  • 30
    • 0015520402 scopus 로고
    • Crystal and molecular structure of an antiinflammatory agent, indomethacin, 1-(p-chlorobenzoyl)-5-methoxy-2-methylindole-3-acetic acid
    • T. J. Kistenmacher, E. Marsh, Crystal and molecular structure of an antiinflammatory agent, indomethacin, 1-(p-chlorobenzoyl)-5-methoxy-2- methylindole-3-acetic acid, J. Am. Chem. Soc. 94 (1972) 1340-1345.
    • (1972) J. Am. Chem. Soc. , vol.94 , pp. 1340-1345
    • Kistenmacher, T.J.1    Marsh, E.2
  • 31
    • 0022601812 scopus 로고
    • Effect of environmental temperature on polymorphic solid-state transformation of indomethacin during grinding
    • M. Otsuka, T. Matsumoto, N. Kaneniwa, Effect of environmental temperature on polymorphic solid-state transformation of indomethacin during grinding, Chem. Pharm. Bull. 34 (1986) 1784-1793.
    • (1986) Chem. Pharm. Bull. , vol.34 , pp. 1784-1793
    • Otsuka, M.1    Matsumoto, T.2    Kaneniwa, N.3
  • 33
    • 0031772192 scopus 로고    scopus 로고
    • The versatile surface properties of poly (cyclopentadiene)-modified silica particles (PCPD-silica). XPS and electrokinetic studies
    • F. Simon, H. J. Jacobasch, S. Spange, The versatile surface properties of poly (cyclopentadiene) -modified silica particles (PCPD-silica). XPS and electrokinetic studies, Colloid Polym. Sci. 276 (1998) 930-939.
    • (1998) Colloid Polym. Sci. , vol.276 , pp. 930-939
    • Simon, F.1    Jacobasch, H.J.2    Spange, S.3
  • 35
    • 3042766813 scopus 로고    scopus 로고
    • Molecular orbital study on the solid state reaction between indomethacin and silica under mechanical stress
    • in press
    • T. Watanabe, N. Wakiyama, A. Kusai, M. Senna, Molecular orbital study on the solid state reaction between indomethacin and silica under mechanical stress, Powder Technology, in press.
    • Powder Technology
    • Watanabe, T.1    Wakiyama, N.2    Kusai, A.3    Senna, M.4


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