Use of 2-azido-3-[125I]iodo-7,8-dibromodibenzo-p-dioxin as a probe to determine the relative ligand affinity of human versus mouse aryl hydrocarbon receptor in cultured cells

Molecular Pharmacology

Volumn 66, Issue 1, 2004, Pages 129-136

  Ramadoss, Preeti ^a   Perdew, Gary H ^a  

^a PENNSYLVANIA STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2 AZIDO 3 IODO 7,8 DIBROMODIBENZO PARA DIOXIN I 125; 2,3,7,8 TETRACHLORODIBENZO PARA DIOXIN; AROMATIC HYDROCARBON RECEPTOR; CHOLINERGIC RECEPTOR; TRANSCRIPTION FACTOR; UNCLASSIFIED DRUG;

ALLELE; ANIMAL CELL; ARTICLE; BINDING AFFINITY; CELL CULTURE; COMPETITIVE INHIBITION; CONFORMATIONAL TRANSITION; DRUG DETERMINATION; HUMAN; HUMAN CELL; LIGAND BINDING; MEMBRANE POTENTIAL; MOLECULAR PROBE; MOUSE; NONHUMAN; PHOTOAFFINITY LABELING; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR OCCUPANCY; SAMPLING; STRAIN DIFFERENCE; STRUCTURE ANALYSIS; TRANSACTIVATION;

ALANINE; ANIMALS; BINDING, COMPETITIVE; CELLS, CULTURED; COS CELLS; DIOXINS; HUMANS; IODINE RADIOISOTOPES; MICE; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, ARYL HYDROCARBON; SPECIES SPECIFICITY; TETRACHLORODIBENZODIOXIN; VALINE;

EID: 3042677511     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.66.1.129     Document Type: Article

References (20)

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