Process development of a large-scale synthesis of TKA731: A tachykinin receptor antagonist

Organic Process Research and Development

Volumn 8, Issue 3, 2004, Pages 330-340

  Prashad, Mahavir ^a   Har, Denis ^a   Hu, Bin ^a   Kim, Hong Yong ^a   Girgis, Michael J ^a   Chaudhary, Apurva ^a   Repič, Oljan ^a   Blacklock, Thomas J ^a   Marterer, Wolfgang ^b  

^a NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH   (United States)

^b NOVARTIS PHARMA AG   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

CARBON DIOXIDE; DIMETHYL SULFATE; QUINAZOLINONE DERIVATIVE; TACHYKININ RECEPTOR ANTAGONIST; TKA 731; URETHAN;

ARTICLE; DEPROTECTION REACTION; DRUG SYNTHESIS; METHYLATION; PROCESS DEVELOPMENT;

EID: 3042635346     PISSN: 10836160     EISSN: None     Source Type: Journal    
DOI: 10.1021/op0341824     Document Type: Article

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