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1
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0037435046
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Recent reviews on SERMs:
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Recent reviews on SERMs: Jordan V.C. J. Med. Chem. 46:2003;883
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Jordan, V.C.1
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6
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15144355781
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Representative SERMs: EVISTA:
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Representative SERMs: EVISTA: Grese T.A., Pennington L.D., Sluka J.P., Adrian M.D., Cole H.W., Fuson T.R., Magee D.E., Phillips D.L., Rowley E.R., Shetler P.K., Short L.L., Venugopalan M., Yang N.N., Sato M., Glasebrook A.L., Bryant H.U. J. Med. Chem. 41:1998;1272
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Grese, T.A.1
Pennington, L.D.2
Sluka, J.P.3
Adrian, M.D.4
Cole, H.W.5
Fuson, T.R.6
Magee, D.E.7
Phillips, D.L.8
Rowley, E.R.9
Shetler, P.K.10
Short, L.L.11
Venugopalan, M.12
Yang, N.N.13
Sato, M.14
Glasebrook, A.L.15
Bryant, H.U.16
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8
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0035714539
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EM-652, SCH57068:
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EM-652, SCH57068: Labrie M., Labrie C., Belanger A., Simard J., Giguere V., Tremblay A., Tremblay G. J. Steroid. Biochem. Mol. Biol. 79:2001;213
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Labrie, M.1
Labrie, C.2
Belanger, A.3
Simard, J.4
Giguere, V.5
Tremblay, A.6
Tremblay, G.7
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9
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0001236520
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Lasofoxifene:
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Lasofoxifene: Ke H.Z., Paralkar V.M., Grasser W.A., Crawford D.T., Qi H., Simmons H.A., Pirie C.M., Chidsey-Frink K.L., Owen T.A., Smock S.L., Chen H.K., Jee W.S.S., Cameron K.O., Rosati R.L., Brown T.A., DaSilva Jardine P., Thompson D.D. Endocrinology. 139:1998;2068
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(1998)
Endocrinology
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Ke, H.Z.1
Paralkar, V.M.2
Grasser, W.A.3
Crawford, D.T.4
Qi, H.5
Simmons, H.A.6
Pirie, C.M.7
Chidsey-Frink, K.L.8
Owen, T.A.9
Smock, S.L.10
Chen, H.K.11
Jee, W.S.S.12
Cameron, K.O.13
Rosati, R.L.14
Brown, T.A.15
Dasilva Jardine, P.16
Thompson, D.D.17
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10
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0035942513
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Bazedoxifene:
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Bazedoxifene: Miller C.P., Collini M.D., Tran B.D., Harris H.A., Kharode Y.P., Marzolf J.T., Moran R.A., Henderson R.A., Bender R.H.W., Unwalla R.J., Greenberger L.M., Yardley J.P., Abou-Gharbia M.A.A., Lyttle C.R., Komm B.S. J. Med. Chem. 44:2001;1654
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Miller, C.P.1
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Marzolf, J.T.6
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Henderson, R.A.8
Bender, R.H.W.9
Unwalla, R.J.10
Greenberger, L.M.11
Yardley, J.P.12
Abou-Gharbia, M.A.A.13
Lyttle, C.R.14
Komm, B.S.15
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11
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0030579801
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Kuiper G.G.J.M., Enmark E., Pelto-Huikko M., Nilsson S., Gustafsson J.A. Proc. Natl. Acad. Sci. U.S.A. 93:1996;5925
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(1996)
Proc. Natl. Acad. Sci. U.S.A.
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Kuiper, G.G.J.M.1
Enmark, E.2
Pelto-Huikko, M.3
Nilsson, S.4
Gustafsson, J.A.5
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13
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11144356286
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Kim S., Wu J.Y., Birzin E.T., Frisch K., Chan W., Pai L.-Y., Yang Y.T., Mosley R.T., Fitzgerald P.M.D., Sharma N., Dahllund J., Thorsell A.-G., DiNinno F., Rohrer S.P., Schaeffer J.M., Hammond M.L. J. Med. Chem. 47:2004;2171
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Kim, S.1
Wu, J.Y.2
Birzin, E.T.3
Frisch, K.4
Chan, W.5
Pai, L.-Y.6
Yang, Y.T.7
Mosley, R.T.8
Fitzgerald, P.M.D.9
Sharma, N.10
Dahllund, J.11
Thorsell, A.-G.12
Dininno, F.13
Rohrer, S.P.14
Schaeffer, J.M.15
Hammond, M.L.16
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14
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11144354858
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Chen H.Y., Kim S., Wu J.Y., Birzin E.T., Chan W., Yang Y.T., DiNinno F., Rohrer S.P., Schaeffer J.M., Hammond M.L. Bioorg. Med. Chem. Lett. 14:2004;2551
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Chen, H.Y.1
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Yang, Y.T.6
Dininno, F.7
Rohrer, S.P.8
Schaeffer, J.M.9
Hammond, M.L.10
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15
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2342467515
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Kim S., Wu J.Y., Chen H.Y., Birzin E.T., Chan W., Pai L.-Y., Yang Y.T., Colwell L., Li S., Dahllund J., DiNinno F., Rohrer S.P., Schaeffer J.M., Hammond M.L. Bioorg. Med. Chem. Lett. 14:2004;2741
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Kim, S.1
Wu, J.Y.2
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Pai, L.-Y.6
Yang, Y.T.7
Colwell, L.8
Li, S.9
Dahllund, J.10
Dininno, F.11
Rohrer, S.P.12
Schaeffer, J.M.13
Hammond, M.L.14
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16
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2942625956
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in press
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Tan, Q.; Birzin, E. T.; Chan, W.; Yang, Y. T.; Pai, L.-Y.; Hayes, E. C.; DaSilva, C. A.; DiNinno, F.; Rohrer, S. P.; Schaeffer, J. M.; Hammond, M. L. Bioorg. Med. Chem. Lett. 2004, 14, in press
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(2004)
Bioorg. Med. Chem. Lett.
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Tan, Q.1
Birzin, E.T.2
Chan, W.3
Yang, Y.T.4
Pai, L.-Y.5
Hayes, E.C.6
Dasilva, C.A.7
Dininno, F.8
Rohrer, S.P.9
Schaeffer, J.M.10
Hammond, M.L.11
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19
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2942574026
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Bromoketone 16 was obtained via α-bromination (THF, PTAB, 0°C to rt, 79%) of the corresponding ketone, which was made according to the method in Ref. [4a, b]
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Bromoketone 16 was obtained via α-bromination (THF, PTAB, 0°C to rt, 79%) of the corresponding ketone, which was made according to the method in Ref. [4a, b]
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