Companion animal physiology and dosage form performance

Advanced Drug Delivery Reviews

Volumn 56, Issue 10, 2004, Pages 1383-1398

  Sutton, Steven C ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United States)

Author keywords

Cat; Controlled release; Dog; Gastrointestinal transit; IVIVC

Indexed keywords

CONTROLLED DRUG DELIVERY; DRUG DOSAGE; MECHANICAL PERMEABILITY; PHYSIOLOGY; SOLUBILITY;

ANATOMY; BILE SALTS;

VETERINARY MEDICINE;

ASCORBIC ACID; BILE SALT; CALCIUM CARBONATE; CALCIUM SALT; CELLULOSE; CHLORAMPHENICOL; CIMETIDINE; GLYCEROL 1 NITRATE; INTESTINE ENZYME; LACTOSE; LACTULOSE; MITOTANE; PALMITIC ACID; PSEUDOEPHEDRINE; XYLOSE;

BREED; CAT; COLON; CONTROLLED RELEASE FORMULATION; DIET RESTRICTION; DOG; DRUG ADSORPTION; DRUG DEGRADATION; DRUG FORMULATION; DRUG PENETRATION; DRUG RELEASE; DRUG SOLUBILITY; EATING HABIT; FEEDING; HUMAN; INTESTINE ABSORPTION; INTESTINE MUCOSA PERMEABILITY; INTESTINE TRANSIT TIME; MEAL; NONHUMAN; OSMOSIS; PRIORITY JOURNAL; REVIEW; STOMACH EMPTYING; STOMACH EROSION; STOMACH PH; TABLET;

EID: 2942521757     PISSN: 0169409X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.addr.2004.02.013     Document Type: Article

References (43)

1. Stevens C.E., Hume I.D. Comparative Physiology of the Vertebrate Digestive System. 2nd edn. 1995;400 Cambridge Univ. Press, New York
2. Johnson L.R. 3rd edn. Physiology of the Gastrointestinal Tract. vol. I:1994;633 Raven Press, New York
3. Brown B.P., Schulze-Delrieu K., Schrier J.E., Abu-Yousef M.M. The configuration of the human gastroduodenal junction in the separate emptying of liquids and solids. Gastroenterology. 105:1993;433-440
4. Code C., Marlett J. The interdigestive myo-electric complex of the stomach and small bowel of dogs. J. Physiol. 246:1975;289-309
5. Johnston K.L., Ballevre O.P., Batt R.M. Use of an orally administered combined sugar solution to evaluate intestinal absorption and permeability in cats. Am. J. Vet. Res. 62:2001;111-118
6. Chiou W.L., Jeong H., Chung S. Evaluation of using the dog as an animal model to study the fraction of oral dose absorbed of 43 drugs in humans. Pharm. Res. 17:2000;135-140
7. Sutton S.C. Use of the dog colon model and a physiologic-pharmacokinetic computer model to simulate controlled release plasma profiles. Proc. Int. Symp. Control. Release Bioact. Mater. 2000;57-58
8. Chandler M., Guilford G., Lawoko C. Radiopaque markers to evaluate gastric emptying and small intestinal transit time in healthy cats. J. Vet. Intern. Med. 11:1997;361-364
9. Chandler M.L., Guilford W.G., Lawoko C.R., Whittem T. Gastric emptying and intestinal transit times of radiopaque markers in cats fed a high-fiber diet with and without low-dose intravenous diazepam. Vet. Radiol. Ultrasound. 40:1999;3-8
10. Fix J.A., Cargill R., Engle K. Controlled gastric emptying: III. Gastric residence time of a nondisintegrating geometric shape in human volunteers. Pharm. Res. 10:1993;1087-1089
11. Ahmed I., Kasraian K. Pharmaceutical challenges in veterinary product development. Adv. Drug Deliv. Rev. 54:2002;871-882
12. Sutton S.C. Animal physiology, drug disposition and dosage form performance. Proc. Int. Symp. Control. Release Bioact. Mater. 2001
13. Watson A. Bioavailability and bioinequivalence of drug formulations in small animals. J. Vet. Pharmacol. Ther. 15:1992;151-159
14. Fleisher D. Nutrient effects on intestinal drug absorption. J. Control. Release. 11:1990;41-49
15. Fleisher D., Li C., Zhou Y., Pao L.H., Karim A. Drug, meal and formulation interactions influencing drug absorption after oral administration: clinical implications. Clin. Pharmacokinet. 36:1999;233-254
16. Ebel J.P., Jay M., Beihn R.M. An in vitro/in vivo correlation for the disintegration and onset of drug release from enteric-coated pellets. Pharm. Res. 10:1993;233-238
17. Digenis G.A., Sandefer E.P., Beihn R.M., Parr A.F. Dual-isotope imaging of neutron-activated erbium-171 and samarium-153 and the in vivo evaluation of a dual-labeled bilayer tablet by gamma scintigraphy. Pharm. Res. 8:1991;1335-1340
18. Borin M.T., Khare S., Beihn R.M., Jay M. The effect of food on gastrointestinal (GI) transit of sustained-release ibuprofen tablets as evaluated by gamma scintigraphy. Pharm. Res. 7:1990;304-307
19. L.A.F. Evans, K.A. Norton, M.J. Puz, S.C. Sutton, Use of gamma scintigraphy as a tool in the development of in vitro and in vivo relationships of compound A for controlled release formulations in dogs, In: American Assoc. for Laboratory. Animal Science National Meeting, 1999, Indianapolis.
20. Zentner G.M., McClelland G.A., Sutton S.C. Controlled porosity solubility- and resin- modulated osmotic drug delivery systems for release of diltiazem hydrochloride. J. Control. Release. 16:1991;237-244
21. McClelland G.A., Sutton S.C., Engle K., Zentner G.M. The solubility modulated osmotic pump: in vitro/in vivo release of diltiazem hydrochloride. Pharm. Res. 8:1991;88-92
22. Gillespie W. Convolution-based approaches for in vitro in vivo correlation modeling. Young D., Devane J., Butler J. In Vitro In Vivo Correlations. 1997;53-65 Plenum, New York
23. Thombre A.G., Appel L.E., Chidlaw M.B., Daugherity P.D., Dumont F., Evans L.A.F., Sutton S.C. Osmotic drug delivery using swellable-core technology. J. Controlled. Release. 94:2004;75-89
24. Basit A.W., Lacey L.F. Colonic metabolism of ranitidine: implications for its delivery and absorption. Int. J. Pharm. 227:2001;157-165
25. Evans L.A.F., Sutton S.C. Canine model to predict colonic microflora degradation and non-specific adsorption of compounds. AAPS Northeastern Regional Discussion Group Mtg. 2003;. Rocky Hill, CT
26. Kararli T. Comparison of the gastrointestinal anatomy, physiology, and biochemistry of humans and commonly used laboratory animals. Biopharm. Drug Dispos. 16:1995;351-380
27. Dressman J.B. Comparison of canine and human gastrointestinal physiology. Pharm. Res. 3:1986;123-131
28. Itoh I. Gastric emptying of indigestible particles and intragastric pH in the beagle dog. Pharmaceutical Chemistry. 1987;161 University of Kansas, Lawrence
29. Youngberg C., Wlodyga J., Schmaltz S., Dressman J. Radiotelemetric determination of gastrointestinal pH in four healthy beagles. Am. J. Vet. Res. 46:1985;1516-1521
30. Oberle E. The influence of the interdigestive migrating myoelectric complex on the gastric emptying of liquids and oral absorption of cimetidine. Pharmaceutics. 1988;396 University of Michigan, Ann Arbor
31. Coupe A., Davis S., Evans D., Wilding I. Correlation of the gastric emptying of nondisintegrating tablets with gastrointestinal motility. Pharm. Res. 8:1991;1281-1285
32. Itoh T., Higuchi T., Gardner C., Caldwell L. Effect of particle size and food on gastric residence time of non-disintegrating solids in beagle dogs. J. Pharm. Pharmacol. 38:1986;801-806
33. Gupta P., Robinson J. Gastric empyting of liquids in the fasted dog. Int. J. Pharm. 43:1988;45-52
34. Miyabayashi T., Morgan J., Atilola M., Muhumuza L. Small intestinal emptying time in normal beagle dogs. Vet. Radiol. 27:1986;164-168
35. Sako K., Mizumoto T., Kajiyama A., Ohmura T. Influence of physical factors in gastrointestinal tract on acetaminophen release from controlled-release tablets in fasted dogs. Int. J. Pharm. 137:1996;225-232
36. Sarr M., Kelly K. Patterns of movement of liquids and solids through canine jejunum. Am. J. Physiol. 239:1980;G497-G503
37. Itoh T. Gastric Emptying of Indigestible Particles and Intragastric pH in the Beagles. 1987;149-161 Department of Pharmaceutical Chemistry, University of Kansas. Chap. 6
38. Mann F., Bollman J. The reaction of the content of the gastro-intestinal tract. J. Am. Med. Assoc. 1930;1722-1724
39. Davis S., Wilding E., Wilding I. Gastrointestinal transit of a matrix tablet formulation: comparison of canine and human data. Int. J. Pharm. 94:1993;235-238
40. Quigley E., Turnberg L. pH of the microclimate lining human gastric and duodenal mucosa in vivo. Gastroenterology. 92:1987;1876-1884
41. Calabrese E. Principles of Animal Extrapolation. 1991;183 Lewis, Chelsea
42. Taylor D., Grundy R., Loveday B. Chronic dog intestinal loop model for studying drug absorption as exemplified by beta-adrenoreceptor blocking agents, atenolol and propranolol. J. Pharm. Sci. 70:1981;516-521
43. Maxwell J., Ferguson A., Watson W. The effect of gastric secretory status on jejunal pH measured by radiotelemetery. Digestion. 4:1971;345-352