Facile synthesis of pyrazolo[1,5-a]pyrimidine derivatives via microwave irradiation and biological activity research

Chinese Journal of Organic Chemistry

Volumn 25, Issue 10, 2005, Pages 1230-1234

  Li, Ming ^a,b   Guo, Wei Si ^a   Wen, Li Rong ^a   Yang, Hua Zheng ^a  

^a QINGDAO UNIVERSITY OF SCIENCE AND TECHNOLOGY   (China)

^b NANKAI UNIVERSITY   (China)

Author keywords

Biological activity; Enaminone; Microwave irradiation; Pyrazolo 1,5 a pyrimidine; Synthesis

Indexed keywords

EID: 29144458233     PISSN: 02532786     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (25)

1. Caddick, S. Tetrahedron 1995, 51, 10403.
2. Galema, S. A. Chem. Soc. Rev. 1997, 26, 233.
3. Gao, Y.; Tu, S. J.; Li, T. J.; Zhang, X. J.; Zhu S. L.; Fang, F.; Shi, D. Q. Synth. Commun. 2004, 34, 1295.
4. Hamrlin, J.; Benhaoua, H.; Kasmi, S. Tetrahedron Lett. 1998, 39(44), 8093.
5. Huang, H.-M.; Yu, H.-T.; Chen, P.-L.; Han, J.; Meng, J.-B. Chin. J. Org. Chem. 2004, 24, 502 (in Chinese).
6. Jeselnik, M.; Varma, R. S.; Polanc, S.; Kocevar, M. Green Chem. 2002, 4, 35.
7. Loupy, A.; Ferreux, L. Tetrahedron 2001, 57, 9199.
8. Wang, J.; Jiang, F.-C. Chin. J. Org. Chem. 2002, 22, 212 (in Chinese).
9. Yoshino, H.; Ueda, N.; Niijima, J.; Sugumi, H. J. Med. Chem. 1992, 35, 2496.
10. Li, J. J.; Anderson, D.; Burton, E. G.; Cogburn, J. N. J. Med. Chem. 1995, 38, 4570.
11. Zoni, F.; Vicini, P. Arch. Pharm. 1998, 331, 219.
12. Senga, K.; Novinson, F.; Wilson, H. R.; Robins, R. K. J. Med. Chem. 1981, 24, 610.
13. Elmoghayer, M. R. H.; Elnagdi, M. H. Arch. Pharm. (Weinheim) 1983, 316, 697.
14. Monte, W. T.; Kleschick, W. A.; Border, J. J. Heterocycl. Chem. 1999, 36, 2183.
15. ElGemeie, G. E. H.; El-Ezbywy, S. E.; Ali, H. A.; Mansour, A. K. Bull Chem. Soc. Jpn. 1994, 67(3), 738.
16. Fathalla, O. A.; Zaki, M. E. A. Indian J. Chem. 1998, 37B, 484.
17. Ammar, Y. A.; El-Sharief, A. M. S.; Zahran, M. A.; El-Said, M. Z.; El-Said, U. H. J. Chem. Res., Synop. 1995, 324.
18. Olivera, R.; SanMartin, R.; Dominguez, E. Tetrahedron Lett. 2000, 41, 4353.
19. Hernandez, S.; SanMartin, R.; Tellitu, I.; Dominguez, E. Org. Lett. 2003, 5(7), 1095.
20. Dawood, K. M.; Kandeel, Z. E.; Farag, A. M. Heteroat. Chem. 1999, 10(5), 417.
21. Dalpozzo, R.; Nino, A. D.; Miele, D.; Procopio, A.; Tagarelli, A.; Bartoli, G. Heteroat. Chem. 2000, 11(1), 1.
22. El-Taweei, F. M. A. A; Elangdi, M. H. J. Heterocycl. Chem. 2001, 38, 981.
23. Li, M.; Guo, W.-S.; Wen, L.-R.; Zhong, H.-M.; Yang, H.-Z. Acta Chim. Sinica 2005, 63, 855 (in Chinese).
24. Lu, R.-J.; Yang, H.-Z.; Zhao, G.-F.; Liu, H.-Y. Chem. J. Chin. Univ. 1996, 17, 1231 (in Chinese).
25. Tseng, S. S.; Epstein, J. W.; Brabander, H. J.; Francisco, G. J. Heterocycl. Chem. 1987, 24, 837.