Alternative methods for labeling the 5-HT1A receptor agonist, 1-[2-(4-fluorobenzoylamino)ethyl]-4-(7-methoxynaphthyl)piperazine (S14506), with carbon-11 or fluorine-18

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 48, Issue 13, 2005, Pages 971-981

  Lu, Shui Yu ^a   Hong, Jinsoo ^a   Musachio, John L ^a   Chin, Frederick T ^a   Vermeulen, Erik S ^b   Wikström, Håkan V ^b   Pike, Victor W ^a  

^a NATIONAL INSTITUTES OF HEALTH   (United States)

^b UNIVERSITY OF GRONINGEN   (Netherlands)

Author keywords

5 HT1A; Agonist; Carbon 11; Fluorine 18; Microwave; Radioligand

Indexed keywords

CARBON; DIMETHYLFORMAMIDE; FLUORIDATION; FLUORINE; POSITRONS;

5-HT1A; AGONIST; CARBON-11; FLUORINE-18; LABELINGS; PROSPECTIVES; RADIOCHEMICAL YIELD; RADIOLIGANDS; RADIOSYNTHESIS; SPECIFIC ACTIVITY;

POSITRON EMISSION TOMOGRAPHY;

1 [2 (4 FLUOROBENZAMIDO)ETHYL] 4 (7 METHOXY 1 NAPHTHYL)PIPERAZINE; CARBON 11; FLUORINE 18; RADIOLIGAND; SEROTONIN 1A AGONIST;

ARTICLE; CHEMICAL STRUCTURE; CYCLOTRON; FLUORIDATION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOTOPE LABELING; MICROWAVE IRRADIATION; POSITRON EMISSION TOMOGRAPHY; PROTON NUCLEAR MAGNETIC RESONANCE; RADIOCHEMISTRY; SEROTONINERGIC SYSTEM; SYNTHESIS; TEMPERATURE SENSITIVITY;

EID: 28944451492     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/jlcr.1009     Document Type: Article

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