Compatibility studies between ibuprofen or ketoprofen with cellulose ether polymer mixtures using thermal analysis

Drug Development and Industrial Pharmacy

Volumn 31, Issue 10, 2005, Pages 943-949

  Vueba, M L ^a   Veiga, F ^a   Sousa, J J ^a   Pina, Maria Eugénia ^a  

^a UNIVERSITY OF COIMBRA   (Portugal)

Author keywords

Cellulose ether derivatives; Drug polymer interaction; DSC; Ibuprofen; Ketoprofen; Thermal analysis

Indexed keywords

CELLULOSE; IBUPROFEN; KETOPROFEN; METHYLCELLULOSE; POLYMER;

ARTICLE; BIOAVAILABILITY; CONTROLLED DRUG RELEASE; DIFFERENTIAL SCANNING CALORIMETRY; EVALUATION; SOLID; THERMAL ANALYSIS;

EID: 28744440137     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.1080/03639040500306153     Document Type: Article

References (26)

1. Alvarez-Lorenzo, C., Gómez-Amoza, J. L., Martínez-Pacheco, R., Souto, C., & Concheiro, A. (2000). Interactions between hydroxypropylcelluloses and vapour/liquid water. European Journal of Pharmaceutics and Biopharmaceutics, 50, 307-318.
2. Botha, S. A., & Lotter, A. P. (1989). Compatibility study between ketoprofen and tablet excipients using differential scanning calorimetry. Drug Development and Industrial Pharmacy, 15(3), 415-426.
3. Budavári, Z., Zelkó, I., Rácz, I., & Marton, S. (1999). Compatibility study between folic acid, vitamin B6, and tablet excipients using differential scanning calorimetry. Pharmazie, 54(11), 861-862.
4. Byrn, S. R., Pfeiffer, R. R., Stephenson, G., Grant, D. J. W., & Gleason, W. B. (1994). Solid-state pharmaceutical chemistry. Chemistry of Materials, 6, 1148-1158.
5. De Villiers, M. M., Liebenberg, W., Malan, S. F., & Gerber, J. J. (1999). The dissolution and complexing properties of ibuprofen and ketoprofen when mixed with N-methylglucamine. Drug Development and Industrial Pharmacy, 25(8), 967-972.
6. Ebube, N. K., & Jones, A. B. (2004). Sustained release of acetaminophen from a heterogeneous mixture of two hydrophilic non-ionic cellulose ether polymers. International Journal of Pharmaceutics, 272, 19-27.
7. Ford, J. L. (1999). Thermal analysis of hydroxypropylmethylcellulose and methylcellulose: powders, gels and matrix tablets. International Journal of Pharmaceutics, 179, 209-228.
8. Gómez-Carracedo, A., Alvarez-Lorenzo, C., Gómez-Amoza, J. L., & Concheiro, A. (2003). Chemical structure and glass transition temperature of non-ionic cellulose ethers DSC, TMDSC®. Oscillatory rheometry study. Journal of Thermal Analysis and Calorimetry, 73, 587-596.
9. Gordon, R. E., VanKoevering, C. L., & Reits, D. J. (1984). Utilization of differential scanning calorimetry in the compatibility screening of ibuprofen with the stearate lubricants and construction of phase diagrams. International Journal of Pharmaceutics, 21, 99-105.
10. Hatakeyama, H., & Hatakeyama, T. (1998). Interaction between water and hydrophilic polymers. Thermochimica Acta, 308, 3-22.
11. Higginis, J. D., Gilmor, T. P., Martellucci, S. A., Bruce, R. D., & Brittain, H. G. (2001). Ibuprofen. In: K. Florey (Ed.), Analytical Profiles of Drug Substances. Vol. 27. New York: Academic Press, 265-299.
12. Holgado, M. A., Fernández-Arévalo, M., Ginés, J. M., Caraballo, I., & Rabasco, A. M. (1995). Compatibility study between carteolol hydrochloride and tablet excipients using differential scanning calorimetry and hot stage microscopy. Pharmazie, 50(H.3), 195-198.
13. Kumar, V., & Banker, G. S. (1993). Chemically modified cellulosic polymers. Drug Development and Industrial Pharmacy, 19, 1-31.
14. Liversidge, G. G. (1989). Ketoprofen. In: K. Florey (Ed.), Analytical Profiles of Drug Substances. Vol. 10. New York: Academic Press, 443-471.
15. McPhillips, H., Craig, D. Q. M., Royall, P. G., & Hill, V. L. (1999). Characterization of the glass transition of HPMC using modulated temperature differential scanning calorimetry. International Journal of Pharmaceutics, 180, 83-90.
16. Mura, P., Manderioli, A., Bramanti, G., Furlanetto, S., & Pinzauti, S. (1995). Utilization of differential scanning calorimetry as a screening technique to determine the compatibility of ketoprofen with excipients. International Journal of Pharmaceutics, 119, 71-79.
17. Mura, P., Bettinetti, G. P., Manderioli, A., Faucci, M. T., Bramanti, G., & Sorrenti, S. (1998). Interactions of ketoprofen and ibuprofen with β-cyclodextrins in solution and in the solid. International Journal of Pharmaceutics, 166, 189-203.
18. Mura, P., Faucci, M. T., Parrini, P. L., Furlanetto, S., & Pinzauti, S. (1999). Influence of the preparation method on the physicochemical properties of ketoprofen-cyclodextrin binary systems. International Journal of Pharmaceutics, 179, 117-128.
19. Mura, P., Faucci, M. T., & Parrini, P. L. (2001). Effects of grinding with microcrystalline cellulose and cyclodextrins on the ketoprofen physicochemical properties. Drug Development and Industrial Pharmacy, 27(2), 119-128.
20. Nokhodchi, A., Ford, J. L., Rowe, P. H., & Rubinstein, M. H. (1996a). The influence of moisture content on the consolidation properties of hydroxypropylmethylcellulose K4M (HPMC 2208). Journal of Pharmacy and Pharmacology, 48, 1116-1121.
21. Nokhodchi, A., Ford, J. L., Rowe, P. H., & Rubinstein, M. H. (1996b). The effect of moisture on the Hecker and energy analysis of hydroxypropylmethylcellulose 2208 (HPMC K4M). Journal of Pharmacy and Pharmacology, 48, 1122-1127.
22. Nokhodchi, A., Ford, J. L., & Rubinstein, M. H. (1997). Studies on the interaction between water and (hydroxypropyl)methylcellulose. Journal of Pharmaceutical Sciences, 86(5), 608-615.
23. Smith, A. (1982). Use of thermal analysis in predicting drug-excipient interactions. Analytical Proceedings, 559-561.
24. Van Dooren, A. A., & Duphar, B. V. (1983). Design for drug-excipient interaction studies. Drug Development and Industrial Pharmacy, 9, 43-45.
25. Verma, R. K., & Garg, S. (2004). Compatibility studies between isosorbide mononitrate and selected excipients used in the development of extended release formulations. Journal of Pharmaceutical and Biomedical Analysis, 35(19), 449-458.
26. Vueba, M. I., Batista de Carvalho, L. A. E., Veiga, F., Sousa, J. J., & Pina, M. E. (2004). Influence of cellulose ether polymers on ketoprofen release from hydrophilic matrix tablets. European Journal of Pharmaceutics and Biopharmaceutics, 58, 51-59.