The esterase-inhibiting activity and toxicity of O,O-dialkyl S-ethoxycarbonylbromomethylthiophosphates

Russian Journal of Bioorganic Chemistry

Volumn 25, Issue 1, 1999, Pages 6-10

  Makhaeva, G F ^a   Yankovskaya, V L ^a   Kovaleva, N V ^a   Fetisov, V I ^a   Malygin, V V ^a   Torgaseva, N A ^b   Khaskin, B A ^b  

^a INSTITUTE OF PHYSIOLOGICALLY ACTIVE COMPOUNDS   (Russian Federation)

^b Res Inst of Plant Protect Chem   (Russian Federation)

Author keywords

Acetylcholinesterase; Acute toxicity; Butyryl cholinesterase; Carboxyl esterase; Enzyme inhibition; O,O dialkyl S ethoxycarbonylbromomethylthiophosphates; Quantitative analysis; Structure enzyme inhibiting activity

Indexed keywords

EID: 27544496048     PISSN: 10681620     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (24)

1. Kagan, Yu.S., Toksikologiya fosfororganicheskikh pestitsidov (Toxicology of Organophosphorus Pesticides), Moscow: Meditsyna, 1977.
2. Rozengart, V.I. and Sherstobitov, O.E., Izbiratel'naya toksichnost' fosfororganicheskikh insektoakaritsidov (Selective Toxicity of Organophosphorus Insecticides and Acaricides), Leningrad: Nauka, 1978.
3. Matsumura, F., Toxicology of Insecticides, New York: Plenum, 1985.
4. Makhaeva, G.F., Veselova, V.L., Mastryukova, T.A., Shipov, A.E., Zhdanova, G.V., and Kabachnik, M.I., Bioorg. Khim., 1983, vol. 9, pp. 920-925.
5. Makhaeva, G.F., Yankovskaya, V.L., Odoeva, G.A., Shestakova, N.N., Khovanskikh, A.E, Mastryukova, T.A., Shipov, A.E., Zhdanova, G.V., and Kabachnik, M.I., Bioorg. Khim., 1985, vol. 11, pp. 957-962.
6. Fonnum, F., Sterri, S.H., Aas, P., and Johnsen, H., Fundam. Appl. Toxicol., 1985, vol. 5, pp. 29-38.
7. Russel, R.W. and Overstreet, D.H., Progress in Neurobiology, 1987, vol. 28, pp. 97-129.
8. Makhaeva, G.F., Fetisov, V.I., Sokolov, V.B., Yankovskaya, V.L., Goreva, T.V., Malygin, V.V., Beznosko, B.K., Galenko, T.G., Kolomiets, A.F., and Martynov, I.V., Bioorg. Khim., 1987, vol. 13, pp. 33-37.
9. Makhaeva, G.F., Yankovskaya, V.L., Kochetova, L.M., Beznosko, B.K., Sokolpv, V.B., Brel', V.K., Malygin, V.V., and Martynov, I.V., Fiziol. Akt. Veshchestva, 1989, vol. 21, pp. 68-74.
10. Malygin, V. and Makhaeva, G., Toxicol. Lett., 1995, vol. 78, Suppl. 1, p. 56.
11. Khaskin, B.A., Makhaeva, G.F., Torgasheva, N.A., Ishmuratov, A.S., Yankovskaya, V.L., Fetisov, V.I., Malygin, V.V., and Martynov, I.V., Izv. Akad. Nauk SSSR, Ser. Khim., 1989, no. 12, pp. 2741-2746.
12. Khaskin, B.A., Torgasheva, N.A., and Ishmuratov, A.S., Zh. Obshch. Khim., 1991, vol. 61, pp. 1090-1095.
13. Makhaeva, G.F., Yankovskaya, V.L., Kovaleva, N.V., Fetisov, V.I., Malygin, V.V., Torgasheva, N.A., and Khaskin, B.A., Bioorg. Khim., 1999, vol. 25, pp. 3-7.
14. Fetisov, V.I., Makhaeva, G.F., Loshadkin, N.A., Martynov, I.V., and Khaskin, B.A., Bioorg. Khim., 1984, vol. 10, pp. 1353-1358.
15. Hansch, C. and Leo, A., Substituent Constants for Correlation Analysis in Chemistry and Biology, New York: Wiley, 1979.
16. Kubinyi, H., Arzneimittel-Forsch., 1976, vol. 26, pp. 1991-1997.
17. Kabachnik, M.I., Brestkin, A.P., Godovikov, N.N., Michelson, M.J., Rosengart, E.V., and Rosengart, V.I., Pharmacol. Rev., 1970, vol. 22, pp. 355-388.
18. Tailor, P., Radic, Z., Hosea, N.A., Camp, S., Marchot, P., and Berman, H.A., Toxicol. Lett., 1995, vol. 82/83, pp. 453-458.
19. Makhaeva, G.F., Malygin, V.V., Yakubov, Sh.M., and Gorbunov, S.M., Khim.-Farm. Zh., 1994, vol. 28, pp. 6-9.
20. Makhaeva, G.F., Malygin, V.V., Yakubov, Sh.M., and Gorbunov, S.M., Khim.-Farm. Zh., 1994, vol. 28, pp. 14-18.
21. Plyamovatyi, A.Kh., Vandyukova, I.I., Shagidullin, R.R., Makhaeva, G.F., and Malygin, V.V., Khim.-Farm. Zh., 1997, vol. 31, pp. 38-43.
22. Yakovlev, V.A., Kinetika fermentativnogo kataliza (Kinetics of Enzymic Catalysis), Moscow: Nauka, 1965, pp. 115-117.
23. L'vovskii, E.N., Statisticheskie metody postroeniya empiricheskikh formul (Statistical Methods for Obtaining Empirical Formulas), Moscow: Vysshaya Shkola, 1988.
24. Litchfield, J.T. and Wilcoxon, F., J. Pharm. Exp. Therap., 1949, vol. 96, pp. 99-113.