A convenient synthesis of diastereomeric synthons: Ethyl 3-methyl-1,2,3,4-tetrahydroisoquinoline-1-acetates by direct and reverse substituent introductions

Heterocycles

Volumn 43, Issue 8, 1996, Pages 1605-1606

  Fülop, Ferenc ^a   Tari, János ^a   Bernáth, Gábor ^a   Sohár, Pál ^b  

^a UNIVERSITY OF SZEGED   (Hungary)

^b EÖTVÖS LORÁND UNIVERSITY   (Hungary)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 2742528821     PISSN: 03855414     EISSN: None     Source Type: Journal    
DOI: 10.3987/com-96-7509     Document Type: Article

References (13)

1. F. Fülöp, H. Wamhoff, and P. Sohár, Synthesis, 1995, 863.
2. B. Lal, R. M. Gidwani, and N. J. deSouza, J. Org. Chem., 1990, 55, 5117.
3. J. E. Sounes, B. K. Diocee, W. Martin, and S. A. Moodie, Biochem. J., 1990, 266, 127.
4. J. Kóbor, P. Sohár, and F. Fülöp, Tetrahedron, 1994, 50, 4873.
5. F. Fülöp, E. Semega, G. Bernáth, and P. Sohár, J. Heterocycl. Chem., 1990, 27, 957.
6. J. C. Pelletier and M. P. Cava, Synthesis, 1987, 474.
7. J. C, Pelletier and M. P. Cava, J. Org. Chem., 1987, 52, 616, and references cited therein.
8. W. S. Ide and J. S. Buck, J. Am. Chem. Soc., 1940, 62, 425.
9. E. R. Shepard, J. F. Noth, H. D. Porter, and C. K. Simmans, J. Am. Chem. Soc., 1952, 74, 4611.
10. 3), 111.5 (5-C), 115.8 (8-C), 116.9 (8a-C), 132.5 (4a-C), 149.4 (7-C), 157.6 (6-C), 163.4 (1-C).
11. 2), 108.0, 110.5, 110.7 (5,8,1′-C), 121.3 (8a-C), 129.6 (4a-C), 147.8 (7-C), 151.1 (6-C), 156.4 (1-C), 171.2 (C=O).
12. 3), 109.3 (8-C), 111.5 (5-C), 127.0 (8a-C), 129.2 (4a-C), 147.3, 147.7 (6,7-C), 172.3 (C=O).
13. 2), 108.1 (8-C), 111.6 (5-C), 128.1. 129.2 (4a,8a-C), 147.2, 147.5 (6,7-C), 172.5 (C=O).