QSAR study on carbonic anhydrase inhibitors: Water-soluble sulfonamides incorporating β-alanyl moieties, possessing long lasting-intra ocular pressure lowering properties - A molecular connectivity approach

European Journal of Medicinal Chemistry

Volumn 40, Issue 10, 2005, Pages 1002-1012

  Agrawal, Vijay K ^a   Banerji, Meghna ^a   Gupta, Madhu ^b   Singh, Jyoti ^a   Khadikar, Padmakar V ^c   Supuran, Claudiu T ^d  

^a A P S UNIVERSITY   (India)

^b MMH College   (India)

^c Laxmi Pest and Fumigation Pvt Ltd   (India)

^d UNIVERSITY OF FLORENCE   (Italy)

Author keywords

Carbonic anhydrase inhibitor; Molecular connectivity index; QSAR; Regression analysis; Topological index

Indexed keywords

BETA ALANINE; CARBONATE DEHYDRATASE INHIBITOR; ISOENZYME; SULFONAMIDE; WATER;

ARTICLE; CYTOSOL; INTRAOCULAR PRESSURE; MEMBRANE; QUANTITATIVE STRUCTURE ACTIVITY RELATION; REGRESSION ANALYSIS; STATISTICAL ANALYSIS;

ALANINE; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; HUMANS; INTRAOCULAR PRESSURE; MOLECULAR STRUCTURE; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; SOLUBILITY; SULFONAMIDES; WATER;

EID: 26444436908     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2005.04.006     Document Type: Article

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