The synthesis and antimicrobial evaluation of a new series of isoxazolinyl oxazolidinones

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 12, 2004, Pages 3069-3072

  Weidner Wells, Michele A ^a   Werblood, Harvey M ^a   Goldschmidt, Raul ^a   Bush, Karen ^a   Foleno, Barbara D ^a   Hilliard, Jamese J ^a   Melton, John ^a   Wira, Ellyn ^a   Macielag, Mark J ^a  

^a Johnson Johnson Pharmaceutical R D   (United States)

Author keywords

Antibacterial; Oxazolidinone; Resistant bacteria

Indexed keywords

ANTIINFECTIVE AGENT; ISOXAZOLE DERIVATIVE; LINEZOLID; NITRILE; OXAZOLIDINONE DERIVATIVE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL INFECTION; CONTROLLED STUDY; CYCLOADDITION; DRUG SCREENING; DRUG SENSITIVITY; DRUG SYNTHESIS; FEMALE; GRAM POSITIVE BACTERIUM; IN VITRO STUDY; MOUSE; NONHUMAN; REACTION ANALYSIS; SEPTICEMIA; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTI-BACTERIAL AGENTS; DRUG EVALUATION, PRECLINICAL; FEMALE; ISOXAZOLES; MICE; MICROBIAL SENSITIVITY TESTS; OXAZOLIDINONES;

POSIBACTERIA;

EID: 2442526307     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.04.037     Document Type: Article

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