Synthesis and evaluation of bifunctional nitrocatechol inhibitors of pig liver catechol-O-methyltransferase

Bioorganic and Medicinal Chemistry

Volumn 13, Issue 20, 2005, Pages 5740-5749

  Bailey, Karl ^a   Tan, Eng Wui ^a  

^a UNIVERSITY OF OTAGO   (New Zealand)

Author keywords

Bifunctional; Catechol O methyltransferase; Enzyme inhibitors

Indexed keywords

CATECHOL METHYLTRANSFERASE INHIBITOR;

ANALYTIC METHOD; ANIMAL TISSUE; ARTICLE; CHEMICAL BOND; CONTROLLED STUDY; DRUG SCREENING; DRUG SYNTHESIS; IN VITRO STUDY; LIVER; NONHUMAN; STATISTICAL SIGNIFICANCE; SWINE;

ANIMALS; CATECHOLS; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; LIVER; MAGNETIC RESONANCE SPECTROSCOPY; NITRO COMPOUNDS; SWINE;

SUS SCROFA;

EID: 24344491784     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.05.069     Document Type: Article

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