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Volumn 3, Issue 2, 2002, Pages

Flurbiprofen release from Eudragrit RS and RL aqueous nanosuspensions: A kinetic study by DSC and dialysis experiments

Author keywords

Differential Scanning Calorimetry (DSC); Dimyristoylphosphatidylcholine (DMPC); Eudragit; Flurbiprofen (FLU); Membrane Model; Membrane permeation; Nanosuspensions; Phosphatidylcholine

Indexed keywords

DIMYRISTOYLPHOSPHATIDYLCHOLINE; EUDRAGIT; EUDRAGIT RL100; EUDRAGIT RS; EUDRAGIT RS100; FLURBIPROFEN; LIPOSOME; SOLVENT; ACRYLIC ACID RESIN; DRUG CARRIER;

EID: 23144464360     PISSN: 15309932     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (25)

References (36)
  • 2
    • 0003611227 scopus 로고
    • Recent advances in microencapsulation of drugs to obtain reduced gastric irritation
    • Donbrow M, ed. Boca Raton, FL: CRC Press
    • Bakan JA, Powell TC, Szotak PS. Recent advances in microencapsulation of drugs to obtain reduced gastric irritation. In: Donbrow M, ed. Microcapsules and Nanoparticles in Medicine Pharmacy. Boca Raton, FL: CRC Press; 1991:183-192.
    • (1991) Microcapsules and Nanoparticles in Medicine Pharmacy , pp. 183-192
    • Bakan, J.A.1    Powell, T.C.2    Szotak, P.S.3
  • 3
    • 0022445026 scopus 로고
    • Preparation and dissolution pattern of Eudragit RS microcapsules containing Ketoprofen
    • Kawata M, Nakamura M, Goto T, Ayoama T. Preparation and dissolution pattern of Eudragit RS microcapsules containing Ketoprofen. Chem Pharm Bull. 1968;34: 2618-2623.
    • (1968) Chem. Pharm. Bull. , vol.34 , pp. 2618-2623
    • Kawata, M.1    Nakamura, M.2    Goto, T.3    Ayoama, T.4
  • 4
    • 0022826259 scopus 로고
    • Eudragit RS and RL (acrylic resins) micro-capsules as pH insensitive and sustained release preparations of ketoprofen
    • Goto S, Kawata M, Nakamura M, Maekauwa K, Ayoama T. Eudragit RS and RL (acrylic resins) micro-capsules as pH insensitive and sustained release preparations of ketoprofen. J Microencapsulation. 1986;3:293-304.
    • (1986) J. Microencapsulation , vol.3 , pp. 293-304
    • Goto, S.1    Kawata, M.2    Nakamura, M.3    Maekauwa, K.4    Ayoama, T.5
  • 5
    • 0024594727 scopus 로고
    • Preparation of prolonged-release spherical micromatrix of ibuprofen with acrylic polymer by the emulsion solvent diffusion method for improving bioavailability
    • Kawashima Y, Niwa T, Handa T, Takeuchi H, Iwamoto T, Ito Y. Preparation of prolonged-release spherical micromatrix of ibuprofen with acrylic polymer by the emulsion solvent diffusion method for improving bioavailability. Chem Pharm Bull. 1989;37:425-429.
    • (1989) Chem. Pharm. Bull. , vol.37 , pp. 425-429
    • Kawashima, Y.1    Niwa, T.2    Handa, T.3    Takeuchi, H.4    Iwamoto, T.5    Ito, Y.6
  • 6
    • 0025867170 scopus 로고
    • Preparation and characterization of a new controlled release ibuprofen suspension for improving suspendability
    • Kawashima Y, Niwa T, Handa T, Takeuchi H, Ito Y. Preparation and characterization of a new controlled release ibuprofen suspension for improving suspendability. Int J Pharm. 1991;75:25-36.
    • (1991) Int. J. Pharm. , vol.75 , pp. 25-36
    • Kawashima, Y.1    Niwa, T.2    Handa, T.3    Takeuchi, H.4    Ito, Y.5
  • 7
    • 0026575166 scopus 로고
    • Control of prolonged drug release and compression properties of ibuprofen microsponges with acrylic polymer; Eudragit RS, changing their intrapartical porosity
    • Kawashima Y, Toshiyuki H, Takeuchi H, Hino T, Ito Y. Control of prolonged drug release and compression properties of ibuprofen microsponges with acrylic polymer; Eudragit RS, changing their intrapartical porosity. Chem Pharm Bull. 1992;40:196-201.
    • (1992) Chem. Pharm. Bull. , vol.40 , pp. 196-201
    • Kawashima, Y.1    Toshiyuki, H.2    Takeuchi, H.3    Hino, T.4    Ito, Y.5
  • 8
    • 0031544835 scopus 로고    scopus 로고
    • Properties of Tolmetin-loaded Eudragit RL100 and RS100 microparticles prepared by different techniques
    • Pignatello R, Vandelli MA, Giunchedi P, Puglisi G. Properties of Tolmetin-loaded Eudragit RL100 and RS100 microparticles prepared by different techniques. STP Pharma Sci. 1997;7:148-157.
    • (1997) STP Pharma. Sci. , vol.7 , pp. 148-157
    • Pignatello, R.1    Vandelli, M.A.2    Giunchedi, P.3    Puglisi, G.4
  • 9
    • 0032900521 scopus 로고    scopus 로고
    • Interaction of two Diclofenac acid salts with copolymers of ammoniomethacrylate: Effect of additives and release profiles
    • Khalil E, Sallam A. Interaction of two Diclofenac acid salts with copolymers of ammoniomethacrylate: effect of additives and release profiles. Drug Dev Ind Pharmacy. 1999;25:419-427.
    • (1999) Drug Dev. Ind. Pharmacy , vol.25 , pp. 419-427
    • Khalil, E.1    Sallam, A.2
  • 10
    • 0033844401 scopus 로고    scopus 로고
    • The effect of pre-operative topical Flurbiprofen or Diclofenac on pupil dilatation
    • Thaller VT, Kulshrestha MK, Bell K. The effect of pre-operative topical Flurbiprofen or Diclofenac on pupil dilatation. Eye. 2000;14:642-645.
    • (2000) Eye , vol.14 , pp. 642-645
    • Thaller, V.T.1    Kulshrestha, M.K.2    Bell, K.3
  • 11
    • 0025856637 scopus 로고
    • Nuclear magnetic resonance and differential scanning calorimetry as tools for studying drug-membrane interactions
    • Seydel JK. Nuclear magnetic resonance and differential scanning calorimetry as tools for studying drug-membrane interactions. Trends Pharmacol Sci. 1991;12:368-371.
    • (1991) Trends Pharmacol. Sci. , vol.12 , pp. 368-371
    • Seydel, J.K.1
  • 12
    • 0002629145 scopus 로고
    • Control of membrane fusion by divalent cations, phospholipid headgroups and proteins
    • Conti F, Blumberg WE, De Gier J, Pocciari F, eds. New York, NY: Plenum Press
    • Duzgunes N, Wilschut J, Papahadjopoulos D. Control of membrane fusion by divalent cations, phospholipid headgroups and proteins. In: Conti F, Blumberg WE, De Gier J, Pocciari F, eds. Physical Methods on Biological Membranes and their Model Systems. New York, NY: Plenum Press; 1985:193-218.
    • (1985) Physical Methods on Biological Membranes and Their Model Systems , pp. 193-218
    • Duzgunes, N.1    Wilschut, J.2    Papahadjopoulos, D.3
  • 13
    • 0003893817 scopus 로고
    • Mobility of the lipid and protein components of biological membranes
    • New York, NY: Wiley and Sons
    • Houslay MD, Stanley KK. Mobility of the lipid and protein components of biological membranes. In: Dynamics of Biological Membranes. New York, NY: Wiley and Sons; 1983:40-91.
    • (1983) Dynamics of Biological Membranes , pp. 40-91
    • Houslay, M.D.1    Stanley, K.K.2
  • 14
    • 0025981964 scopus 로고
    • On the reversibility of the phase transitions in lipid-water systems
    • Tenchov B. On the reversibility of the phase transitions in lipid-water systems. Chem Phys Lipids. 1991;57:165-177.
    • (1991) Chem. Phys. Lipids , vol.57 , pp. 165-177
    • Tenchov, B.1
  • 15
    • 0002182090 scopus 로고    scopus 로고
    • Physical characterization of liposomes for understanding structure-function relationships in biological membranes
    • Barenholzand Y, Lasic DD, eds. Boca Raton, FL:CRC Press
    • Marsh D. Physical characterization of liposomes for understanding structure-function relationships in biological membranes. In: Barenholzand Y, Lasic DD, eds. Nonmedical Applications of Liposomes. Boca Raton, FL:CRC Press; 1996:1-16.
    • (1996) Nonmedical Applications of Liposomes , pp. 1-16
    • Marsh, D.1
  • 16
    • 0002134199 scopus 로고
    • Differential scanning calorimetry of liposomes
    • Knight CG, ed. Amsterdam, The Netherlands: Elsevier/North-Holland Biomedical Press
    • Mabrey-Gaud S. Differential scanning calorimetry of liposomes. In: Knight CG, ed. Liposomes: From Physical Structure to Therapeutic Applications. Amsterdam, The Netherlands: Elsevier/North-Holland Biomedical Press; 1981:105-138.
    • (1981) Liposomes: From Physical Structure to Therapeutic Applications , pp. 105-138
    • Mabrey-Gaud, S.1
  • 17
    • 0001989286 scopus 로고
    • Calorimetric studies of model and natural biomembranes
    • Chapman D, ed. London, England: MacMillan Press
    • Bach D. Calorimetric studies of model and natural biomembranes. In: Chapman D, ed. Biomembrane Structure and Function. London, England: MacMillan Press; 1984:1-41.
    • (1984) Biomembrane Structure and Function , pp. 1-41
    • Bach, D.1
  • 18
    • 0026096905 scopus 로고
    • Thermotropic properties of phospholipid analogues
    • Silvius JR. Thermotropic properties of phospholipid analogues. Chem Phys Lipids. 1991;57:241-252.
    • (1991) Chem. Phys. Lipids , vol.57 , pp. 241-252
    • Silvius, J.R.1
  • 19
    • 0017397725 scopus 로고
    • Effect of small molecules on the Dipalmitoyllecithin liposomial bilayer: III Phase transition in lipid bilayer
    • Jain MK, Wu NM. Effect of small molecules on the Dipalmitoyllecithin liposomial bilayer: III Phase transition in lipid bilayer. J Membrane Biol. 1977;34:151-201.
    • (1977) J. Membrane Biol. , vol.34 , pp. 151-201
    • Jain, M.K.1    Wu, N.M.2
  • 20
    • 0003129716 scopus 로고
    • Order and dynamics in bilayers
    • Jain MK, ed. New York, NY: Wiley and Sons
    • Jain MK. Order and dynamics in bilayers. In: Jain MK, ed. Introduction to biological membranes. New York, NY: Wiley and Sons; 1988:122-165.
    • (1988) Introduction to Biological Membranes , pp. 122-165
    • Jain, M.K.1
  • 21
    • 0024308410 scopus 로고
    • Calorimetric studies of the interaction of 4-Biphenylacetic acid and its β inclusion compound with lipid model membrane
    • Castelli F, Puglisi G, Pignatello R, Gurrieri S. Calorimetric studies of the interaction of 4-Biphenylacetic acid and its β inclusion compound with lipid model membrane. Int J Pharm. 1989; 52:115-121.
    • (1989) Int. J. Pharm. , vol.52 , pp. 115-121
    • Castelli, F.1    Puglisi, G.2    Pignatello, R.3    Gurrieri, S.4
  • 22
    • 0026084947 scopus 로고
    • Effects of small organic molecules on phospholipid phase transitions
    • Lohner K. Effects of small organic molecules on phospholipid phase transitions. Chem Phys Lipids. 1991;57:341-362.
    • (1991) Chem. Phys. Lipids , vol.57 , pp. 341-362
    • Lohner, K.1
  • 23
    • 0032053915 scopus 로고    scopus 로고
    • Modeling specific heat transient anomalies during permeation of liposomes by water-soluble substances
    • Raudino A, Castelli F. Modeling specific heat transient anomalies during permeation of liposomes by water-soluble substances. J Coll Interf Sci. 1998;200: 52-58.
    • (1998) J. Coll. Interf. Sci. , vol.200 , pp. 52-58
    • Raudino, A.1    Castelli, F.2
  • 24
    • 0030007603 scopus 로고    scopus 로고
    • Effect of molecular weight and storage times on Tolmetin release from poly-D,L-lactide microspheres to lipid model membrane: A calorimetric study
    • Castelli F, Conti B, Puglisi G, Conte U. Effect of molecular weight and storage times on Tolmetin release from poly-D,L-lactide microspheres to lipid model membrane: a calorimetric study. J Controlled Rel. 1996;40:277-284.
    • (1996) J. Controlled Rel. , vol.40 , pp. 277-284
    • Castelli, F.1    Conti, B.2    Puglisi, G.3    Conte, U.4
  • 25
    • 0031018101 scopus 로고    scopus 로고
    • Effect of pH on the transfer kinetics of an anti-inflammatory drug from polyaspartamide hydrogels to lipid model membrane
    • Castelli F, Pitarresi G, Tomarchio V, Giammona G. Effect of pH on the transfer kinetics of an anti-inflammatory drug from polyaspartamide hydrogels to lipid model membrane. J Controlled Rel. 1997;45:103-111.
    • (1997) J. Controlled Rel. , vol.45 , pp. 103-111
    • Castelli, F.1    Pitarresi, G.2    Tomarchio, V.3    Giammona, G.4
  • 26
    • 0032962760 scopus 로고    scopus 로고
    • Differences between Coumaric and Cinnamic acids in membrane permeation as evidenced by time-dependent calorimetry
    • Castelli F, Uccella N, Saija A, Trombetta D. Differences between Coumaric and Cinnamic acids in membrane permeation as evidenced by time-dependent calorimetry. J Agr Food Chem. 1999;47:991-995.
    • (1999) J. Agr. Food Chem. , vol.47 , pp. 991-995
    • Castelli, F.1    Uccella, N.2    Saija, A.3    Trombetta, D.4
  • 27
    • 0033998157 scopus 로고    scopus 로고
    • Influence of different parameters on drug release from hydrogel systems to biomembrane model: Evaluation by differential scanning calorimetry technique
    • Castelli F, Pitarresi G, Giammona G. Influence of different parameters on drug release from hydrogel systems to biomembrane model: evaluation by differential scanning calorimetry technique. Biomaterials. 2000;21:821-833.
    • (2000) Biomaterials , vol.21 , pp. 821-833
    • Castelli, F.1    Pitarresi, G.2    Giammona, G.3
  • 28
    • 0035999781 scopus 로고    scopus 로고
    • Flurbiprofen-loaded acrylate polymer nano-suspensions for ophthalmic application
    • Pignatello R, Spedalieri G, Bucolo C, Maltese A, Puglisi G. Flurbiprofen-loaded acrylate polymer nano-suspensions for ophthalmic application. Biomaterials. 2002;15:3247-3255.
    • (2002) Biomaterials , vol.15 , pp. 3247-3255
    • Pignatello, R.1    Spedalieri, G.2    Bucolo, C.3    Maltese, A.4    Puglisi, G.5
  • 29
    • 0014779155 scopus 로고
    • Two-dimensional thin-layer chromatographic separation of polar lipids and determination of phospholipids by phosphorous analysis of spots
    • Rouser G, Fleischer S, Yamamoto A. Two-dimensional thin-layer chromatographic separation of polar lipids and determination of phospholipids by phosphorous analysis of spots. Lipids. 1970;5:494-496.
    • (1970) Lipids , vol.5 , pp. 494-496
    • Rouser, G.1    Fleischer, S.2    Yamamoto, A.3
  • 30
    • 0025963179 scopus 로고
    • The effects of density fluctuations on the partitioning of foreign molecules into bilayers: Application to anaesthetics and insecticides
    • Jorgensen K, Ipsen JH, Mouritsen OG, Bennet D, Zuckermann MJ. The effects of density fluctuations on the partitioning of foreign molecules into bilayers: application to anaesthetics and insecticides. Biochim Biophys Acta. 1991;1062: 227-238.
    • (1991) Biochim. Biophys. Acta , vol.1062 , pp. 227-238
    • Jorgensen, K.1    Ipsen, J.H.2    Mouritsen, O.G.3    Bennet, D.4    Zuckermann, M.J.5
  • 31
    • 0003428288 scopus 로고
    • Cell biology: A series of monographs, vol 5: Phospholipid bilayers: Physical principles and models
    • Bittar EE, ed. New York, NY: Wiley; New York
    • Cevc G, Marsh D. Cell biology: a series of monographs, vol 5: phospholipid bilayers: physical principles and models, In: Bittar EE, ed. Phospholipid Bilayers Physical Principles and Models. New York, NY: Wiley; New York, 1987:1-441.
    • (1987) Phospholipid Bilayers Physical Principles and Models , pp. 1-441
    • Cevc, G.1    Marsh, D.2
  • 33
    • 0027979462 scopus 로고
    • Characterization of acrylic resin matrix films and mechanisms of drug-polymer interactions
    • Jenquin MR, McGinity JW. Characterization of acrylic resin matrix films and mechanisms of drug-polymer interactions. Int J Pharm. 1994;10:23-34.
    • (1994) Int. J. Pharm. , vol.10 , pp. 23-34
    • Jenquin, M.R.1    McGinity, J.W.2
  • 34
    • 33544472586 scopus 로고    scopus 로고
    • Preparation of solid dispersions of non-steroidal anti-inflammatory drugs with acrylic polymers and studies on mechanisms of drug-polymer interactions
    • In press
    • Pignatello R, Ferro M, Puglisi G. Preparation of solid dispersions of non-steroidal anti-inflammatory drugs with acrylic polymers and studies on mechanisms of drug-polymer interactions. PharmSciTech. In press.
    • Pharm. Sci. Tech
    • Pignatello, R.1    Ferro, M.2    Puglisi, G.3
  • 35
    • 0025126368 scopus 로고
    • Physical and chemical factors influencing the release of drugs from acrylic resins films
    • Jenquin MR, Liebowitz SM, Sarabia RE, McGinity JW. Physical and chemical factors influencing the release of drugs from acrylic resins films. J Pharm Sci. 1990;79:811-816.
    • (1990) J. Pharm. Sci. , vol.79 , pp. 811-816
    • Jenquin, M.R.1    Liebowitz, S.M.2    Sarabia, R.E.3    McGinity, J.W.4
  • 36
    • 0034835233 scopus 로고    scopus 로고
    • Effect of pH on diclofenac release from Eudragit RS100® microparticles: A kinetic study by DSC
    • Castelli F, Messina C, Pignatello R, Puglisi G. Effect of pH on diclofenac release from Eudragit RS100® microparticles: a kinetic study by DSC. Drug Delivery. 2001;8:173-177.
    • (2001) Drug Delivery , vol.8 , pp. 173-177
    • Castelli, F.1    Messina, C.2    Pignatello, R.3    Puglisi, G.4


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