Sublimation characterization and vapor pressure estimation of an HIV nonnucleoside reverse transcriptase inhibitor using thermogravimetric analysis

AAPS PharmSciTech

Volumn 4, Issue 2, 2003, Pages

  Xie, Minli ^a,c   Ziemba, Theresa M ^a   Maurin, Michael B ^a,b  

^a DUPONT COMPANY   (United States)

^b QS Pharma   (United States)

^c BRISTOL MYERS SQUIBB   (United States)

Author keywords

Sublimation; Thermogravimetric analysis infrared (TGA IR); Vapor pressure

Indexed keywords

4 CYCLOPROPYLETHYNYL 5,6 DIFLUORO 3,4 DIHYDRO 4 TRIFLUOROMETHYL 2(1H) QUINAZOLINONE; 4 CYCLOPROPYLETHYNYL 5,6 DIFLUORO 4 TRIFLUOROMETHYL 3,4 DIHYDRO 2(1H) QUINAZOLINONE; BENZOIC ACID; RNA DIRECTED DNA POLYMERASE; RNA DIRECTED DNA POLYMERASE INHIBITOR; UNCLASSIFIED DRUG; VIRUS ENZYME; QUINOLONE DERIVATIVE;

ACCURACY; ARTICLE; CALCULATION; CONTROLLED STUDY; DIFFERENTIAL SCANNING CALORIMETRY; DRUG FORMULATION; DRUG MANUFACTURE; DRUG RESEARCH; DRUG STRUCTURE; ENTHALPY; ENTROPY; EVAPORATION; HUMAN IMMUNODEFICIENCY VIRUS 1; INFRARED SPECTROSCOPY; SAFETY; STRUCTURE ANALYSIS; TEMPERATURE DEPENDENCE; THERMOGRAVIMETRY; VAPOR PRESSURE; X RAY DIFFRACTION; CHEMISTRY; DRUG EFFECT; HUMAN IMMUNODEFICIENCY VIRUS; PHARMACEUTICS; PHYSICAL CHEMISTRY; THERMODYNAMICS; VOLATILIZATION;

CHEMISTRY, PHARMACEUTICAL; CHEMISTRY, PHYSICAL; HIV; QUINOLONES; REVERSE TRANSCRIPTASE INHIBITORS; TECHNOLOGY, PHARMACEUTICAL; THERMODYNAMICS; THERMOGRAVIMETRY; VOLATILIZATION;

EID: 23144436082     PISSN: 15309932     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/pt040223     Document Type: Article

References (9)

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