메뉴 건너뛰기




Volumn 6, Issue 3, 2005, Pages 139-147

Distribution of zolmitriptan into the CNS in healthy volunteers: A positron emission tomography study

Author keywords

[No Author keywords available]

Indexed keywords

CARBON 11; CARBON MONOXIDE; CARBONYL DERIVATIVE; OXYGEN 15; RADIOACTIVE MATERIAL; SEROTONIN 1B AGONIST; SEROTONIN 1D AGONIST; TRACER; ZOLMITRIPTAN;

EID: 22244480049     PISSN: 11745886     EISSN: None     Source Type: Journal    
DOI: 10.2165/00126839-200506030-00002     Document Type: Article
Times cited : (24)

References (24)
  • 1
    • 0026697460 scopus 로고
    • Sumatriptan is a potent vasoconstrictor of human dural arteries via a 5-HT1-like receptor
    • Jansen I, Edvinsson L, Mortensen A, et al. Sumatriptan is a potent vasoconstrictor of human dural arteries via a 5-HT1-like receptor. Cephalalgia 1992; 12 (4): 202-5
    • (1992) Cephalalgia , vol.12 , Issue.4 , pp. 202-205
    • Jansen, I.1    Edvinsson, L.2    Mortensen, A.3
  • 2
    • 0026688045 scopus 로고
    • Antimigraine drug sumatriptan increases blood flow velocity in large cerebral arteries during migraine attacks
    • Caekebeke JF, Ferrari MD, Zwetsloot CP, et al. Antimigraine drug sumatriptan increases blood flow velocity in large cerebral arteries during migraine attacks. Neurology 1992; 42 (8): 1522-6
    • (1992) Neurology , vol.42 , Issue.8 , pp. 1522-1526
    • Caekebeke, J.F.1    Ferrari, M.D.2    Zwetsloot, C.P.3
  • 3
    • 0030272955 scopus 로고    scopus 로고
    • Inhibition of trigeminal neurons by intravenous administration of the serotonin (5HT)1B/D agonist zolmitriptan (311C90): Are brain stem sites therapeutic targets in migraine?
    • Goadsby PJ, Hoskin KL. Inhibition of trigeminal neurons by intravenous administration of the serotonin (5HT)1B/D agonist zolmitriptan (311C90): are brain stem sites therapeutic targets in migraine? Pain 1996; 67: 355-9
    • (1996) Pain , vol.67 , pp. 355-359
    • Goadsby, P.J.1    Hoskin, K.L.2
  • 4
    • 0030974392 scopus 로고    scopus 로고
    • Direct evidence for central sites of action of zolmitriptan (311C90): An autoradiographic study in cat
    • Goadsby PJ, Knight YE. Direct evidence for central sites of action of zolmitriptan (311C90): an autoradiographic study in cat. Cephalalgia 1997; 17: 153-8
    • (1997) Cephalalgia , vol.17 , pp. 153-158
    • Goadsby, P.J.1    Knight, Y.E.2
  • 5
    • 0030778444 scopus 로고    scopus 로고
    • 1B/1D agonist for migraine
    • 1B/1D agonist for migraine. Cephalalgia 1997; 17 Suppl. 18: 4-14
    • (1997) Cephalalgia , vol.17 , Issue.18 SUPPL. , pp. 4-14
    • Martin, G.R.1
  • 6
    • 0032217263 scopus 로고    scopus 로고
    • The effects of 5 HT1A, 5 HT1B and 5 HT1D receptor agonists on trigeminal nociceptive neurotransmission in anaesthetized rats
    • Cumberbatch MJ, Hill RG, Hargreaves RJ. The effects of 5 HT1A, 5 HT1B and 5 HT1D receptor agonists on trigeminal nociceptive neurotransmission in anaesthetized rats. Eur J Pharmacol 1998; 362: 43-6
    • (1998) Eur J Pharmacol , vol.362 , pp. 43-46
    • Cumberbatch, M.J.1    Hill, R.G.2    Hargreaves, R.J.3
  • 7
    • 14644432159 scopus 로고    scopus 로고
    • Zolmitriptan is detectable in plasma 2 to 5 minutes after administration by nasal spray
    • Uemura N, Charlesworth B, Onishi T, et al. Zolmitriptan is detectable in plasma 2 to 5 minutes after administration by nasal spray [abstract]. Headache 2003; 43 (5): S159
    • (2003) Headache , vol.43 , Issue.5
    • Uemura, N.1    Charlesworth, B.2    Onishi, T.3
  • 8
    • 14644407228 scopus 로고    scopus 로고
    • Zolmitriptan demonstrates good pharmacokinetic consistency between and within individuals following intranasal administration
    • Kågedal M, Duvauchelle T, Hovsepian L, et al. Zolmitriptan demonstrates good pharmacokinetic consistency between and within individuals following intranasal administration. Br J Clin Pharmacol 2004; 57 (5): 679-80
    • (2004) Br J Clin Pharmacol , vol.57 , Issue.5 , pp. 679-680
    • Kågedal, M.1    Duvauchelle, T.2    Hovsepian, L.3
  • 9
    • 0036838322 scopus 로고    scopus 로고
    • Preliminary studies of the pharmacokinetics and tolerability of zolmitriptan nasal spray in healthy volunteers
    • Yates R, Nairn K, Dixon R, et al. Preliminary studies of the pharmacokinetics and tolerability of zolmitriptan nasal spray in healthy volunteers. J Clin Pharmacol 2002; 42: 1237-43
    • (2002) J Clin Pharmacol , vol.42 , pp. 1237-1243
    • Yates, R.1    Nairn, K.2    Dixon, R.3
  • 10
    • 0032790029 scopus 로고    scopus 로고
    • Zolmitriptan: A review of its use in migraine
    • Spencer CM, Gunasekara NS, Hills C. Zolmitriptan: a review of its use in migraine. Drugs 1999; 58(2): 347-74
    • (1999) Drugs , vol.58 , Issue.2 , pp. 347-374
    • Spencer, C.M.1    Gunasekara, N.S.2    Hills, C.3
  • 11
    • 0141706482 scopus 로고    scopus 로고
    • Positron emission tomography microdosing: A new concept with application in tracer and early clinical drug development
    • Bergstr̈om M, Grahńen A, Låangström B. Positron emission tomography microdosing: a new concept with application in tracer and early clinical drug development. Eur J Clin Pharmacol 2003; 59: 357-66
    • (2003) Eur J Clin Pharmacol , vol.59 , pp. 357-366
    • Bergstr̈om, M.1    Grahńen, A.2    Låangström, B.3
  • 12
    • 0141671876 scopus 로고    scopus 로고
    • In vivo activity of bupropion at the human dopamine transporter as measured by positron emission tomography
    • Learned-Coughlin SM, Bergström M, Savitcheva I, et al. In vivo activity of bupropion at the human dopamine transporter as measured by positron emission tomography. Biol Psychiatry 2003; 54 (8): 800-5
    • (2003) Biol Psychiatry , vol.54 , Issue.8 , pp. 800-805
    • Learned-Coughlin, S.M.1    Bergström, M.2    Savitcheva, I.3
  • 13
    • 0036297032 scopus 로고    scopus 로고
    • Positron emission tomography and brain monoamine neurotransmission: Entries for study of drug interactions
    • Hartvig P, Bergström M, Antoni G, et al. Positron emission tomography and brain monoamine neurotransmission: entries for study of drug interactions. Curr Pharm Des 2002; 8 (16): 1417-34
    • (2002) Curr Pharm des , vol.8 , Issue.16 , pp. 1417-1434
    • Hartvig, P.1    Bergström, M.2    Antoni, G.3
  • 14
    • 0035055247 scopus 로고    scopus 로고
    • D2 and 5HT2A receptor occupancy of different doses of quetiapine in schizophrenia: A PET study
    • Gefvert O, Lundberg T, Wieselgren I-M, et al. D2 and 5HT2A receptor occupancy of different doses of quetiapine in schizophrenia: a PET study. Eur Neuropsychopharmacol 2001; 11 (2): 105-10
    • (2001) Eur Neuropsychopharmacol , vol.11 , Issue.2 , pp. 105-110
    • Gefvert, O.1    Lundberg, T.2    Wieselgren, I.-M.3
  • 15
    • 0031963279 scopus 로고    scopus 로고
    • Time course of central nervous dopamine-D2 and 5-HT2 receptor blockade and plasma drug concentrations after discontinuation of que-tiapine (Seroquel) in patients with schizophrenia
    • Berl
    • Gefvert O, Bergström M, Långström B, et al. Time course of central nervous dopamine-D2 and 5-HT2 receptor blockade and plasma drug concentrations after discontinuation of que-tiapine (Seroquel) in patients with schizophrenia. Psycho-pharmacology (Berl) 1998; 135: 119-26
    • (1998) Psychopharmacology , vol.135 , pp. 119-126
    • Gefvert, O.1    Bergström, M.2    Långström, B.3
  • 16
    • 0032993862 scopus 로고    scopus 로고
    • 11C]zanamivir following administration as an intranasal spray: Evaluation with positron emission tomography
    • 11C]zanamivir following administration as an intranasal spray: evaluation with positron emission tomography. Clin Pharmacokinet 1999; 36 Suppl. 1: 33-9
    • (1999) Clin Pharmacokinet , vol.36 , Issue.1 SUPPL. , pp. 33-39
    • Bergström, M.1    Cass, L.M.R.2    Valind, S.3
  • 19
    • 11844253775 scopus 로고    scopus 로고
    • Zolmitriptan 5mg nasal spray: Efficacy and onset of action in the acute treatment of migraine: results from phase 1 of the REALIZE study
    • Gawel M, Aschoff J, May A, et al. Zolmitriptan 5mg nasal spray: efficacy and onset of action in the acute treatment of migraine: results from phase 1 of the REALIZE study. Headache 2005 Jan; 45 (1): 7-16
    • (2005) Headache , vol.45 , Issue.1 , pp. 7-16
    • Gawel, M.1    Aschoff, J.2    May, A.3
  • 20
    • 0028938469 scopus 로고
    • A rapid and accurate method to realign PET scans utilizing image edge transformation
    • Anderson JL. A rapid and accurate method to realign PET scans utilizing image edge transformation. J Nucl Med 1995; 36 (4): 657-69
    • (1995) J Nucl Med , vol.36 , Issue.4 , pp. 657-669
    • Anderson, J.L.1
  • 21
    • 21044446775 scopus 로고    scopus 로고
    • The speed of onset, efficacy and tolerability of zolmitriptan nasal spray in the acute management of migraine
    • Dodick D, Brandes J, Elkind A, et al. The speed of onset, efficacy and tolerability of zolmitriptan nasal spray in the acute management of migraine [abstract]. Headache 2004; 44 (5): 469
    • (2004) Headache , vol.44 , Issue.5 , pp. 469
    • Dodick, D.1    Brandes, J.2    Elkind, A.3
  • 22
    • 0032959306 scopus 로고    scopus 로고
    • Effects of zolmitriptan (Zomig™) on central serotonergic neurotransmission as assessed by active oddball auditory event-related potentials in volunteers without migraine
    • Hughes AM, Dixon R, Dane A, et al. Effects of zolmitriptan (Zomig™) on central serotonergic neurotransmission as assessed by active oddball auditory event-related potentials in volunteers without migraine. Cephalalgia 1999; 19: 100-6
    • (1999) Cephalalgia , vol.19 , pp. 100-106
    • Hughes, A.M.1    Dixon, R.2    Dane, A.3
  • 24
    • 0344364570 scopus 로고    scopus 로고
    • Zolmitriptan nasal spray: Advances in migraine treatment
    • Syrett N, Abu-Shakra S, Yates R. Zolmitriptan nasal spray: advances in migraine treatment. Neurology 2003; 61 (8 Suppl. 4): S27-30
    • (2003) Neurology , vol.61 , Issue.8 SUPPL. 4
    • Syrett, N.1    Abu-Shakra, S.2    Yates, R.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.