Unidirectional inversion of ibuprofen in Caco-2 cells: Developing a suitable model for presystemic chiral inversion study

Biological and Pharmaceutical Bulletin

Volumn 28, Issue 4, 2005, Pages 682-687

  Hao, Haiping ^a   Wang, Guangji ^a   Sun, Jianguo ^a   Ding, Zuoqi ^a   Wu, Xiaolan ^a   Roberts, Michael ^b  

^a CHINA PHARMACEUTICAL UNIVERSITY   (China)

^b UNIVERSITY OF QUEENSLAND   (Australia)

Author keywords

Caco 2 cell; Coenzyme A (CoA); Ibuprofen; Palmitic acid; Presystemic inversion

Indexed keywords

COENZYME A; IBUPROFEN; PALMITIC ACID; SODIUM AZIDE;

ARTICLE; CELL DENSITY; CELL STRAIN CACO 2; CHIRALITY; CONTROLLED STUDY; CULTURE MEDIUM; DOSE RESPONSE; DRUG METABOLISM; ENANTIOMER; ENZYME SUBSTRATE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; ISOMERISM; QUANTITATIVE ANALYSIS; SERUM; STEREOCHEMISTRY;

ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; CACO-2 CELLS; CELL CULTURE TECHNIQUES; COENZYME A; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; IBUPROFEN; INTESTINES; PALMITIC ACID; SODIUM AZIDE; STEREOISOMERISM;

EID: 21144434526     PISSN: 09186158     EISSN: None     Source Type: Journal    
DOI: 10.1248/bpb.28.682     Document Type: Article

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