Synthesis and structure-activity relationships of piperidinylpyrrolopyridine derivatives as potent and selective H1 antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 4, 2005, Pages 1165-1167

  Fonquerna, Silvia ^a   Miralpeix, Montse ^a   Pagès, Lluís ^a   Puig, Carles ^a   Cardús, Arantxa ^a   Antón, Francisca ^a   Vilella, Dolors ^a   Aparici, Mónica ^a   Prieto, José ^a   Warrellow, Graham ^a   Beleta, Jorge ^a   Ryder, Hamish ^a  

^a Research Center ^*  (Spain)

Author keywords

Antihistamine; H1 antagonists; Piperidinylpyrrolopyridines

Indexed keywords

HISTAMINE H1 RECEPTOR ANTAGONIST; PYRIDINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; SEDATION; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

EID: 20144389407     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.12.008     Document Type: Article

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