Evaluation of 3-substituted arginine analogs as selective inhibitors of human nitric oxide synthase isozymes

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 11, 2005, Pages 2881-2885

  Ijuin, Ryosuke ^a   Umezawa, Naoki ^a   Nagai, Shin Ichi ^a   Higuchi, Tsunehiko ^a  

^a NAGOYA CITY UNIVERSITY   (Japan)

Author keywords

Arginine; Docking study; Inhibitor; Nitric oxide; Nitric oxide synthase

Indexed keywords

ARGININE DERIVATIVE; NITRIC OXIDE SYNTHASE INHIBITOR;

ARTICLE; COMPARATIVE STUDY; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; IC 50; MATHEMATICAL MODEL;

ANIMALS; ARGININE; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; HUMANS; ISOENZYMES; MODELS, MOLECULAR; NITRIC OXIDE SYNTHASE; RECOMBINANT PROTEINS; SPODOPTERA;

EID: 19544379712     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.078     Document Type: Article

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