Benzothieno[3,2-b]indole derivatives as potent selective estrogen receptor modulators

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 11, 2005, Pages 2891-2893

  Ji, Qinggang ^a   Gao, Jie ^b   Wang, Junbo ^a   Yang, Chunhao ^a   Hui, Xin ^b   Yan, Xueming ^a   Wu, Xihan ^a   Xie, Yuyuan ^a   Wang, Ming Wei ^b  

^a SHANGHAI INSTITUTE OF MATERIA MEDICA   (China)

^b National Center for Drug Screening   (China)

Author keywords

Benzothieno 3,2 b indole; Estrogen receptor; SERM

Indexed keywords

ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; INDOLE DERIVATIVE; RALOXIFENE; RECEPTOR SUBTYPE; SELECTIVE ESTROGEN RECEPTOR MODULATOR;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BONE; BONE DENSITY; CONTROLLED STUDY; DRUG ACTIVITY; DRUG EFFECT; DRUG POTENTIATION; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; MOUSE; NONHUMAN; OVARIECTOMY; UTERUS;

ANIMALS; FEMALE; HUMANS; INDOLES; MICE; SELECTIVE ESTROGEN RECEPTOR MODULATORS;

EID: 19544364498     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.111     Document Type: Article

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