Synthesis of 3H- and 14C-labeled AR-A000002, a new and selective 5-HT1B/1D ligand

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 47, Issue 3, 2004, Pages 175-180

  Werner, Tom ^a   Berg, Stefan ^a   Johansson, Rolf ^a  

^a ASTRAZENECA R AND D   (Sweden)

Author keywords

5 HT1B; 5 HT1D; 14C; 3H; Rosenmund von Braun

Indexed keywords

14C; 3H; 5-HT1B; 5-HT1D; EXTRACELLULAR CONCENTRATION; GUINEA PIGS; HIGH AFFINITY; IN-VIVO; RECEPTOR ANTAGONISTS; ROSENMUND-VON BRAUN;

CHELATION;

5 HYDROXYINDOLEACETIC ACID; AR A000002; CARBON 14; SEROTONIN; SEROTONIN 1B ANTAGONIST; TRITIUM;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN; DRUG LABELING; DRUG SYNTHESIS; FRONTAL CORTEX; GUINEA PIG; ISOTOPE LABELING; MOOD DISORDER; NONHUMAN;

CAVIA PORCELLUS; SUS SCROFA;

EID: 1942534039     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/jlcr.810     Document Type: Article

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