Targeting specific PDZ domains of PSD-95: Structural basis for enhanced affinity and enzymatic stability of a cyclic peptide

Chemistry and Biology

Volumn 11, Issue 4, 2004, Pages 469-473

  Piserchio, Andrea ^a   Salinas, Gregory D ^a   Li, Tao ^b   Marshall, John ^a   Spaller, Mark R ^b   Mierke, Dale F ^a  

^a BROWN UNIVERSITY   (United States)

^b WAYNE STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CYCLOPEPTIDE; KAINIC ACID RECEPTOR; LIGAND; NERVE PROTEIN; POSTSYNAPTIC DENSITY PROTEINS;

ARTICLE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; ENZYME STABILITY; METABOLISM; PHYSIOLOGY; PROTEIN BINDING; PROTEIN TERTIARY STRUCTURE; STRUCTURE ACTIVITY RELATION;

ENZYME STABILITY; LIGANDS; MODELS, MOLECULAR; NERVE TISSUE PROTEINS; PEPTIDES, CYCLIC; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, KAINIC ACID; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 1942509545     PISSN: 10745521     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.chembiol.2004.03.013     Document Type: Article

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