Design and synthesis of a new type of non steroidal human aromatase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 9, 1998, Pages 1041-1044

  Sonnet, P ^a   Guillon, J ^a   Enguehard, C ^a   Dallemagne, P ^a   Bureau, R ^a   Rault, S ^a   Auvray, P ^b   Moslemi, S ^b   Sourdaine, P ^b   Galopin, S ^b   Seralini G E ^b  

^a Laboratoire de Pharmacochimie   (France)

^b UNIVERSITÉ DE CAEN   (France)

Author keywords

[No Author keywords available]

Indexed keywords

AROMATASE INHIBITOR; CHLOROPHENYLPYRIDYLMETHYLENETETRAHYDROINDOLIZINONE; FADROZOLE; MR 20814; UNCLASSIFIED DRUG; VOROZOLE;

ARTICLE; DRUG DESIGN; DRUG SYNTHESIS; ENZYME ACTIVE SITE; ENZYME INHIBITION; ESTROGEN SYNTHESIS; HYDROPHOBICITY; MOLECULAR MODEL; NONHUMAN; STRUCTURE ACTIVITY RELATION; ULTRAVIOLET SPECTROSCOPY;

AROMATASE INHIBITORS; DRUG DESIGN; ENZYME INHIBITORS; FADROZOLE; FEMALE; HUMANS; INDICATORS AND REAGENTS; INDOLIZINES; MICROSOMES; PLACENTA; PREGNANCY; PYRIDINES; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZOLES;

EID: 18844478759     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00157-7     Document Type: Article

References (10)

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