New progesterone receptor antagonists: 3,3-disubstituted-5-aryloxindoles

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 23, 2002, Pages 3487-3490

  Fensome, Andrew ^a   Bender, Reinhold ^a   Cohen, Jeffrey ^a   Collins, Mark A ^a   Mackner, Valerie A ^a   Miller, Lori L ^a   Ullrich, John W ^a   Winneker, Richard ^a   Wrobel, Jay ^a   Zhang, Puwen ^a   Zhang, Zhiming ^a   Zhu, Yuan ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

INDOLE DERIVATIVE; OXINDOLE; RECEPTOR BLOCKING AGENT; ALKALINE PHOSPHATASE; CYCLOHEXANE DERIVATIVE; PROGESTERONE RECEPTOR;

ARTICLE; DRUG ACTIVITY; DRUG SYNTHESIS; ENZYME ASSAY; STRUCTURE ACTIVITY RELATION; ANIMAL; BINDING COMPETITION; BIOASSAY; BREAST TUMOR; CELL CULTURE; CHEMISTRY; DECIDUA; DRUG ANTAGONISM; DRUG EFFECT; FEMALE; HUMAN; IC 50; METABOLISM; RAT;

ALKALINE PHOSPHATASE; ANIMALS; BINDING, COMPETITIVE; BIOLOGICAL ASSAY; BREAST NEOPLASMS; CYCLOHEXANES; DECIDUA; FEMALE; HUMANS; INDOLES; INHIBITORY CONCENTRATION 50; RATS; RECEPTORS, PROGESTERONE; STRUCTURE-ACTIVITY RELATIONSHIP; TUMOR CELLS, CULTURED;

EID: 18644369735     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00746-1     Document Type: Article

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