3-Cyanoindole-based inhibitors of inosine monophosphate dehydrogenase: Synthesis and initial structure-activity relationships

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 20, 2003, Pages 3557-3560

  Dhar, T G Murali ^a   Shen, Zhongqi ^a   Gu, Henry H ^a   Chen, Ping ^a   Norris, Derek ^a   Watterson, Scott H ^a   Ballentine, Shelley K ^a   Fleener, Catherine A ^a   Rouleau, Katherine A ^a   Barrish, Joel C ^a   Townsend, Robert ^a   Hollenbaugh, Diane L ^a   Iwanowicz, Edwin J ^a  

^a BRISTOL MYERS SQUIBB   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

INOSINATE DEHYDROGENASE INHIBITOR;

ANTIVIRAL ACTIVITY; ARTICLE; CANCER THERAPY; CATALYSIS; DRUG SYNTHESIS; IMMUNOSUPPRESSIVE TREATMENT; IN VITRO STUDY; NUCLEOTIDE METABOLISM; STRUCTURE ACTIVITY RELATION;

EID: 1842551076     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00757-1     Document Type: Article

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