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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 4, 2002, Pages 575-579

2-(Anilinomethyl)imidazolines as α1A adrenergic receptor agonists: 2′-heteroaryl and 2′-oxime ether series

(11) Navas III, Frank a Bishop, Michael J a Garrison, Deanna T a Hodson, Stephen J a Speake, Jason D a Bigham, Eric C a Drewry, David H a Saussy, David L a Liacos, James H a Irving, Paul E a Gobel, M Jeffrey a

a GLAXOSMITHKLINE (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA 1A ADRENERGIC RECEPTOR; ALPHA 1B ADRENERGIC RECEPTOR; ALPHA 1D ADRENERGIC RECEPTOR; ALPHA ADRENERGIC RECEPTOR STIMULATING AGENT; ETHER DERIVATIVE; IMIDAZOLINE DERIVATIVE; RECEPTOR SUBTYPE; ADRENERGIC RECEPTOR ALPHA(1A); ADRENERGIC RECEPTOR ALPHA(1B); ADRENERGIC RECEPTOR ALPHA(1D); ALPHA 1 ADRENERGIC RECEPTOR; HETEROCYCLIC COMPOUND; IMIDAZOLE DERIVATIVE; OXIME; PHENYLEPHRINE;

ARTICLE; DRUG ACTIVITY; DRUG EFFICACY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG SYNTHESIS; IN VITRO STUDY; NONHUMAN; ANIMAL; CALCIUM SIGNALING; CELL LINE; CHEMISTRY; DRUG EFFECT; DRUG POTENTIATION; HUMAN; METABOLISM; MOLECULAR CLONING; PROTEIN BINDING; RAT; SYNTHESIS;

ADRENERGIC ALPHA-AGONISTS; ANIMALS; CALCIUM SIGNALING; CELL LINE; CLONING, MOLECULAR; HETEROCYCLIC COMPOUNDS; HUMANS; IMIDAZOLES; OXIMES; PHENYLEPHRINE; PROTEIN BINDING; RATS; RECEPTORS, ADRENERGIC, ALPHA-1;

EID: 18244405366 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)00822-8 Document Type: Article

Times cited : (12)

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