Synthesis and relative bioavailability of meptazinol benzoyl esters as prodrugs

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 10, 2005, Pages 2607-2609

  Lu, Meiyan ^a   Zhang, Chengji ^a   Hao, Jinglai ^a   Qiu, Zhuibai ^a  

^a FUDAN UNIVERSITY   (China)

Author keywords

Analgesic; Benzoic ester; Meptazinol; Prodrug

Indexed keywords

(2 AMINE 6 METHYL)BENZOIC ACID MEPTAZINOL ESTER; ESTER DERIVATIVE; MEPTAZINOL; MEPTAZINOL DERIVATIVE; PRODRUG; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG EFFICACY; DRUG SYNTHESIS; INTESTINE ABSORPTION; MASS SPECTROMETRY; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; RAT;

EID: 18144388687     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.039     Document Type: Article

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