Design, synthesis and analysis of novel bicyclic and bifunctional protease inhibitors

Protein Engineering, Design and Selection

Volumn 17, Issue 9, 2004, Pages 681-687

  Jaulent, Agnès M ^a   Leatherbarrow, Robin J ^a  

^a IMPERIAL COLLEGE LONDON   (United Kingdom)

Author keywords

Bowman Birk inhibitor; Peptide synthesis; Protease inhibitor; Sunflower trypsin inhibitor

Indexed keywords

ENZYME KINETICS; PROTEINS;

BIFUNCTIONAL INHIBITION; BOWMAN BIRK INHIBITOR (BBI); PROTEOLYSIS; SUNFLOWER TRYPSIN INHIBITOR-1 (SFTI-1);

ENZYME INHIBITION;

BOWMAN BIRK INHIBITOR; PROTEINASE INHIBITOR; SUNFLOWER TRYPSIN INHIBITOR; TRYPSIN; UNCLASSIFIED DRUG;

ARTICLE; ENZYME ACTIVE SITE; ENZYME ANALYSIS; ENZYME STRUCTURE; ENZYME SYNTHESIS; HYDROLYSIS; PRIORITY JOURNAL; PROTEIN DEGRADATION; PROTEINASE INHIBITION; STOICHIOMETRY; STRUCTURE ANALYSIS;

BINDING SITES; CHYMOTRYPSIN; CYCLIZATION; HELIANTHUS; HYDROLYSIS; PEPTIDES, CYCLIC; PROTEASE INHIBITORS; PROTEIN ENGINEERING; PROTEIN STRUCTURE, TERTIARY; TRYPSIN; TRYPSIN INHIBITOR, BOWMAN-BIRK SOYBEAN; TRYPSIN INHIBITORS;

HELIANTHUS;

EID: 18044368932     PISSN: 17410126     EISSN: None     Source Type: Journal    
DOI: 10.1093/protein/gzh077     Document Type: Article

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