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Volumn 57, Issue 30, 2001, Pages 6511-6522

Total synthesis of a pepstatin analog incorporating two trifluoromethyl hydroxymethylene isosteres (Tfm-GABOB) and evaluation of Tfm-GABOB containing peptides as inhibitors of HIV-1 protease and MMP-9

(13) Pesenti, Cristina a Arnone, Alberto a Bellosta, Stefano b Bravo, Pierfrancesco a Canavesi, Monica b Corradi, Eleonora a Frigerio, Massimo a Meille, Stefano V a Monetti, Mara b Panzeri, Walter a Viani, Fiorenza a Venturini, Romina c Zanda, Matteo a

a CNR (Italy)

b UNIVERSITY OF MILAN (Italy)

c UNIVERSITY OF TRIESTE (Italy)

Author keywords

Asymmetric synthesis; HIV; Metalloproteinase; Peptide isosteres; Trifluoromethyl group

Indexed keywords

BUTYRIC ACID DERIVATIVE; GAMMA TRIFLUOROMETHYL GAMMA AMINO BETA HYDROXYBUTYRIC ACID; GELATINASE B; PEPSTATIN DERIVATIVE; PROTEINASE; STATINE; UNCLASSIFIED DRUG; VIRUS ENZYME;

ARTICLE; CONTROLLED STUDY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; MACROPHAGE; NONHUMAN; PRIORITY JOURNAL; REACTION ANALYSIS;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 17844378965 PISSN: 00404020 EISSN: None Source Type: Journal
DOI: 10.1016/S0040-4020(01)00543-9 Document Type: Article

Times cited : (36)

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