A novel super-potent neurokinin a receptor antagonist containing dehydroalanine

Bioorganic and Medicinal Chemistry Letters

Volumn 8, Issue 10, 1998, Pages 1153-1156

  Lombardi, Angela ^a   D'Agostino, Bruno ^b   Nastri, Flavia ^a   D'Andrea, Luca D ^a   Filippelli, Amelia ^b   Falciani, Maddalena ^b   Rossi, Francesco ^b   Pavone, Vincenzo ^a  

^a UNIVERSITY OF NAPLES FEDERICO II   (Italy)

^b SECOND UNIVERSITY OF NAPLES   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

CYCLOPEPTIDE; DEHYDROALANINE; HEXAPEPTIDE; MEN 10627; NEUROKININ 1 RECEPTOR; NEUROKININ 2 RECEPTOR ANTAGONIST; NEUROKININ 3 RECEPTOR;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; MOLECULAR DYNAMICS; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; RAT; STRUCTURE ACTIVITY RELATION; VAS DEFERENS;

ALANINE; AMINO ACID SEQUENCE; ANIMALS; MALE; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PEPTIDES, CYCLIC; PROTEIN CONFORMATION; RATS; RECEPTORS, NEUROKININ-2; STRUCTURE-ACTIVITY RELATIONSHIP; VAS DEFERENS;

ANIMALIA;

EID: 17444452500     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(98)00178-4     Document Type: Article

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