-
1
-
-
0343680287
-
Distinct functional muscarinic receptor subtypes in rat atrium and guinea-pig gallbladder
-
Akbulut, H., Akin, S.B., Gören, Z., Özdemir, O., Oktay, S., 1995. Distinct functional muscarinic receptor subtypes in rat atrium and guinea-pig gallbladder. Life Sci. 56, 1039.
-
(1995)
Life Sci.
, vol.56
, pp. 1039
-
-
Akbulut, H.1
Akin, S.B.2
Gören, Z.3
Özdemir, O.4
Oktay, S.5
-
2
-
-
0009644628
-
Some quantitative uses of drug antagonists
-
Arunlakshana, O., Schild, H.O., 1959. Some quantitative uses of drug antagonists. Br. J. Pharmacol. 14, 48-58.
-
(1959)
Br. J. Pharmacol.
, vol.14
, pp. 48-58
-
-
Arunlakshana, O.1
Schild, H.O.2
-
3
-
-
0023062987
-
Inositol triphosphate and diacylglycerol: Two interacting second messengers
-
Berridge, M.J., 1987. Inositol triphosphate and diacylglycerol: Two interacting second messengers. Ann. Rev. Biochem. 56, 159-193.
-
(1987)
Ann. Rev. Biochem.
, vol.56
, pp. 159-193
-
-
Berridge, M.J.1
-
4
-
-
0026579901
-
Antagonism by antimuscarinic and neuroleptic compounds at the five cloned human muscarinic cholinergic receptors expressed in Chinese hamster ovary cells
-
Bolden, C., Cusack, B., Richelson, E., 1992. Antagonism by antimuscarinic and neuroleptic compounds at the five cloned human muscarinic cholinergic receptors expressed in Chinese hamster ovary cells. J. Pharmacol. Exp. Ther. 260, 576-580.
-
(1992)
J. Pharmacol. Exp. Ther.
, vol.260
, pp. 576-580
-
-
Bolden, C.1
Cusack, B.2
Richelson, E.3
-
5
-
-
0024472059
-
New types of muscarinic acetylcholine receptors
-
Bonner, T.I., 1989. New types of muscarinic acetylcholine receptors. Trends Pharmacol. Sci. 10 (Suppl.), 11-15.
-
(1989)
Trends Pharmacol. Sci.
, vol.10
, Issue.SUPPL.
, pp. 11-15
-
-
Bonner, T.I.1
-
6
-
-
0027496789
-
Muscarinic acetylcholine receptor subtypes: Localization and structure/function
-
Brann, M.R., Ellis, J., Jørgensen, H., Hill-Eubanks, D., Jones, S.V.P., 1993. Muscarinic acetylcholine receptor subtypes: Localization and structure/function. Prog. Brain Res. 98, 121-127.
-
(1993)
Prog. Brain Res.
, vol.98
, pp. 121-127
-
-
Brann, M.R.1
Ellis, J.2
Jørgensen, H.3
Hill-Eubanks, D.4
Jones, S.V.P.5
-
7
-
-
0039410502
-
Pharmacology of muscarinic acetylcholine receptor subtypes (m1-m5): High throughput assays in mammalian cells
-
Bräuner-Osborne, H., Brann, M.R., 1996. Pharmacology of muscarinic acetylcholine receptor subtypes (m1-m5): high throughput assays in mammalian cells. Eur. J. Pharmacol. 295, 93-102.
-
(1996)
Eur. J. Pharmacol.
, vol.295
, pp. 93-102
-
-
Bräuner-Osborne, H.1
Brann, M.R.2
-
8
-
-
0024507616
-
Antagonist binding properties of five cloned muscarinic receptors expressed in CHO-K1 cells
-
Buckley, N.J., Bonner, T.I., Buckley, C.M., Brann, M.R., 1989. Antagonist binding properties of five cloned muscarinic receptors expressed in CHO-K1 cells. Mol. Pharmacol. 35, 469-476.
-
(1989)
Mol. Pharmacol.
, vol.35
, pp. 469-476
-
-
Buckley, N.J.1
Bonner, T.I.2
Buckley, C.M.3
Brann, M.R.4
-
9
-
-
0025918366
-
4 muscarinic receptor mediating Ca-current inhibition in neuroblastoma X glioma hybrid (NG 108-15) cells
-
4 muscarinic receptor mediating Ca-current inhibition in neuroblastoma X glioma hybrid (NG 108-15) cells. Br. J. Pharmacol. 104, 39-44.
-
(1991)
Br. J. Pharmacol.
, vol.104
, pp. 39-44
-
-
Caulfield, M.P.1
Brown, D.A.2
-
10
-
-
0027525338
-
Characterization of muscarinic receptors in guinea-pig uterus
-
Doods, H.N., Willim, K.D., Boddeke, H.W.G.M., Entzeroth, M., 1993. Characterization of muscarinic receptors in guinea-pig uterus. Eur. J. Pharmacol. 250, 223-230.
-
(1993)
Eur. J. Pharmacol.
, vol.250
, pp. 223-230
-
-
Doods, H.N.1
Willim, K.D.2
Boddeke, H.W.G.M.3
Entzeroth, M.4
-
11
-
-
0025046203
-
Novel pharmacological profile of muscarinic receptors mediating contraction of the guinea-pig uterus
-
Dörje, F., Friebe, T., Tacke, R., Mutschler, E., Lambrecht, G., 1990. Novel pharmacological profile of muscarinic receptors mediating contraction of the guinea-pig uterus. Naunyn-Schmiedeberg's Arch. Pharmacol. 342, 284-289.
-
(1990)
Naunyn-Schmiedeberg's Arch. Pharmacol.
, vol.342
, pp. 284-289
-
-
Dörje, F.1
Friebe, T.2
Tacke, R.3
Mutschler, E.4
Lambrecht, G.5
-
12
-
-
0026050428
-
Immunological detection of muscarinic receptor subtype proteins (m1-m5) in rabbit peripheral tissues
-
Dörje, F., Levey, A.I., Brann, M.R., 1991a. Immunological detection of muscarinic receptor subtype proteins (m1-m5) in rabbit peripheral tissues. Mol. Pharmacol. 40, 459-462.
-
(1991)
Mol. Pharmacol.
, vol.40
, pp. 459-462
-
-
Dörje, F.1
Levey, A.I.2
Brann, M.R.3
-
13
-
-
0026033504
-
Antagonist binding profiles of five cloned human muscarinic receptor subtypes
-
Dörje, F., Wess, J., Lambrecht, G., Tacke, R., Mutschler, E., Brann, M.R., 1991b. Antagonist binding profiles of five cloned human muscarinic receptor subtypes. J. Pharmacol. Exp. Ther. 256, 727-733.
-
(1991)
J. Pharmacol. Exp. Ther.
, vol.256
, pp. 727-733
-
-
Dörje, F.1
Wess, J.2
Lambrecht, G.3
Tacke, R.4
Mutschler, E.5
Brann, M.R.6
-
14
-
-
0024576921
-
Characterization of the muscarinic receptor subtype mediating contraction of the guinea-pig uterus
-
Eglen, R.M., Michel, A.D., Whiting, R.L., 1989. Characterization of the muscarinic receptor subtype mediating contraction of the guinea-pig uterus. Br. J. Pharmacol. 96, 497-499.
-
(1989)
Br. J. Pharmacol.
, vol.96
, pp. 497-499
-
-
Eglen, R.M.1
Michel, A.D.2
Whiting, R.L.3
-
15
-
-
0026645180
-
Acute desensitization of muscarinic receptors in the isolated guinea-pig ileal longitudinal muscle
-
Eglen, R.M., Adham, N., Whiting, R.L., 1992. Acute desensitization of muscarinic receptors in the isolated guinea-pig ileal longitudinal muscle. J. Auton. Pharmacol. 12, 137-148.
-
(1992)
J. Auton. Pharmacol.
, vol.12
, pp. 137-148
-
-
Eglen, R.M.1
Adham, N.2
Whiting, R.L.3
-
16
-
-
0030442725
-
Muscarinic receptor subtypes and smooth muscle function
-
Eglen, R.M., Hedge, S.S., Watson, N., 1996. Muscarinic receptor subtypes and smooth muscle function. Pharmacol. Rev. 48, 531-565.
-
(1996)
Pharmacol. Rev.
, vol.48
, pp. 531-565
-
-
Eglen, R.M.1
Hedge, S.S.2
Watson, N.3
-
17
-
-
0023821640
-
2-receptors mediating opposite effects on neuromuscular transmission in rabbit vas deferens
-
2-receptors mediating opposite effects on neuromuscular transmission in rabbit vas deferens. Eur. J. Pharmacol. 151, 205-221.
-
(1988)
Eur. J. Pharmacol.
, vol.151
, pp. 205-221
-
-
Eltze, M.1
-
18
-
-
0028182611
-
4 receptors in vagally stimulated contractions of rabbit bronchus/trachea
-
4 receptors in vagally stimulated contractions of rabbit bronchus/trachea. Pulm. Pharmacol. 7, 109-120.
-
(1994)
Pulm. Pharmacol.
, vol.7
, pp. 109-120
-
-
Eltze, M.1
Galvan, M.2
-
19
-
-
0024805917
-
Cyproheptadine displays high affinity for muscarinic receptors but does not discriminate between receptor subtypes
-
Eltze, M., Lambrecht, G., Mutschler, E., 1989. Cyproheptadine displays high affinity for muscarinic receptors but does not discriminate between receptor subtypes. Eur. J. Pharmacol. 173, 219-222.
-
(1989)
Eur. J. Pharmacol.
, vol.173
, pp. 219-222
-
-
Eltze, M.1
Lambrecht, G.2
Mutschler, E.3
-
20
-
-
0027216505
-
Characterization of muscarinic receptors mediating vasodilation in rat perfused kidney
-
Eltze, M., Ullrich, B., Mutschler, E., Moser, U., Bungardt, E., Friebe, T., Gubitz, C., Tacke, R., Lambrecht, G., 1993. Characterization of muscarinic receptors mediating vasodilation in rat perfused kidney. Eur. J. Pharmacol. 238, 343-355.
-
(1993)
Eur. J. Pharmacol.
, vol.238
, pp. 343-355
-
-
Eltze, M.1
Ullrich, B.2
Mutschler, E.3
Moser, U.4
Bungardt, E.5
Friebe, T.6
Gubitz, C.7
Tacke, R.8
Lambrecht, G.9
-
23
-
-
0025361044
-
Muscarinic receptor subtypes
-
Hulme, E.C., Birdsall, N.J.M., Buckley, N.J., 1990. Muscarinic receptor subtypes. Annu. Rev. Pharmacol. Toxicol. 30, 633-673.
-
(1990)
Annu. Rev. Pharmacol. Toxicol.
, vol.30
, pp. 633-673
-
-
Hulme, E.C.1
Birdsall, N.J.M.2
Buckley, N.J.3
-
24
-
-
0026003009
-
Muscarinic receptor subtypes of the guinea-pig common bile duct
-
Karahan, F., Alican, I., Özkutlu, U., Onat, F., Yegen, B.C., Ulusoy, N.B., Oktay, S., 1991. Muscarinic receptor subtypes of the guinea-pig common bile duct. Arch. Int. Pharmacodyn. Ther. 312, 140-145.
-
(1991)
Arch. Int. Pharmacodyn. Ther.
, vol.312
, pp. 140-145
-
-
Karahan, F.1
Alican, I.2
Özkutlu, U.3
Onat, F.4
Yegen, B.C.5
Ulusoy, N.B.6
Oktay, S.7
-
25
-
-
0002083250
-
Schild regressions as indicators of non-equilibrium steady-states and heterogeneous receptor populations
-
Kenakin, T.P., 1985. Schild regressions as indicators of non-equilibrium steady-states and heterogeneous receptor populations. Trends Pharmacol. Sci. 6, 68-72.
-
(1985)
Trends Pharmacol. Sci.
, vol.6
, pp. 68-72
-
-
Kenakin, T.P.1
-
26
-
-
0002261623
-
Stimulus-response mechanism
-
Kenakin, T.P. (Ed.), Raven Press, New York, NY
-
Kenakin, T.P., 1987. Stimulus-response mechanism. In: Kenakin, T.P. (Ed.), Pharmacologic Analysis of Drug-Receptor Interactions. Raven Press, New York, NY, pp. 31-51.
-
(1987)
Pharmacologic Analysis of Drug-Receptor Interactions
, pp. 31-51
-
-
Kenakin, T.P.1
-
27
-
-
0025690787
-
Muscarinic receptor subtypes of guinea-pig gallbladder smooth muscle
-
Kurtel, H., Yegen, B.C., Dedeoglu, A., Ulusoy, N.B., Oktay, S., 1990. Muscarinic receptor subtypes of guinea-pig gallbladder smooth muscle. Arch. Int. Pharmacodyn. 308, 39-46.
-
(1990)
Arch. Int. Pharmacodyn.
, vol.308
, pp. 39-46
-
-
Kurtel, H.1
Yegen, B.C.2
Dedeoglu, A.3
Ulusoy, N.B.4
Oktay, S.5
-
28
-
-
0028936859
-
The design and pharmacology of novel selective muscarinic agonists and antagonists
-
Lambrecht, G., Gross, J., Hacksell, U., Hermanni, U., Hildebrandt, C., Hou, X., Moser, U., Nilsson, B.M., Pfaff, O., Waelbroeck, M., Wehrle, J., Mutschler, E., 1995. The design and pharmacology of novel selective muscarinic agonists and antagonists. Life Sci. 56, 815-822.
-
(1995)
Life Sci.
, vol.56
, pp. 815-822
-
-
Lambrecht, G.1
Gross, J.2
Hacksell, U.3
Hermanni, U.4
Hildebrandt, C.5
Hou, X.6
Moser, U.7
Nilsson, B.M.8
Pfaff, O.9
Waelbroeck, M.10
Wehrle, J.11
Mutschler, E.12
-
29
-
-
0027313323
-
35S]-GTPγS binding mediated by human muscarinic m1-m4 receptors: Antagonist studies
-
35S]-GTPγS binding mediated by human muscarinic m1-m4 receptors: Antagonist studies. Br. J. Pharmacol. 109, 1120-1127.
-
(1993)
Br. J. Pharmacol.
, vol.109
, pp. 1120-1127
-
-
Lazareno, S.1
Birdsall, N.J.M.2
-
30
-
-
0025572697
-
4 binding sites in rabbit lung, chicken heart, and NG108-15 cells
-
4 binding sites in rabbit lung, chicken heart, and NG108-15 cells. Mol. Pharmacol. 38, 805-815.
-
(1990)
Mol. Pharmacol.
, vol.38
, pp. 805-815
-
-
Lazareno, S.1
Buckley, N.J.2
Roberts, F.F.3
-
31
-
-
0027465882
-
Immunological localization of m1-m5 muscarinic acetylcholine receptors in peripheral tissues and brain
-
Proc. Subtypes Muscarinic Receptors V
-
Levey, A.I., 1993. Immunological localization of m1-m5 muscarinic acetylcholine receptors in peripheral tissues and brain. Proc. Subtypes Muscarinic Receptors V., Life Sci. 52, 441-448.
-
(1993)
Life Sci.
, vol.52
, pp. 441-448
-
-
Levey, A.I.1
-
33
-
-
0028169674
-
Binding profile of the selective muscarinic antagonist tripitramine
-
Maggio, R., Barbier, P., Bolognesi, M.L., Minarini, A., Tedeschi, D., Melchiorre, C., 1994. Binding profile of the selective muscarinic antagonist tripitramine. Eur. J. Pharmacol. 268, 459-462.
-
(1994)
Eur. J. Pharmacol.
, vol.268
, pp. 459-462
-
-
Maggio, R.1
Barbier, P.2
Bolognesi, M.L.3
Minarini, A.4
Tedeschi, D.5
Melchiorre, C.6
-
36
-
-
0028967878
-
The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists
-
Melchiorre, C., Minarini, A., Budriesi, R., Chiarini, A., Spampinato, S., Tumiatti, V., 1995. The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists. Life Sci. 56, 837-844.
-
(1995)
Life Sci.
, vol.56
, pp. 837-844
-
-
Melchiorre, C.1
Minarini, A.2
Budriesi, R.3
Chiarini, A.4
Spampinato, S.5
Tumiatti, V.6
-
37
-
-
0024346566
-
Binding characteristics of the muscarinic receptor subtype of the NG108-12 cell line
-
Michel, A.D., Delmendo, R., Stefanich, E., Whiting, R.L., 1989. Binding characteristics of the muscarinic receptor subtype of the NG108-12 cell line. Naunyn-Schmiedeberg's Arch. Pharmacol. 340, 62-67.
-
(1989)
Naunyn-Schmiedeberg's Arch. Pharmacol.
, vol.340
, pp. 62-67
-
-
Michel, A.D.1
Delmendo, R.2
Stefanich, E.3
Whiting, R.L.4
-
39
-
-
0027945826
-
Design, synthesis, and biological activity of methoctramine-related tetraamines bearing an 11-acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4] benzodiazepin-6-one moiety: Structural requirements for optimum occupancy of muscarinic receptor subtypes as revealed by symmetrical and asymmetrical polyamines
-
Minarini, A., Bolognesi, M.L., Budriesi, R., Canossa, M., Chiarini, A., Spampinato, S., Melchiorre, C., 1994. Design, synthesis, and biological activity of methoctramine-related tetraamines bearing an 11-acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4] benzodiazepin-6-one moiety: Structural requirements for optimum occupancy of muscarinic receptor subtypes as revealed by symmetrical and asymmetrical polyamines. J. Med. Chem. 30, 3363-3372.
-
(1994)
J. Med. Chem.
, vol.30
, pp. 3363-3372
-
-
Minarini, A.1
Bolognesi, M.L.2
Budriesi, R.3
Canossa, M.4
Chiarini, A.5
Spampinato, S.6
Melchiorre, C.7
-
40
-
-
0013640165
-
The binding profile of the novel muscarinic receptor antagonist darifenacin against the five cloned human muscarinic receptors expressed in CHO cells
-
Nunn, P.A., Greengrass, P.M., Newgreen, D.T., Naylor, A.M., Wallis, R.M., 1996. The binding profile of the novel muscarinic receptor antagonist darifenacin against the five cloned human muscarinic receptors expressed in CHO cells. Br. J. Pharmacol. 117 (Suppl.), 130P.
-
(1996)
Br. J. Pharmacol.
, vol.117
, Issue.SUPPL.
-
-
Nunn, P.A.1
Greengrass, P.M.2
Newgreen, D.T.3
Naylor, A.M.4
Wallis, R.M.5
-
41
-
-
0006927211
-
Characterization of muscarinic receptors in guinea-pig gallbladder
-
Oktay, S., Toker, F., Özkutlu, U., Alican, I., Onat, F., Yegen, B.C., Ulusoy, N.B., 1993. Characterization of muscarinic receptors in guinea-pig gallbladder. Life Sci. 52, 579.
-
(1993)
Life Sci.
, vol.52
, pp. 579
-
-
Oktay, S.1
Toker, F.2
Özkutlu, U.3
Alican, I.4
Onat, F.5
Yegen, B.C.6
Ulusoy, N.B.7
-
42
-
-
0028108365
-
Muscarinic receptors in guinea-pig gallbladder
-
Oktay, S., Ulusoy, N.B., Yegen, B.C., 1994. Muscarinic receptors in guinea-pig gallbladder (letter). Gastroenterology 107, 631-632.
-
(1994)
Gastroenterology
, vol.107
, pp. 631-632
-
-
Oktay, S.1
Ulusoy, N.B.2
Yegen, B.C.3
-
43
-
-
0343680276
-
Binding affinity profile of selective muscarinic antagonists in guinea-pig gallbladder
-
Oktay, S., Iskender, E., Onat, F., Yegen, B.C., Ulusoy, N.B., 1995. Binding affinity profile of selective muscarinic antagonists in guinea-pig gallbladder. Life Sci. 56, 1039.
-
(1995)
Life Sci.
, vol.56
, pp. 1039
-
-
Oktay, S.1
Iskender, E.2
Onat, F.3
Yegen, B.C.4
Ulusoy, N.B.5
-
44
-
-
0027246572
-
Are m-cholinoceptors of guinea-pig gallbladder smooth muscle of m4 subtype?
-
Özkutlu, U., Alican, I., Karahan, F., Onat, F., Yegen, B.C., Ulusoy, N.B., Oktay, S., 1993. Are m-cholinoceptors of guinea-pig gallbladder smooth muscle of m4 subtype?. Pharmacology 46, 308-314.
-
(1993)
Pharmacology
, vol.46
, pp. 308-314
-
-
Özkutlu, U.1
Alican, I.2
Karahan, F.3
Onat, F.4
Yegen, B.C.5
Ulusoy, N.B.6
Oktay, S.7
-
45
-
-
0013550718
-
Functional characterization of muscarinic receptors in rat duodenum
-
Pfaff, O., Gross, J., Waelbroeck, M., Mutschler, E., Lambrecht, G., 1995. Functional characterization of muscarinic receptors in rat duodenum. Life Sci. 56, 1038.
-
(1995)
Life Sci.
, vol.56
, pp. 1038
-
-
Pfaff, O.1
Gross, J.2
Waelbroeck, M.3
Mutschler, E.4
Lambrecht, G.5
-
46
-
-
0028108365
-
Muscarinic receptors in guinea-pig gallbladder
-
Von Schrenck, T., 1994. Muscarinic receptors in guinea-pig gallbladder (reply). Gastroenterology 107, 631-632.
-
(1994)
Gastroenterology
, vol.107
, pp. 631-632
-
-
Von Schrenck, T.1
-
47
-
-
0027358768
-
Characterization of muscarinic receptors on guinea-pig gallbladder smooth muscle
-
Von Schrenck, T., Sievers, J., Mirau, S., Raedler, A., Greten, H., 1993. Characterization of muscarinic receptors on guinea-pig gallbladder smooth muscle. Gastroenterology 105, 1341-1349.
-
(1993)
Gastroenterology
, vol.105
, pp. 1341-1349
-
-
Von Schrenck, T.1
Sievers, J.2
Mirau, S.3
Raedler, A.4
Greten, H.5
-
48
-
-
0028264811
-
Signal transduction pathway of the muscarinic receptors mediating gallbladder contraction
-
Von Schrenck, T., Mackensen, B., Mende, U., Schmitz, W., Sievers, J., Mirau, S., Raedler, A., Greten, H., 1994. Signal transduction pathway of the muscarinic receptors mediating gallbladder contraction. Naunyn-Schmiedeberg's Arch. Pharmacol. 349, 346-354.
-
(1994)
Naunyn-Schmiedeberg's Arch. Pharmacol.
, vol.349
, pp. 346-354
-
-
Von Schrenck, T.1
Mackensen, B.2
Mende, U.3
Schmitz, W.4
Sievers, J.5
Mirau, S.6
Raedler, A.7
Greten, H.8
-
50
-
-
0024330294
-
Binding and functional properties of antimuscarinics of the hexocyclium/silahexocyclium and hexahydro-diphenidol/hexahydro-sila-diphenidol type to muscarinic receptor subtypes
-
Waelbroeck, M., Tastenoy, M., Camus, J., Christophe, J., Strohmann, C., Linoh, H., Zilch, H., Tacke, R., Mutschler, E., Lambrecht, G., 1989. Binding and functional properties of antimuscarinics of the hexocyclium/silahexocyclium and hexahydro-diphenidol/hexahydro-sila-diphenidol type to muscarinic receptor subtypes. Br. J. Pharmacol. 98, 197-205.
-
(1989)
Br. J. Pharmacol.
, vol.98
, pp. 197-205
-
-
Waelbroeck, M.1
Tastenoy, M.2
Camus, J.3
Christophe, J.4
Strohmann, C.5
Linoh, H.6
Zilch, H.7
Tacke, R.8
Mutschler, E.9
Lambrecht, G.10
-
52
-
-
0028899016
-
3 receptor antagonists
-
3 receptor antagonists. Life Sci. 56, 861-868.
-
(1995)
Life Sci.
, vol.56
, pp. 861-868
-
-
Wallis, R.M.1
-
53
-
-
0028793587
-
Characterization of the interaction of zamifenacin at muscarinic receptors in vitro
-
Watson, N., Reddy, H., Stefanich, E., Eglen, R.M., 1995. Characterization of the interaction of zamifenacin at muscarinic receptors in vitro. Eur. J. Pharmacol. 285, 135-142.
-
(1995)
Eur. J. Pharmacol.
, vol.285
, pp. 135-142
-
-
Watson, N.1
Reddy, H.2
Stefanich, E.3
Eglen, R.M.4
|