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Volumn 327, Issue 2-3, 1997, Pages 239-246

Overcoming of multidrug resistance by VA-033, a novel derivative of apovincaminic acid ester

Author keywords

Ca2+ current; Chemotherapeutic; P glycoprotein; Verapamil

Indexed keywords

APOVINCAMINIC ACID; AZIDOPINE; DOXORUBICIN; GLYCOPROTEIN P; UNCLASSIFIED DRUG; VA 033; VERAPAMIL; VINCRISTINE;

EID: 16744363513     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(97)89667-7     Document Type: Article
Times cited : (4)

References (24)
  • 1
    • 0021905666 scopus 로고
    • Isolation and genetic characterization of human KB cell lines resistant to multiple drugs
    • Akiyama S., Fojo A., Hanover J.A., Pastan I., Gottesman M.M. Isolation and genetic characterization of human KB cell lines resistant to multiple drugs. Somat. Cell Mol. Genet. 11:1985;117-126.
    • (1985) Somat. Cell Mol. Genet. , vol.11 , pp. 117-126
    • Akiyama, S.1    Fojo, A.2    Hanover, J.A.3    Pastan, I.4    Gottesman, M.M.5
  • 2
    • 0023836456 scopus 로고
    • Most drugs that reverse multidrug resistance also inhibit photoaffinity labeling of P-glycoprotein by a vinblastine analogue
    • Akiyama S., Cornwell M.M., Kuwano M., Pastan I., Gottesman M.M. Most drugs that reverse multidrug resistance also inhibit photoaffinity labeling of P-glycoprotein by a vinblastine analogue. Mol. Pharmacol. 33:1988;144-147.
    • (1988) Mol. Pharmacol. , vol.33 , pp. 144-147
    • Akiyama, S.1    Cornwell, M.M.2    Kuwano, M.3    Pastan, I.4    Gottesman, M.M.5
  • 3
    • 0025562606 scopus 로고
    • Mechanisms of multidrug resistance in human tumor cells; The role of P-glycoprotein, DNA topoisomerase 2 and other factors
    • Beck W.T. Mechanisms of multidrug resistance in human tumor cells; the role of P-glycoprotein, DNA topoisomerase 2 and other factors. Cancer Treat. Rev. 17:1990;11-20.
    • (1990) Cancer Treat. Rev. , vol.17 , pp. 11-20
    • Beck, W.T.1
  • 4
    • 0014767029 scopus 로고
    • Cellular resistance to actinomycin D in Chinese hamster cells in vitro: Cross-resistance, radioautographic and cytogenetic studies
    • Biedler J.L., Riehm H. Cellular resistance to actinomycin D in Chinese hamster cells in vitro: cross-resistance, radioautographic and cytogenetic studies. Cancer Res. 30:1970;1174-1184.
    • (1970) Cancer Res. , vol.30 , pp. 1174-1184
    • Biedler, J.L.1    Riehm, H.2
  • 6
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein dye binding
    • Bradford M.A. A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein dye binding. Anal. Biochem. 72:1976;248-254.
    • (1976) Anal. Biochem. , vol.72 , pp. 248-254
    • Bradford, M.A.1
  • 7
    • 0023130372 scopus 로고
    • Evaluation of a tetrazolium-based semiautomated colorimetric assay: Assessment of chemosensitivity testing
    • Carmichael J., DeGraff W.G., Gazdar A.F., Minna J.D., Mitchell J.B. Evaluation of a tetrazolium-based semiautomated colorimetric assay: assessment of chemosensitivity testing. Cancer Res. 47:1987;943-946.
    • (1987) Cancer Res. , vol.47 , pp. 943-946
    • Carmichael, J.1    Degraff, W.G.2    Gazdar, A.F.3    Minna, J.D.4    Mitchell, J.B.5
  • 8
    • 0022972654 scopus 로고
    • Internal duplication and homology with bacterial transport proteins in the mdr 1 (P-glycoprotein) gene from multidrug-resistant human cells
    • Chen C.-j., Chin J.E., Ueda K., Clark D.P., Pastan I., Gottesman M.M., Roninson I.B. Internal duplication and homology with bacterial transport proteins in the mdr 1 (P-glycoprotein) gene from multidrug-resistant human cells. Cell. 47:1986;381-389.
    • (1986) Cell , vol.47 , pp. 381-389
    • Chen, C.-j.1    Chin, J.E.2    Ueda, K.3    Clark, D.P.4    Pastan, I.5    Gottesman, M.M.6    Roninson, I.B.7
  • 9
    • 0023234519 scopus 로고
    • Certain calcium channel blockers bind specifically to multidrug-resistant human KB carcinoma membrane vesicle and inhibit drug binding to P-glycoprotein
    • Cornwell M.M., Pastan I., Gottesman M.M. Certain calcium channel blockers bind specifically to multidrug-resistant human KB carcinoma membrane vesicle and inhibit drug binding to P-glycoprotein. J. Biol. Chem. 262:1987;2166-2170.
    • (1987) J. Biol. Chem. , vol.262 , pp. 2166-2170
    • Cornwell, M.M.1    Pastan, I.2    Gottesman, M.M.3
  • 10
    • 0024506222 scopus 로고
    • Drug-resistance in multiple myeloma and non-Hodgkin's lymphoma: Detection of P-glycoprotein and potential circumvention by addition of verapamil to chemotherapy
    • Dalton W.S., Grogan T.M., Meltzer P.S., Sheper R.J., Durie B.G., Taylor C.W., Miller T.P., Salmon S.E. Drug-resistance in multiple myeloma and non-Hodgkin's lymphoma: detection of P-glycoprotein and potential circumvention by addition of verapamil to chemotherapy. J. Clin. Oncol. 7:1989;415-424.
    • (1989) J. Clin. Oncol. , vol.7 , pp. 415-424
    • Dalton, W.S.1    Grogan, T.M.2    Meltzer, P.S.3    Sheper, R.J.4    Durie, B.G.5    Taylor, C.W.6    Miller, T.P.7    Salmon, S.E.8
  • 11
    • 0026475310 scopus 로고
    • P-glycoprotein possesses a 1,4-dihydropyridine-selective drug acceptor site which is allosterically coupled to a vinca-alkaloid-selective binding site
    • Ferry D.R., Russell M.A., Cullen M.H. P-glycoprotein possesses a 1,4-dihydropyridine-selective drug acceptor site which is allosterically coupled to a vinca-alkaloid-selective binding site. Biochem. Biophys. Res. Commun. 188:1992;440-445.
    • (1992) Biochem. Biophys. Res. Commun. , vol.188 , pp. 440-445
    • Ferry, D.R.1    Russell, M.A.2    Cullen, M.H.3
  • 12
    • 0020540118 scopus 로고
    • History of calcium antagonist
    • Fleckenstein A. History of calcium antagonist. Circ. Res. 52:1983;I3-I16.
    • (1983) Circ. Res. , vol.52
    • Fleckenstein, A.1
  • 13
    • 0023019651 scopus 로고
    • Homology between P-glycoprotein and a bacterial haemolysin transport protein suggests a model for multidrug resistance
    • Gerlach J.H., Endicott J.A., Juranka P.F., Henderson G., Sarangi F., Deuchars K., Ling V. Homology between P-glycoprotein and a bacterial haemolysin transport protein suggests a model for multidrug resistance. Nature. 324:1986;485-489.
    • (1986) Nature , vol.324 , pp. 485-489
    • Gerlach, J.H.1    Endicott, J.A.2    Juranka, P.F.3    Henderson, G.4    Sarangi, F.5    Deuchars, K.6    Ling, V.7
  • 14
    • 0022993652 scopus 로고
    • Mammalian multidrug-resistance gene: Complete cDNA sequence indicates strong homology to bacterial transport proteins
    • Gros P., Croop J., Housman D. Mammalian multidrug-resistance gene: complete cDNA sequence indicates strong homology to bacterial transport proteins. Cell. 47:1986;371-380.
    • (1986) Cell , vol.47 , pp. 371-380
    • Gros, P.1    Croop, J.2    Housman, D.3
  • 15
    • 0023840065 scopus 로고
    • Purification of the 170- To 180-kilodalton membrane glycoprotein associated with multidrug resistance
    • Hamada H., Tsuruo T. Purification of the 170- to 180-kilodalton membrane glycoprotein associated with multidrug resistance. J. Biol. Chem. 263:1988;1454-1458.
    • (1988) J. Biol. Chem. , vol.263 , pp. 1454-1458
    • Hamada, H.1    Tsuruo, T.2
  • 16
    • 0019827058 scopus 로고
    • Restored in vitro sensitivity of adriamycin and vincristine-resistant P388 leukemia with reserpine
    • Inaba M., Fujikura R., Tsukagoshi S., Sakurai Y. Restored in vitro sensitivity of adriamycin and vincristine-resistant P388 leukemia with reserpine. Biochem. Pharmacol. 30:1981;2191-2194.
    • (1981) Biochem. Pharmacol. , vol.30 , pp. 2191-2194
    • Inaba, M.1    Fujikura, R.2    Tsukagoshi, S.3    Sakurai, Y.4
  • 17
    • 0022381201 scopus 로고
    • On the mechanisms of beta-adrenergic regulation of the Ca channel in the guinea-pig heart
    • Kameyama M., Hofmann F., Trautwein W. On the mechanisms of beta-adrenergic regulation of the Ca channel in the guinea-pig heart. Pflüg. Arch. 405:1985;285-293.
    • (1985) Pflüg. Arch. , vol.405 , pp. 285-293
    • Kameyama, M.1    Hofmann, F.2    Trautwein, W.3
  • 19
    • 0017342653 scopus 로고
    • Active amino acid transport in plasma membrane vesicles from simian virus 40-transformed mouse fibroblasts
    • Lever J.E. Active amino acid transport in plasma membrane vesicles from simian virus 40-transformed mouse fibroblasts. J. Biol. Chem. 252:1977;1990-1997.
    • (1977) J. Biol. Chem. , vol.252 , pp. 1990-1997
    • Lever, J.E.1
  • 20
    • 0026643024 scopus 로고
    • Effect of a dihydropyridine analogue, 2-[benzyl(phenyl)amino]ethyl 1,4-dihydro-2,6-dimethyl-5-(5,5-dimethyl-2-oxo-1,3,2-dioxaphosphorinan-2-yl)-1- (2-morpholino-ethl)-4-(3-nitrophenyl)-3 pyridinecarboxylate on reversing in vivo resistance of tumor cells to adriamycin
    • Niwa K., Yamada K., Furukawa T., Shudo N., Seto K., Matsumoto T., Takao S., Akiyama S., Shimazu H. Effect of a dihydropyridine analogue, 2-[benzyl(phenyl)amino]ethyl 1,4-dihydro-2,6-dimethyl-5-(5,5-dimethyl-2-oxo-1,3,2-dioxaphosphorinan-2-yl)-1- (2-morpholino-ethl)-4-(3-nitrophenyl)-3 pyridinecarboxylate on reversing in vivo resistance of tumor cells to adriamycin. Cancer Res. 52:1992;3655-3660.
    • (1992) Cancer Res. , vol.52 , pp. 3655-3660
    • Niwa, K.1    Yamada, K.2    Furukawa, T.3    Shudo, N.4    Seto, K.5    Matsumoto, T.6    Takao, S.7    Akiyama, S.8    Shimazu, H.9
  • 21
    • 0023226943 scopus 로고
    • Identification of the multidrug resistance-related membrane glycoprotein as an acceptor for calcium channel blocker
    • Safa A.R., Glover C.J., Sewell J.L., Meyers M.B., Biedler J.L., Felsted R.L. Identification of the multidrug resistance-related membrane glycoprotein as an acceptor for calcium channel blocker. J. Biol. Chem. 262:1987;7884-7888.
    • (1987) J. Biol. Chem. , vol.262 , pp. 7884-7888
    • Safa, A.R.1    Glover, C.J.2    Sewell, J.L.3    Meyers, M.B.4    Biedler, J.L.5    Felsted, R.L.6
  • 22
    • 0028597419 scopus 로고
    • Calcium current in rat diabetic ventricular myocytes
    • Tsuchida K., Watajima H., Otomo S. Calcium current in rat diabetic ventricular myocytes. Am. J. Physiol. 367:1994;H2280-H2289.
    • (1994) Am. J. Physiol. , vol.367
    • Tsuchida, K.1    Watajima, H.2    Otomo, S.3
  • 23
    • 0019430432 scopus 로고
    • Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil
    • Tsuruo T., Iida H., Tsukagoshi S., Sakurai Y. Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil. Cancer Res. 41:1981;1967-1972.
    • (1981) Cancer Res. , vol.41 , pp. 1967-1972
    • Tsuruo, T.1    Iida, H.2    Tsukagoshi, S.3    Sakurai, Y.4
  • 24
    • 0021180629 scopus 로고
    • Effects of quinidine and related compounds on cytotoxicity and cellular accumulation of vincristine and adriamycin in drug-resistant tumor cells
    • Tsuruo T., Iida H., Kitatani Y., Yokota K., Tsukagoshi S., Sakurai Y. Effects of quinidine and related compounds on cytotoxicity and cellular accumulation of vincristine and adriamycin in drug-resistant tumor cells. Cancer Res. 44:1984;4303-4307.
    • (1984) Cancer Res. , vol.44 , pp. 4303-4307
    • Tsuruo, T.1    Iida, H.2    Kitatani, Y.3    Yokota, K.4    Tsukagoshi, S.5    Sakurai, Y.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.